Literature DB >> 22473747

A bulky biaryl phosphine ligand allows for palladium-catalyzed amidation of five-membered heterocycles as electrophiles.

Mingjuan Su1, Stephen L Buchwald.   

Abstract

Entities:  

Mesh：

Substances：

Year:  2012        PMID： 22473747      PMCID： PMC3407381          DOI： 10.1002/anie.201201244

Source DB:  PubMed          Journal:  Angew Chem Int Ed Engl        ISSN： 1433-7851            Impact factor:   15.336


× No keyword cloud information.
  23 in total

1.  Discovery of imidazo[1,2-a]pyrazine-based Aurora kinase inhibitors.

Authors:  David B Belanger; Patrick J Curran; Alan Hruza; Johannes Voigt; Zhaoyang Meng; Amit K Mandal; M Arshad Siddiqui; Andrea D Basso; Kimberly Gray
Journal:  Bioorg Med Chem Lett       Date:  2010-07-08       Impact factor: 2.823

2.  Efficient pd-catalyzed amination of heteroaryl halides.

Authors:  Mark D Charles; Phillip Schultz; Stephen L Buchwald
Journal:  Org Lett       Date:  2005-09-01       Impact factor: 6.005

3.  Palladium-catalyzed intermolecular coupling of aryl halides and amides.

Authors:  J Yin; S L Buchwald
Journal:  Org Lett       Date:  2000-04-20       Impact factor: 6.005

4.  Imidazo[1,2-a]pyridin-3-amines as potential HIV-1 non-nucleoside reverse transcriptase inhibitors.

Authors:  Moira L Bode; David Gravestock; Simon S Moleele; Christiaan W van der Westhuyzen; Stephen C Pelly; Paul A Steenkamp; Heinrich C Hoppe; Tasmiyah Khan; Lindiwe A Nkabinde
Journal:  Bioorg Med Chem       Date:  2011-06-21       Impact factor: 3.641

Review 5.  The histamine H3 receptor: from gene cloning to H3 receptor drugs.

Authors:  Rob Leurs; Remko A Bakker; Henk Timmerman; Iwan J P de Esch
Journal:  Nat Rev Drug Discov       Date:  2005-02       Impact factor: 84.694

6.  Discovery of a Potent, Injectable Inhibitor of Aurora Kinases Based on the Imidazo-[1,2-a]-Pyrazine Core.

Authors:  Tao Yu; Jayaram R Tagat; Angela D Kerekes; Ronald J Doll; Yonglian Zhang; Yushi Xiao; Sara Esposite; David B Belanger; Patrick J Curran; Amit K Mandal; M Arshad Siddiqui; Neng-Yang Shih; Andrea D Basso; Ming Liu; Kimberly Gray; Seema Tevar; Jennifer Jones; Suining Lee; Lianzhu Liang; Samad Ponery; Elizabeth B Smith; Alan Hruza; Johannes Voigt; Lata Ramanathan; Winifred Prosise; Mengwei Hu
Journal:  ACS Med Chem Lett       Date:  2010-06-07       Impact factor: 4.345

7.  Imidazo[1,2-b]pyridazines: a potent and selective class of cyclin-dependent kinase inhibitors.

Authors:  Kate F Byth; Nicola Cooper; Janet D Culshaw; David W Heaton; Sandra E Oakes; Claire A Minshull; Richard A Norman; Richard A Pauptit; Julie A Tucker; Jason Breed; Andrew Pannifer; Siân Rowsell; Judith J Stanway; Anna L Valentine; Andrew P Thomas
Journal:  Bioorg Med Chem Lett       Date:  2004-05-03       Impact factor: 2.823

8.  Pd-catalyzed N-arylation of secondary acyclic amides: catalyst development, scope, and computational study.

Authors:  Jacqueline D Hicks; Alan M Hyde; Alberto Martinez Cuezva; Stephen L Buchwald
Journal:  J Am Chem Soc       Date:  2009-11-25       Impact factor: 15.419

9.  An Efficient System For the Pd-Catalyzed Cross-Coupling of Amides and Aryl Chlorides.

Authors:  Brett P Fors; Karin Dooleweerdt; Qingle Zeng; Stephen L Buchwald
Journal:  Tetrahedron       Date:  2009-08-15       Impact factor: 2.457

10.  Highly reactive, general and long-lived catalysts for palladium-catalyzed amination of heteroaryl and aryl chlorides, bromides, and iodides: scope and structure-activity relationships.

Authors:  Qilong Shen; Tokutaro Ogata; John F Hartwig
Journal:  J Am Chem Soc       Date:  2008-04-30       Impact factor: 15.419
View more
  25 in total

1.  Metallaphotoredox Difluoromethylation of Aryl Bromides.

Authors:  Vlad Bacauanu; Sébastien Cardinal; Motoshi Yamauchi; Masaru Kondo; David F Fernández; Richard Remy; David W C MacMillan
Journal:  Angew Chem Int Ed Engl       Date:  2018-08-28       Impact factor: 15.336

2.  Structure and Reactivity of [(L•Pd)n•(1,5-cyclooctadiene)] (n=1-2) Complexes Bearing Biaryl Phosphine Ligands.

Authors:  Hong Geun Lee; Phillip J Milner; Michael T Colvin; Loren Andreas; Stephen L Buchwald
Journal:  Inorganica Chim Acta       Date:  2014-10-01       Impact factor: 2.545

3.  Mild and general palladium-catalyzed synthesis of methyl aryl ethers enabled by the use of a palladacycle precatalyst.

Authors:  Chi Wai Cheung; Stephen L Buchwald
Journal:  Org Lett       Date:  2013-07-24       Impact factor: 6.005

4.  Suzuki-Miyaura cross-coupling of unprotected, nitrogen-rich heterocycles: substrate scope and mechanistic investigation.

Authors:  M Alexander Düfert; Kelvin L Billingsley; Stephen L Buchwald
Journal:  J Am Chem Soc       Date:  2013-08-16       Impact factor: 15.419

5.  A Metallaphotoredox Strategy for the Cross-Electrophile Coupling of α-Chloro Carbonyls with Aryl Halides.

Authors:  Tiffany Q Chen; David W C MacMillan
Journal:  Angew Chem Int Ed Engl       Date:  2019-09-05       Impact factor: 15.336

6.  Investigating the dearomative rearrangement of biaryl phosphine-ligated Pd(II) complexes.

Authors:  Phillip J Milner; Thomas J Maimone; Mingjuan Su; Jiahao Chen; Peter Müller; Stephen L Buchwald
Journal:  J Am Chem Soc       Date:  2012-11-27       Impact factor: 15.419

7.  Synthesis and application of palladium precatalysts that accommodate extremely bulky di-tert-butylphosphino biaryl ligands.

Authors:  Nicholas C Bruno; Stephen L Buchwald
Journal:  Org Lett       Date:  2013-05-15       Impact factor: 6.005

8.  Mild and highly selective palladium-catalyzed monoarylation of ammonia enabled by the use of bulky biarylphosphine ligands and palladacycle precatalysts.

Authors:  Chi Wai Cheung; David S Surry; Stephen L Buchwald
Journal:  Org Lett       Date:  2013-07-01       Impact factor: 6.005

9.  Silyl Radical Activation of Alkyl Halides in Metallaphotoredox Catalysis: A Unique Pathway for Cross-Electrophile Coupling.

Authors:  Patricia Zhang; Chi Chip Le; David W C MacMillan
Journal:  J Am Chem Soc       Date:  2016-06-22       Impact factor: 15.419

Review 10.  Applications of Palladium-Catalyzed C-N Cross-Coupling Reactions.

Authors:  Paula Ruiz-Castillo; Stephen L Buchwald
Journal:  Chem Rev       Date:  2016-09-30       Impact factor: 60.622
View more

北京卡尤迪生物科技股份有限公司 © 2022-2023.