Literature DB >> 22419258

Comparison of open-flow microperfusion and microdialysis methodologies when sampling topically applied fentanyl and benzoic acid in human dermis ex vivo.

R Holmgaard1, E Benfeldt, J B Nielsen, C Gatschelhofer, J A Sorensen, C Höfferer, M Bodenlenz, T R Pieber, F Sinner.   

Abstract

PURPOSE: The purpose of this study is to compare two sampling methods--dermal Open-Flow Microperfusion (dOFM) and dermal Microdialysis (dMD) in an international joint experiment in a single-laboratory setting. We used human ex-vivo skin and sampled topically administered Fentanyl and Benzoic Acid. The second purpose was to provide guidance to researchers in choosing the most efficient method for a given penetrant and give suggestions concerning critical choices for successful dermal sampling.
METHODS: The dOFM and dMD techniques are compared in equal set-ups using three probe-types (one dOFM probe and two dMD probe-types) in donor skin (n = 9)--27 probes of each type sampling each penetrant in solutions applied in penetrationchambers glued to the skin surface over a time range of 20 h.
RESULTS: Pharmacokinetic results demonstrated concordance between dOFM and dMD sampling technique under the given experimental conditions. The methods each had advantages and limitations in technical, practical and hands-on comparisons.
CONCLUSION: When planning a study of cutaneous penetration the advantages and limitations of each probe-type have to be considered in relation to the scientific question posed, the physico-chemical characteristics of the substance of interest, the choice of experimental setting e.g. ex vivo/in vivo and the analytical skills available.

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Year:  2012        PMID: 22419258     DOI: 10.1007/s11095-012-0705-9

Source DB:  PubMed          Journal:  Pharm Res        ISSN: 0724-8741            Impact factor:   4.200


  37 in total

Review 1.  Microdialysis sampling for investigations of bioavailability and bioequivalence of topically administered drugs: current state and future perspectives.

Authors:  R Holmgaard; J B Nielsen; E Benfeldt
Journal:  Skin Pharmacol Physiol       Date:  2010-05-18       Impact factor: 3.479

2.  Efficacy of skin wash on dermal absorption: an in vitro study on four model compounds of varying solubility.

Authors:  Jesper Bo Nielsen
Journal:  Int Arch Occup Environ Health       Date:  2010-05-26       Impact factor: 3.015

3.  Percutaneous penetration through slightly damaged skin.

Authors:  Jesper B Nielsen
Journal:  Arch Dermatol Res       Date:  2005-04-15       Impact factor: 3.017

Review 4.  Microdialysis of large molecules.

Authors:  Geraldine F Clough
Journal:  AAPS J       Date:  2005-10-26       Impact factor: 4.009

5.  Microdialysis of lipophilic compounds: a methodological study.

Authors:  C Carneheim; L Ståhle
Journal:  Pharmacol Toxicol       Date:  1991-11

Review 6.  Transdermal drug delivery and cutaneous metabolism.

Authors:  R H Guy; J Hadgraft; D A Bucks
Journal:  Xenobiotica       Date:  1987-03       Impact factor: 1.908

7.  Measurement of interstitial insulin in human adipose and muscle tissue under moderate hyperinsulinemia by means of direct interstitial access.

Authors:  Manfred Bodenlenz; Lukas A Schaupp; Tatjana Druml; Romana Sommer; Andrea Wutte; Helga C Schaller; Frank Sinner; Paul Wach; Thomas R Pieber
Journal:  Am J Physiol Endocrinol Metab       Date:  2005-03-15       Impact factor: 4.310

8.  Transdermal fentanyl for the treatment of pain caused by rheumatoid arthritis.

Authors:  Gabriel Herrero-Beaumont; Olav Bjorneboe; Ute Richarz
Journal:  Rheumatol Int       Date:  2004-10-05       Impact factor: 2.631

9.  The usual suspects-influence of physicochemical properties on lag time, skin deposition, and percutaneous penetration of nine model compounds.

Authors:  Jesper Bo Nielsen; Jens Ahm Sørensen; Flemming Nielsen
Journal:  J Toxicol Environ Health A       Date:  2009

10.  Transdermal fentanyl for the treatment of back pain caused by vertebral osteoporosis.

Authors:  J D Ringe; H Faber; O Bock; S Valentine; D Felsenberg; M Pfeifer; H W Minne; S Schwalen
Journal:  Rheumatol Int       Date:  2002-07-10       Impact factor: 2.631

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  4 in total

1.  Kinetics of Clobetasol-17-Propionate in Psoriatic Lesional and Non-Lesional Skin Assessed by Dermal Open Flow Microperfusion with Time and Space Resolution.

Authors:  Manfred Bodenlenz; Christian Dragatin; Lisa Liebenberger; Bernd Tschapeller; Beate Boulgaropoulos; Thomas Augustin; Reingard Raml; Christina Gatschelhofer; Nathalie Wagner; Khaled Benkali; Francois Rony; Thomas Pieber; Frank Sinner
Journal:  Pharm Res       Date:  2016-06-06       Impact factor: 4.200

2.  The Impact of Prolonged Inflammation on Wound Healing.

Authors:  Judith C J Holzer-Geissler; Simon Schwingenschuh; Martin Zacharias; Johanna Einsiedler; Sonja Kainz; Peter Reisenegger; Christian Holecek; Elisabeth Hofmann; Barbara Wolff-Winiski; Hermann Fahrngruber; Thomas Birngruber; Lars-Peter Kamolz; Petra Kotzbeck
Journal:  Biomedicines       Date:  2022-04-06

3.  The Skin Reservoir Model: A Tool for Evaluating Microdialysis Sampling of Large Biomarkers from Human Skin.

Authors:  Katrine Baumann; Sidsel Falkencrone; Niels Peter Knudsen; Anders Woetmann; Sally Dabelsteen; Per Stahl Skov
Journal:  Acta Derm Venereol       Date:  2020-01-07       Impact factor: 3.875

4.  Long-term implanted cOFM probe causes minimal tissue reaction in the brain.

Authors:  Thomas Birngruber; Arijit Ghosh; Sonja Hochmeister; Martin Asslaber; Thomas Kroath; Thomas R Pieber; Frank Sinner
Journal:  PLoS One       Date:  2014-03-12       Impact factor: 3.240

  4 in total

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