Literature DB >> 22205617

Early effects of oral administration of omeprazole and roxatidine on intragastric pH.

Hiroshi Iida1, Shingo Kato, Yusuke Sekino, Eiji Sakai, Takashi Uchiyama, Hiroki Endo, Kunihiro Hosono, Yasunari Sakamoto, Koji Fujita, Masato Yoneda, Tomoko Koide, Hirokazu Takahashi, Chikako Tokoro, Ayumu Goto, Yasunobu Abe, Noritoshi Kobayashi, Kensuke Kubota, Eiji Gotoh, Shin Maeda, Atsushi Nakajima, Masahiko Inamori.   

Abstract

OBJECTIVE: The ideal medication for the treatment of acid-related diseases, e.g., peptic ulcers, stress-related gastric bleeding, functional dyspepsia, and gastroesophageal reflux disease, should have a rapid onset of action to promote hemostasis and relieve the symptoms. The aim of our study was to investigate the inhibitory effects on gastric acid secretion of a single oral administration of a proton pump inhibitor, omeprazole 20 mg, and an H(2)-receptor antagonist, roxatidine 75 mg.
METHODS: Ten Helicobacter pylori-negative male subjects participated in this randomized, two-way crossover study. Intragastric pH was monitored continuously for 6 h after single oral administration of omeprazole 20 mg and roxatidine 75 mg. Each administration was separated by a 7-d washout period.
RESULTS: During the 6-h study period, the average pH after administration of roxatidine was higher than that after administration of omeprazole (median: 4.45 vs. 2.65; P=0.0367). Also during the 6-h study period, a longer duration of maintenance at pH above 2, 5, and 6 was observed after administration of roxatidine 75 mg than after administration of omeprazole 20 mg (median: 90.6% vs. 55.2%, P=0.0284; 43.7% vs. 10.6%, P=0.0125; 40.3% vs. 3.3%, P=0.0125; respectively).
CONCLUSIONS: In Helicobacter pylori-negative healthy male subjects, oral administration of roxatidine 75 mg increased the intragastric pH more rapidly than that of omeprazole 20 mg.

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Year:  2012        PMID: 22205617      PMCID: PMC3251749          DOI: 10.1631/jzus.B1100078

Source DB:  PubMed          Journal:  J Zhejiang Univ Sci B        ISSN: 1673-1581            Impact factor:   3.066


  32 in total

1.  Early effects of intravenous administrations of lansoprazole and famotidine on intragastric pH.

Authors:  Hiroshi Iida; Masahiko Inamori; Keiko Akimoto; Hironori Mawatari; Hiroki Endo; Yuichi Nozaki; Tomoyuki Akiyama; Tamon Ikeda; Yasunari Sakamoto; Koji Fujita; Kyoko Yoneda; Hirokazu Takahashi; Masato Yoneda; Ayumu Goto; Yasunobu Abe; Noritoshi Kobayashi; Hiroyuki Kirikoshi; Kensuke Kubota; Satoru Saito; Atsushi Nakajima
Journal:  Hepatogastroenterology       Date:  2009 Mar-Apr

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Authors:  F W Green; M M Kaplan; L E Curtis; P H Levine
Journal:  Gastroenterology       Date:  1978-01       Impact factor: 22.682

3.  Effect of single and repeated intravenous doses of omeprazole on pentagastrin stimulated gastric acid secretion and pharmacokinetics in man.

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Journal:  Gut       Date:  1988-01       Impact factor: 23.059

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Authors:  S Ohara; M Hongo; S Asaki; A Sato; D Shibuya; H Sato; T Motojima; N Yamaguchi; T Ohara; T Tamura
Journal:  Nihon Shokakibyo Gakkai Zasshi       Date:  1988-07

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Journal:  Gut       Date:  1984-07       Impact factor: 23.059

7.  Histamine H2-receptor antagonistic action of N-(3-[3-(1-piperidinylmethyl)phenoxy]propyl)acetoxyacetamide hydrochloride (TZU-0460).

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Journal:  Am J Surg       Date:  1980-12       Impact factor: 2.565

9.  Effects of rabeprazole, lansoprazole and omeprazole on intragastric pH in CYP2C19 extensive metabolizers.

Authors:  T Saitoh; Y Fukushima; H Otsuka; J Hirakawa; H Mori; T Asano; T Ishikawa; T Katsube; K Ogawa; S Ohkawa
Journal:  Aliment Pharmacol Ther       Date:  2002-10       Impact factor: 8.171

10.  Mephenytoin hydroxylation deficiency in Caucasians: frequency of a new oxidative drug metabolism polymorphism.

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Journal:  Clin Pharmacol Ther       Date:  1984-12       Impact factor: 6.875

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  1 in total

1.  Relative bioavailability and pharmacokinetic comparison of two different enteric formulations of omeprazole.

Authors:  Jian Liu; Jian-zhong Shentu; Li-hua Wu; Jing Dou; Qi-yang Xu; Hui-li Zhou; Guo-lan Wu; Ming-zhu Huang; Xing-jiang Hu; Jun-chun Chen
Journal:  J Zhejiang Univ Sci B       Date:  2012-05       Impact factor: 3.066

  1 in total

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