Literature DB >> 22180523

Examination of noninferiority, safety, and tolerability of lopinavir/ritonavir and raltegravir compared with lopinavir/ritonavir and tenofovir/ emtricitabine in antiretroviral-naïve subjects: the progress study, 48-week results.

Jacques Reynes1, Adebayo Lawal, Federico Pulido, Ruth Soto-Malave, Joseph Gathe, Min Tian, Linda M Fredrick, Thomas J Podsadecki, Angela M Nilius.   

Abstract

PURPOSE: Current antiretroviral regimens recommended for treatment-naïve patients include 2 nucleoside/nucleotide reverse transcriptase inhibitors (NRTIs). The purpose of this study is to evaluate whether a new NRTI-sparing regimen may provide an alternative for persons for whom traditional regimens may not be the best option.
METHODS: PROGRESS is a 96-week, randomized, open-label, multicenter trial comparing the efficacy and safety of a boosted protease inhibitor (PI) and an integrase inhibitor (lopi-navir/ritonavir [LPV/r] + raltegravir [RAL]) to a boosted PI and 2 NRTIs (LPV/r + tenofovir/ emtricitabine [TDF/FTC]) in antiretroviral (ARV)-naïve HIV-1-infected adults.
RESULTS: A total of 206 subjects were randomized to receive LPV/r + RAL (n=101) or LPV/r + TDF/FTC (n=105) and analyzed for ARV efficacy using the US Food and Drug Administration time to loss of virologic response (FDA-TLOVR) algorithm. The percentage of subjects with plasma HIV-1 RNA <40 copies/mL at week 48 was 83.2% in the LPV/r + RAL group and 84.8% in the LPV/r + TDF/FTC group (P = .850; difference -1.6%; exact 95% CI, -12.0% to 8.8%). As the lower limit of the exact 95% CI for the difference between regimens was at or above the protocol-defined threshold of -20% (as well as the more stringent threshold of -12%), LPV/r + RAL was noninferior to LPV/r + TDF/FTC. The occurrence of treatment-related, moderate/severe adverse events was similar between treatment groups through 48 weeks of treatment.
CONCLUSIONS: The HIV treatment regimen of LPV/r + RAL resulted in noninferior efficacy and comparable safety and tolerability compared with a traditional NRTI-containing regimen through 48 weeks of treatment. These results support further evaluation of the LPV/r + RAL regimen.

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Year:  2011        PMID: 22180523     DOI: 10.1310/hct1205-255

Source DB:  PubMed          Journal:  HIV Clin Trials        ISSN: 1528-4336


  17 in total

1.  Addition of E138K to R263K in HIV integrase increases resistance to dolutegravir, but fails to restore activity of the HIV integrase enzyme and viral replication capacity.

Authors:  Thibault Mesplède; Nathan Osman; Melissa Wares; Peter K Quashie; Said Hassounah; Kaitlin Anstett; Yingshan Han; Diane N Singhroy; Mark A Wainberg
Journal:  J Antimicrob Chemother       Date:  2014-06-10       Impact factor: 5.790

2.  HIV viral kinetics and T cell dynamics in antiretroviral naïve persons starting an integrase strand transfer inhibitor and protease inhibitor regimen.

Authors:  Maile Y Karris; Sonia Jain; Tyler R C Day; Josué Pérez-Santiago; Miguel Goicoechea; Michael P Dubé; Xiaoying Sun; Celsa Spina; Eric S Daar; Richard H Haubrich; Sheldon Morris
Journal:  HIV Clin Trials       Date:  2017-01-30

3.  Clinical practice guideline for the management of chronic kidney disease in patients infected with HIV: 2014 update by the HIV Medicine Association of the Infectious Diseases Society of America.

Authors:  Gregory M Lucas; Michael J Ross; Peter G Stock; Michael G Shlipak; Christina M Wyatt; Samir K Gupta; Mohamed G Atta; Kara K Wools-Kaloustian; Paul A Pham; Leslie A Bruggeman; Jeffrey L Lennox; Patricio E Ray; Robert C Kalayjian
Journal:  Clin Infect Dis       Date:  2014-09-17       Impact factor: 9.079

4.  Combination antiretroviral therapy with raltegravir leads to rapid immunologic reconstitution in treatment-naive patients with chronic HIV infection.

Authors:  Suresh Pallikkuth; Margaret A Fischl; Savita Pahwa
Journal:  J Infect Dis       Date:  2013-08-06       Impact factor: 5.226

Review 5.  Use of Integrase Inhibitors in HIV-Infected Children and Adolescents.

Authors:  Walter Dehority; Jacobo Abadi; Andrew Wiznia; Rolando M Viani
Journal:  Drugs       Date:  2015-09       Impact factor: 9.546

6.  NRTI backbone in HIV treatment: will it remain relevant?

Authors:  Randall Tressler; Catherine Godfrey
Journal:  Drugs       Date:  2012-11-12       Impact factor: 9.546

7.  HIV lipodystrophy in participants randomised to lopinavir/ritonavir (LPV/r) +2-3 nucleoside/nucleotide reverse transcriptase inhibitors (N(t)RTI) or LPV/r + raltegravir as second-line antiretroviral therapy.

Authors:  Allison Martin; Cecilia L Moore; Patrick W G Mallon; Jennifer F Hoy; Sean Emery; Waldo H Belloso; Praphan Phanuphak; Samuel Ferret; David A Cooper; Mark A Boyd
Journal:  PLoS One       Date:  2013-10-30       Impact factor: 3.240

Review 8.  Clinical use of HIV integrase inhibitors: a systematic review and meta-analysis.

Authors:  Peter Messiaen; Annemarie M J Wensing; Axel Fun; Monique Nijhuis; Nele Brusselaers; Linos Vandekerckhove
Journal:  PLoS One       Date:  2013-01-09       Impact factor: 3.240

9.  The potential cost and benefits of raltegravir in simplified second-line therapy among HIV infected patients in Nigeria and South Africa.

Authors:  Karen Schneider; Chidi Nwizu; Richard Kaplan; Jonathan Anderson; David P Wilson; Sean Emery; David A Cooper; Mark A Boyd
Journal:  PLoS One       Date:  2013-02-15       Impact factor: 3.240

10.  Nucleoside-sparing antiretroviral regimens.

Authors:  Pola de la Torre; Jomy George; John D Baxter
Journal:  Curr Infect Dis Rep       Date:  2014-07       Impact factor: 3.663

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