Literature DB >> 21681118

Low-dose gefitinib treatment for patients with advanced non-small cell lung cancer harboring sensitive epidermal growth factor receptor mutations.

Hironori Satoh1, Akira Inoue, Kunihiko Kobayashi, Makoto Maemondo, Satoshi Oizumi, Hiroshi Isobe, Akihiko Gemma, Yasuo Saijo, Hirohisa Yoshizawa, Koichi Hagiwara, Toshihiro Nukiwa.   

Abstract

INTRODUCTION: Although standard schedule of gefitinib was the administration of 250 mg tablet every day, many patients need dose reduction because of toxicities. However, the efficacy of such low-dose gefitinib for patients with epidermal growth factor receptor-mutated non-small cell lung cancer has rarely been evaluated.
METHODS: A post hoc comparison of the efficacy (response rate and survival) in patients treated with gefitinib with or without any dose reduction in NEJ002 study was performed.
RESULTS: Among 114 patients treated with first-line gefitinib in NEJ002, 61 (54%) continued gefitinib without any dose reduction until their diseases progressed, and 53 (46%) reduced their dose of gefitinib because of some toxicities. There was no significant difference of patient characteristics between the two groups. The progression-free survival of low-dose group tended to be better than that of standard-dose group (median progression-free survival, 11.8 versus 9.9 months; p = 0.144), and the overall survival of low-dose group was also better than that of standard-dose group (median survival time, 32.7 versus 25.3 months; p = 0.049).
CONCLUSIONS: The results suggest that low-dose gefitinib may be clinically not inferior to standard-dose gefitinib for non-small cell lung cancer with sensitive epidermal growth factor receptor mutations. Prospective study of low-dose gefitinib is warranted especially for frail patients who need less toxic treatment.

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Year:  2011        PMID: 21681118     DOI: 10.1097/JTO.0b013e31821d43a8

Source DB:  PubMed          Journal:  J Thorac Oncol        ISSN: 1556-0864            Impact factor:   15.609


  20 in total

1.  Phase 1 study of twice weekly pulse dose and daily low-dose erlotinib as initial treatment for patients with EGFR-mutant lung cancers.

Authors:  H A Yu; C Sima; D Feldman; L L Liu; B Vaitheesvaran; J Cross; C M Rudin; M G Kris; W Pao; F Michor; G J Riely
Journal:  Ann Oncol       Date:  2017-02-01       Impact factor: 32.976

2.  Gefitinib frequently induces liver damage in patients with lung adenocarcinoma previously treated by chemotherapy.

Authors:  Yasoo Sugiura; Etsuo Nemoto; Osamu Kawai; Yasuyuki Ohkubo; Hisae Fusegawa; Shizuka Kaseda
Journal:  Lung Cancer (Auckl)       Date:  2013-06-08

3.  Epidermal growth factor receptor-tyrosine kinase inhibitors for non-small-cell lung cancer patients aged 80 years or older: A retrospective analysis.

Authors:  Makoto Nakao; Hideki Muramatsu; Kazuki Sone; Sachiko Aoki; Harata Akiko; Yusuke Kagawa; Hidefumi Sato; Takefumi Kunieda
Journal:  Mol Clin Oncol       Date:  2014-11-05

4.  Gefitinib treatment in patients with postoperative recurrent non-small-cell lung cancer harboring epidermal growth factor receptor gene mutations.

Authors:  Yuhei Yokoyama; Makoto Sonobe; Tetsu Yamada; Masaaki Sato; Toshi Menju; Akihiro Aoyama; Toshihiko Sato; Fengshi Chen; Mitsugu Omasa; Hiroshi Date
Journal:  Int J Clin Oncol       Date:  2015-05-08       Impact factor: 3.402

Review 5.  Optimized Dosing: The Next Step in Precision Medicine in Non-Small-Cell Lung Cancer.

Authors:  René J Boosman; Jacobus A Burgers; Egbert F Smit; Neeltje Steeghs; Anthonie J van der Wekken; Jos H Beijnen; Alwin D R Huitema; Rob Ter Heine
Journal:  Drugs       Date:  2021-12-11       Impact factor: 9.546

6.  Rational application of gefitinib in NSCLC patients with sensitive EGFR mutations based on pharmacokinetics and metabolomics.

Authors:  Wei Feng; Xi Chen; Shao-Xing Guan; Hong-Lian Ruan; Yan Huang; Hui-Zhen Zhang; Yun-Peng Yang; Wen-Feng Fang; Hong-Yun Zhao; Wei Zhuang; Shuang Xin; You-Hao Chen; Fei Wang; Yue Gao; Min Huang; Xue-Ding Wang; Li Zhang
Journal:  Acta Pharmacol Sin       Date:  2021-11-04       Impact factor: 7.169

7.  Evaluation of gefitinib systemic exposure in EGFR-mutated non-small cell lung cancer patients with gefitinib-induced severe hepatotoxicity.

Authors:  Takahisa Kawamura; Chiyo K Imamura; Hirotsugu Kenmotsu; Tetsuhiko Taira; Shota Omori; Kazuhisa Nakashima; Kazushige Wakuda; Akira Ono; Tateaki Naito; Haruyasu Murakami; Taisei Mushiroda; Toshiaki Takahashi; Yusuke Tanigawara
Journal:  Cancer Chemother Pharmacol       Date:  2020-02-10       Impact factor: 3.333

8.  First-line treatment of advanced epidermal growth factor receptor (EGFR) mutation positive non-squamous non-small cell lung cancer.

Authors:  Janette Greenhalgh; Angela Boland; Victoria Bates; Fabio Vecchio; Yenal Dundar; Marty Chaplin; John A Green
Journal:  Cochrane Database Syst Rev       Date:  2021-03-18

9.  Successful erlotinib treatment for a patient with gefitinib-related hepatotoxicity and lung adenocarcinoma refractory to intermittently administered gefitinib.

Authors:  Tatsuya Nagano; Yoshikazu Kotani; Kazuyuki Kobayashi; Masahiro Katsurada; Yukihisa Hatakeyama; Suya Hori; Daisuke Tamura; Daisuke Kasai; Yasuhiro Funada; Yoshihiro Nishimura
Journal:  Case Rep Pulmonol       Date:  2011-12-25

10.  The gefitinib dose reduction on survival outcomes in epidermal growth factor receptor mutant non-small cell lung cancer.

Authors:  Sung Hoon Sim; Bhumsuk Keam; Dong-Wan Kim; Tae Min Kim; Se-Hoon Lee; Doo Hyun Chung; Dae Seog Heo
Journal:  J Cancer Res Clin Oncol       Date:  2014-07-09       Impact factor: 4.322

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