Literature DB >> 20973023

Glucosamine-6-sulfamate analogues of heparan sulfate as inhibitors of endosulfatases.

Mathias Schelwies1, Diana Brinson, Shuhei Otsuki, Young-Hoon Hong, Martin K Lotz, Chi-Huey Wong, Sarah R Hanson.   

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Year:  2010        PMID： 20973023      PMCID： PMC3086843          DOI： 10.1002/cbic.201000401

Source DB:  PubMed          Journal:  Chembiochem        ISSN： 1439-4227            Impact factor:   3.164


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  29 in total

1.  Synthesis and structure-activity relationships of truncated bisubstrate inhibitors of aminoglycoside 6'-N-acetyltransferases.

Authors:  Feng Gao; Xuxu Yan; Tushar Shakya; Oliver M Baettig; Samia Ait-Mohand-Brunet; Albert M Berghuis; Gerard D Wright; Karine Auclair
Journal:  J Med Chem       Date:  2006-08-24       Impact factor: 7.446

2.  Substrate specificity and domain functions of extracellular heparan sulfate 6-O-endosulfatases, QSulf1 and QSulf2.

Authors:  Xingbin Ai; Anh-Tri Do; Marion Kusche-Gullberg; Ulf Lindahl; Ke Lu; Charles P Emerson
Journal:  J Biol Chem       Date:  2005-12-23       Impact factor: 5.157

3.  Synthesis and evaluation of general mechanism-based inhibitors of sulfatases based on (difluoro)methyl phenyl sulfate and cyclic phenyl sulfamate motifs.

Authors:  Sarah R Hanson; Lisa J Whalen; Chi-Huey Wong
Journal:  Bioorg Med Chem       Date:  2006-10-11       Impact factor: 3.641

4.  Steroidal and nonsteroidal sulfamates as potent inhibitors of steroid sulfatase.

Authors:  L W Woo; N M Howarth; A Purohit; H A Hejaz; M J Reed; B V Potter
Journal:  J Med Chem       Date:  1998-03-26       Impact factor: 7.446

5.  Heparan sulfate 6-O-endosulfatases: discrete in vivo activities and functional co-operativity.

Authors:  William C Lamanna; Rebecca J Baldwin; Michael Padva; Ina Kalus; Gerdy Ten Dam; Toin H van Kuppevelt; John T Gallagher; Kurt von Figura; Thomas Dierks; Catherine L R Merry
Journal:  Biochem J       Date:  2006-11-15       Impact factor: 3.857

6.  Hsulf-1 regulates growth and invasion of pancreatic cancer cells.

Authors:  I Abiatari; J Kleeff; J Li; K Felix; M W Büchler; H Friess
Journal:  J Clin Pathol       Date:  2006-04-07       Impact factor: 3.411

Review 7.  Sulfatases: structure, mechanism, biological activity, inhibition, and synthetic utility.

Authors:  Sarah R Hanson; Michael D Best; Chi-Huey Wong
Journal:  Angew Chem Int Ed Engl       Date:  2004-11-05       Impact factor: 15.336

Review 8.  Human sulfatases: a structural perspective to catalysis.

Authors:  D Ghosh
Journal:  Cell Mol Life Sci       Date:  2007-08       Impact factor: 9.261

9.  Extracellular sulfatases, elements of the Wnt signaling pathway, positively regulate growth and tumorigenicity of human pancreatic cancer cells.

Authors:  Roman Nawroth; Annemieke van Zante; Sara Cervantes; Michael McManus; Matthias Hebrok; Steven D Rosen
Journal:  PLoS One       Date:  2007-04-25       Impact factor: 3.240

10.  Secreted sulfatases Sulf1 and Sulf2 have overlapping yet essential roles in mouse neonatal survival.

Authors:  Charles R Holst; Hani Bou-Reslan; Bryan B Gore; Karen Wong; Deanna Grant; Sreedevi Chalasani; Richard A Carano; Gretchen D Frantz; Marc Tessier-Lavigne; Brad Bolon; Dorothy M French; Avi Ashkenazi
Journal:  PLoS One       Date:  2007-06-27       Impact factor: 3.240
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  9 in total

Review 1.  Intestinal epithelial glycosylation in homeostasis and gut microbiota interactions in IBD.

Authors:  Matthew R Kudelka; Sean R Stowell; Richard D Cummings; Andrew S Neish
Journal:  Nat Rev Gastroenterol Hepatol       Date:  2020-07-24       Impact factor: 46.802

2.  The role of DNA methylation and histone modifications in blood pressure: a systematic review.

Authors:  Valentina Gonzalez-Jaramillo; Eliana Portilla-Fernandez; Marija Glisic; Trudy Voortman; Wichor Bramer; Rajiv Chowdhury; Anton J M Roks; A H Jan Danser; Taulant Muka; Jana Nano; Oscar H Franco
Journal:  J Hum Hypertens       Date:  2019-07-25       Impact factor: 3.012

Review 3.  Modifications of glycans: biological significance and therapeutic opportunities.

Authors:  Saddam M Muthana; Christopher T Campbell; Jeffrey C Gildersleeve
Journal:  ACS Chem Biol       Date:  2012-01-11       Impact factor: 5.100

4.  Sulfatase-activated fluorophores for rapid discrimination of mycobacterial species and strains.

Authors:  Kimberly E Beatty; Monique Williams; Brian L Carlson; Benjamin M Swarts; Robin M Warren; Paul D van Helden; Carolyn R Bertozzi
Journal:  Proc Natl Acad Sci U S A       Date:  2013-07-22       Impact factor: 11.205

5.  The human sulfatase 2 inhibitor 2,4-disulfonylphenyl-tert-butylnitrone (OKN-007) has an antitumor effect in hepatocellular carcinoma mediated via suppression of TGFB1/SMAD2 and Hedgehog/GLI1 signaling.

Authors:  Xin Zheng; Xiaohong Gai; Shaoshan Han; Catherine D Moser; Chunling Hu; Abdirashid M Shire; Robert A Floyd; Lewis R Roberts
Journal:  Genes Chromosomes Cancer       Date:  2012-10-29       Impact factor: 5.006

Review 6.  Post-Synthetic Regulation of HS Structure: The Yin and Yang of the Sulfs in Cancer.

Authors:  Romain R Vivès; Amal Seffouh; Hugues Lortat-Jacob
Journal:  Front Oncol       Date:  2014-01-14       Impact factor: 6.244

7.  Design and synthesis of biphenyl and biphenyl ether inhibitors of sulfatases.

Authors:  Tristan Reuillon; Sari F Alhasan; Gary S Beale; Annalisa Bertoli; Alfie Brennan; Celine Cano; Helen L Reeves; David R Newell; Bernard T Golding; Duncan C Miller; Roger J Griffin
Journal:  Chem Sci       Date:  2016-01-11       Impact factor: 9.825

8.  MYCN-dependent expression of sulfatase-2 regulates neuroblastoma cell survival.

Authors:  Valeria Solari; Lucia Borriello; Gianluca Turcatel; Hiroyuki Shimada; Richard Sposto; G Esteban Fernandez; Shahab Asgharzadeh; Edwin A Yates; Jeremy E Turnbull; Yves A DeClerck
Journal:  Cancer Res       Date:  2014-08-27       Impact factor: 12.701

9.  Sulfatase-2: a prognostic biomarker and candidate therapeutic target in patients with pancreatic ductal adenocarcinoma.

Authors:  Sari F Alhasan; Beate Haugk; Laura F Ogle; Gary S Beale; Anna Long; Alastair D Burt; Dina Tiniakos; Despina Televantou; Fareeda Coxon; David R Newell; Richard Charnley; Helen L Reeves
Journal:  Br J Cancer       Date:  2016-08-25       Impact factor: 7.640
  9 in total

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