Literature DB >> 20922806

Overexpression of receptor tyrosine kinase Axl promotes tumor cell invasion and survival in pancreatic ductal adenocarcinoma.

Xianzhou Song1, Hua Wang, Craig D Logsdon, Asif Rashid, Jason B Fleming, James L Abbruzzese, Henry F Gomez, Douglas B Evans, Huamin Wang.   

Abstract

BACKGROUND: The receptor tyrosine kinase Axl has been reported to be overexpressed in a variety of human cancers. Although previous studies have identified the role of Axl in the transformation, proliferation, survival, and invasion in cancers, the expression and functions of Axl in pancreatic cancer have not been studied in detail.
METHODS: The expression of Axl protein in 12 pancreatic cancer cell lines and 54 patient samples of stage II pancreatic ductal adenocarcinoma (PDA) and their paired non-neoplastic pancreatic tissue samples were examined. Using univariate and multivariate analysis, Axl expression was correlated with survival and other clinicopathologic features. To examine Axl functions in PDA, the effects of Axl knockdown on the invasion ability and radiation-induced apoptosis in PDA cell lines were measured.
RESULTS: Axl was overexpressed in 38 of 54 (70%) stage II PDA samples and 9 of 12 (75%) PDA cell lines. Axl overexpression was associated with higher frequencies of distant metastasis and poor overall and recurrence-free survivals (P = .03 and P = .04, respectively) independent of tumor size and stage or lymph node status in patients with stage II PDA. Knockdown of Axl expression in PDA cells abolished Gas6-mediated Akt activation, decreased invasion, and increased radiation-induced PARP cleavage and the percentage of apoptosis.
CONCLUSIONS: This study showed that Gas6 and Axl are frequently overexpressed in PDA cells and are associated with a poor prognosis in patients with stage II PDA. Axl promotes the invasion and survival of PDA cells. Therefore, targeting the Axl signaling pathway may represent a new approach to the treatment of PDA.
Copyright © 2010 American Cancer Society.

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Year:  2010        PMID: 20922806      PMCID: PMC4403266          DOI: 10.1002/cncr.25483

Source DB:  PubMed          Journal:  Cancer        ISSN: 0008-543X            Impact factor:   6.860


  32 in total

Review 1.  Cell signaling by receptor tyrosine kinases.

Authors:  J Schlessinger
Journal:  Cell       Date:  2000-10-13       Impact factor: 41.582

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Authors:  Aram F Hezel; Alec C Kimmelman; Ben Z Stanger; Nabeel Bardeesy; Ronald A Depinho
Journal:  Genes Dev       Date:  2006-05-15       Impact factor: 11.361

3.  Overexpression of protein tyrosine kinases in human esophageal cancer.

Authors:  T Nemoto; K Ohashi; T Akashi; J D Johnson; K Hirokawa
Journal:  Pathobiology       Date:  1997       Impact factor: 4.342

4.  Expression profile of tyrosine kinases in breast cancer.

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Journal:  Clin Cancer Res       Date:  2002-02       Impact factor: 12.531

5.  Multiple roles for the receptor tyrosine kinase axl in tumor formation.

Authors:  Sacha J Holland; Mark J Powell; Christian Franci; Emily W Chan; Annabelle M Friera; Robert E Atchison; John McLaughlin; Susan E Swift; Erlina S Pali; George Yam; Stephen Wong; Joe Lasaga; Mary R Shen; Simon Yu; Weiduan Xu; Yasumichi Hitoshi; Jakob Bogenberger; Jacques E Nör; Donald G Payan; James B Lorens
Journal:  Cancer Res       Date:  2005-10-15       Impact factor: 12.701

6.  Dominant-negative inhibition of the Axl receptor tyrosine kinase suppresses brain tumor cell growth and invasion and prolongs survival.

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8.  Axl promotes cell invasion by inducing MMP-9 activity through activation of NF-kappaB and Brg-1.

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10.  Receptor tyrosine kinases expressed in metastatic colon cancer.

Authors:  R J Craven; L H Xu; T M Weiner; Y W Fridell; G A Dent; S Srivastava; B Varnum; E T Liu; W G Cance
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3.  Small-Molecule Inhibition of Axl Targets Tumor Immune Suppression and Enhances Chemotherapy in Pancreatic Cancer.

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7.  MERTK Mediates Intrinsic and Adaptive Resistance to AXL-targeting Agents.

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Authors:  C-W Chien; P-C Hou; H-C Wu; Y-L Chang; S-C Lin; S-C Lin; B-W Lin; J-C Lee; Y-J Chang; H S Sun; S-J Tsai
Journal:  Oncogene       Date:  2016-05-02       Impact factor: 9.867

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