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Literature DB >> 20824154

Development of Practical Methodologies for the Synthesis of Functionalized Benzoboroxoles.

J Sravan Kumar¹, Christopher M Bashian, Michael A Corsello, Subash C Jonnalagadda, Venkatram R Mereddy.

Abstract

2-Formylphenylboronic acids upon reaction with activated olefins such as acrylates, methyl vinyl ketone, and acrylonitrile, etc. provide functionalized benzoboroxoles. The corresponding homologated benzoboroxoles were synthesized via the reaction of 2-formylphenylboronic acids with α-bromomethylacrylates.

Entities: Chemical Disease Species

Year: 2010 PMID： 20824154 PMCID： PMC2932456 DOI： 10.1016/j.tetlet.2010.06.077

Source DB: PubMed Journal: Tetrahedron Lett ISSN： 0040-4039 Impact factor: 2.415

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