Literature DB >> 20630750

A DOTA-peptide conjugate by copper-free click chemistry.

Molly E Martin1, Sharavathi G Parameswarappa, M Sue O'Dorisio, F Christopher Pigge, Michael K Schultz.   

Abstract

Attachment of DOTA to a novel monofluoro-cyclooctyne facilitates bioconjugation to an azide-modified peptide via Cu-free click chemistry. The resulting conjugate was radiolabeled with (111)In to afford a potential targeted molecular imaging agent with high specific activity and an excellent radiochemical purity. 2010 Elsevier Ltd. All rights reserved.

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Year:  2010        PMID： 20630750      PMCID： PMC3774834          DOI： 10.1016/j.bmcl.2010.06.111

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN： 0960-894X            Impact factor:   2.823


  20 in total

1.  Synthesis of a cross-bridged cyclam derivative for peptide conjugation and 64Cu radiolabeling.

Authors:  C Andrew Boswell; Celeste A S Regino; Kwamena E Baidoo; Karen J Wong; Ambika Bumb; Heng Xu; Diane E Milenic; James A Kelley; Christopher C Lai; Martin W Brechbiel
Journal:  Bioconjug Chem       Date:  2008-07-03       Impact factor: 4.774

Review 2.  Click-chemistry reactions in radiopharmaceutical chemistry: fast & easy introduction of radiolabels into biomolecules for in vivo imaging.

Authors:  C Wängler; R Schirrmacher; P Bartenstein; B Wängler
Journal:  Curr Med Chem       Date:  2010       Impact factor: 4.530

Review 3.  Click chemistry with DNA.

Authors:  Afaf H El-Sagheer; Tom Brown
Journal:  Chem Soc Rev       Date:  2010-02-09       Impact factor: 54.564

Review 4.  Cu-free click cycloaddition reactions in chemical biology.

Authors:  John C Jewett; Carolyn R Bertozzi
Journal:  Chem Soc Rev       Date:  2010-04       Impact factor: 54.564

5.  Copper-free click chemistry in living animals.

Authors:  Pamela V Chang; Jennifer A Prescher; Ellen M Sletten; Jeremy M Baskin; Isaac A Miller; Nicholas J Agard; Anderson Lo; Carolyn R Bertozzi
Journal:  Proc Natl Acad Sci U S A       Date:  2010-01-14       Impact factor: 11.205

Review 6.  The synthesis and chelation chemistry of DOTA-peptide conjugates.

Authors:  Luis M De León-Rodríguez; Zoltan Kovacs
Journal:  Bioconjug Chem       Date:  2007-12-12       Impact factor: 4.774

7.  Evaluation of [64Cu]Cu-DOTA and [64Cu]Cu-CB-TE2A chelates for targeted positron emission tomography with an alphavbeta6-specific peptide.

Authors:  Sven H Hausner; David L Kukis; M Karen J Gagnon; Catherine E Stanecki; Riccardo Ferdani; John F Marshall; Carolyn J Anderson; Julie L Sutcliffe
Journal:  Mol Imaging       Date:  2009 Mar-Apr       Impact factor: 4.488

8.  Copper-free click chemistry for the in situ crosslinking of photodegradable star polymers.

Authors:  Jeremiah A Johnson; Jeremy M Baskin; Carolyn R Bertozzi; Jeffrey T Koberstein; Nicholas J Turro
Journal:  Chem Commun (Camb)       Date:  2008-04-24       Impact factor: 6.222

Review 9.  Cross-bridged macrocyclic chelators for stable complexation of copper radionuclides for PET imaging.

Authors:  C J Anderson; T J Wadas; E H Wong; G R Weisman
Journal:  Q J Nucl Med Mol Imaging       Date:  2007-11-28       Impact factor: 2.346

10.  Synthesis of novel 1,4,7,10-tetraazacyclodecane-1,4,7,10-tetraacetic acid (DOTA) derivatives for chemoselective attachment to unprotected polyfunctionalized compounds.

Authors:  Sebastian Knör; Armin Modlinger; Thorsten Poethko; Margret Schottelius; Hans-Jürgen Wester; Horst Kessler
Journal:  Chemistry       Date:  2007       Impact factor: 5.236
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  10 in total

1.  Exploring strain-promoted 1,3-dipolar cycloadditions of end functionalized polymers.

Authors:  Petr A Ledin; Nagesh Kolishetti; Manish S Hudlikar; Geert-Jan Boons
Journal:  Chemistry       Date:  2014-06-06       Impact factor: 5.236

2.  A practical guide to the construction of radiometallated bioconjugates for positron emission tomography.

Authors:  Brian M Zeglis; Jason S Lewis
Journal:  Dalton Trans       Date:  2011-03-25       Impact factor: 4.390

3.  Copper-Free Click for PET: Rapid 1,3-Dipolar Cycloadditions with a Fluorine-18 Cyclooctyne.

Authors:  Richard D Carpenter; Sven H Hausner; Julie L Sutcliffe
Journal:  ACS Med Chem Lett       Date:  2011-10-07       Impact factor: 4.345

4.  The hydrazide/hydrazone click reaction as a biomolecule labeling strategy for M(CO)3 (M = Re, (99m)Tc) radiopharmaceuticals.

Authors:  Tanushree Ganguly; Benjamin B Kasten; Dejan-Krešimir Bučar; Leonard R MacGillivray; Clifford E Berkman; Paul D Benny
Journal:  Chem Commun (Camb)       Date:  2011-11-01       Impact factor: 6.222

5.  Improved synthesis and biological evaluation of chelator-modified α-MSH analogs prepared by copper-free click chemistry.

Authors:  Nicholas J Baumhover; Molly E Martin; Sharavathi G Parameswarappa; Kyle C Kloepping; M Sue O'Dorisio; F Christopher Pigge; Michael K Schultz
Journal:  Bioorg Med Chem Lett       Date:  2011-08-08       Impact factor: 2.823

6.  Preparation of a versatile bifunctional zeolite for targeted imaging applications.

Authors:  Nicholas Ndiege; Renugan Raidoo; Michael K Schultz; Sarah Larsen
Journal:  Langmuir       Date:  2011-02-09       Impact factor: 3.882

7.  Multi-Functionalization of Polymers by Strain-Promoted Cycloadditions.

Authors:  Petr A Ledin; Nagesh Kolishetti; Geert-Jan Boons
Journal:  Macromolecules       Date:  2013-10-08       Impact factor: 5.985

8.  Modular strategy for the construction of radiometalated antibodies for positron emission tomography based on inverse electron demand Diels-Alder click chemistry.

Authors:  Brian M Zeglis; Priya Mohindra; Gabriel I Weissmann; Vadim Divilov; Scott A Hilderbrand; Ralph Weissleder; Jason S Lewis
Journal:  Bioconjug Chem       Date:  2011-09-20       Impact factor: 4.774

9.  Aqueous synthesis of a small-molecule lanthanide chelator amenable to copper-free click chemistry.

Authors:  Stephanie C Bishop; Robert Winefield; Asokan Anbanandam; Jed N Lampe
Journal:  PLoS One       Date:  2019-03-27       Impact factor: 3.240

Review 10.  Opportunities for Expanding Encoded Chemical Diversification and Improving Hit Enrichment in mRNA-Displayed Peptide Libraries.

Authors:  Paddy R A Melsen; Ryoji Yoshisada; Seino A K Jongkees
Journal:  Chembiochem       Date:  2022-02-18       Impact factor: 3.461
  10 in total

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