Literature DB >> 20526458

CATALYTIC ENANTIOSELECTIVE BORANE REDUCTION OF BENZYL OXIMES: PREPARATION OF (S)-1-PYRIDIN-3-YL-ETHYLAMINE BIS HYDROCHLORIDE.

Kun Huang1, Margarita Ortiz-Marciales, David Hughes.   

Abstract

Entities:  

Year:  2010        PMID： 20526458      PMCID： PMC2879665     

Source DB:  PubMed          Journal:  Organic Synth        ISSN： 0078-6209


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  15 in total

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3.  Enantioselective reduction of oxime ethers with borane catalyzed by polymer-supported 2-piperazinemethanol

Authors: 
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4.  Spiroborate esters in the borane-mediated asymmetric synthesis of pyridyl and related heterocyclic alcohols.

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5.  One-pot asymmetric synthesis of either diastereomer of tert-butanesulfinyl-protected amines from ketones.

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Review 6.  Neuronal nicotinic acetylcholine receptors as targets for drug discovery.

Authors:  M W Holladay; M J Dart; J K Lynch
Journal:  J Med Chem       Date:  1997-12-19       Impact factor: 7.446

7.  (-)-Spiro[1-azabicyclo[2.2.2]octane-3,5'-oxazolidin-2'-one], a conformationally restricted analogue of acetylcholine, is a highly selective full agonist at the alpha 7 nicotinic acetylcholine receptor.

Authors:  G Mullen; J Napier; M Balestra; T DeCory; G Hale; J Macor; R Mack; J Loch; E Wu; A Kover; P Verhoest; A Sampognaro; E Phillips; Y Zhu; R Murray; R Griffith; J Blosser; D Gurley; A Machulskis; J Zongrone; A Rosen; J Gordon
Journal:  J Med Chem       Date:  2000-11-02       Impact factor: 7.446

8.  Novel and potent 6-chloro-3-pyridinyl ligands for the alpha4beta2 neuronal nicotinic acetylcholine receptor.

Authors:  B Latli; K D'Amour; J E Casida
Journal:  J Med Chem       Date:  1999-06-17       Impact factor: 7.446

9.  Asymmetric synthesis of primary amines via the spiroborate-catalyzed borane reduction of oxime ethers.

Authors:  Xiaogen Huang; Margarita Ortiz-Marciales; Kun Huang; Viatcheslav Stepanenko; Francisco G Merced; Angel M Ayala; Wildeliz Correa; Melvin De Jesús
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Review 10.  Recent developments in the synthesis of nicotinic acetylcholine receptor ligands.

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  4 in total

1.  Synthesis and stability of new spiroaminoborate esters.

Authors:  Viatcheslav Stepanenko; Melvin de Jesús; Carmelo Garcia; Charles L Barnes; Margarita Ortiz-Marciales
Journal:  Tetrahedron Lett       Date:  2012-02-22       Impact factor: 2.415

2.  Chiral epoxides via borane reduction of 2-haloketones catalyzed by spiroborate ester: application to the synthesis of optically pure 1,2-hydroxy ethers and 1,2-azido alcohols.

Authors:  Kun Huang; Haiyang Wang; Viatcheslav Stepanenko; Melvin De Jesús; Carilyn Torruellas; Wildeliz Correa; Margarita Ortiz-Marciales
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3.  Asymmetric synthesis of nonracemic primary amines via spiroborate-catalyzed reduction of pure (E)- and (Z)-O-benzyloximes: applications toward the synthesis of calcimimetic agents.

Authors:  Wenhua Ou; Sandraliz Espinosa; Héctor J Meléndez; Silvia M Farré; Jaime L Alvarez; Valerie Torres; Ileanne Martínez; Kiara M Santiago; Margarita Ortiz-Marciales
Journal:  J Org Chem       Date:  2013-05-13       Impact factor: 4.354

4.  Synthesis of enantiopure 1,2-azido and 1,2-amino alcohols via regio- and stereoselective ring-opening of enantiopure epoxides by sodium azide in hot water.

Authors:  Hai-Yang Wang; Kun Huang; Melvin De Jesús; Sandraliz Espinosa; Luis E Piñero-Santiago; Charles L Barnes; Margarita Ortiz-Marciales
Journal:  Tetrahedron Asymmetry       Date:  2016-02-15
  4 in total

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