Literature DB >> 20480486

A chloroacetamidine-based inactivator of protein arginine methyltransferase 1: design, synthesis, and in vitro and in vivo evaluation.

Obiamaka Obianyo1, Corey P Causey, Tanesha C Osborne, Justin E Jones, Young-Ho Lee, Michael R Stallcup, Paul R Thompson.   

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Year:  2010        PMID： 20480486      PMCID： PMC3060404          DOI： 10.1002/cbic.201000209

Source DB:  PubMed          Journal:  Chembiochem        ISSN： 1439-4227            Impact factor:   3.164


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  21 in total

1.  Structure of the predominant protein arginine methyltransferase PRMT1 and analysis of its binding to substrate peptides.

Authors:  Xing Zhang; Xiaodong Cheng
Journal:  Structure       Date:  2003-05       Impact factor: 5.006

Review 2.  The development and application of methods for activity-based protein profiling.

Authors:  Nadim Jessani; Benjamin F Cravatt
Journal:  Curr Opin Chem Biol       Date:  2004-02       Impact factor: 8.822

3.  Activation of nuclear receptor coactivator PGC-1alpha by arginine methylation.

Authors:  Catherine Teyssier; Han Ma; Roger Emter; Anastasia Kralli; Michael R Stallcup
Journal:  Genes Dev       Date:  2005-06-15       Impact factor: 11.361

4.  Regulation of transcription by a protein methyltransferase.

Authors:  D Chen; H Ma; H Hong; S S Koh; S M Huang; B T Schurter; D W Aswad; M R Stallcup
Journal:  Science       Date:  1999-06-25       Impact factor: 47.728

Review 5.  Arginine methylation an emerging regulator of protein function.

Authors:  Mark T Bedford; Stéphane Richard
Journal:  Mol Cell       Date:  2005-04-29       Impact factor: 17.970

Review 6.  Protein arginine deiminase 4 (PAD4): Current understanding and future therapeutic potential.

Authors:  Justin E Jones; Corey P Causey; Bryan Knuckley; Jessica L Slack-Noyes; Paul R Thompson
Journal:  Curr Opin Drug Discov Devel       Date:  2009-09

7.  A colorimetric 96-well microtiter plate assay for the determination of enzymatically formed citrulline.

Authors:  M Knipp; M Vasák
Journal:  Anal Biochem       Date:  2000-11-15       Impact factor: 3.365

8.  Kinetic characterization of protein arginine deiminase 4: a transcriptional corepressor implicated in the onset and progression of rheumatoid arthritis.

Authors:  Patricia L Kearney; Monica Bhatia; Nelroy G Jones; Luo Yuan; Mary C Glascock; Kristen L Catchings; Michiyuki Yamada; Paul R Thompson
Journal:  Biochemistry       Date:  2005-08-09       Impact factor: 3.162

9.  Small molecule regulators of protein arginine methyltransferases.

Authors:  Donghang Cheng; Neelu Yadav; Randall W King; Maurice S Swanson; Edward J Weinstein; Mark T Bedford
Journal:  J Biol Chem       Date:  2004-03-31       Impact factor: 5.157

10.  PRMT 3, a type I protein arginine N-methyltransferase that differs from PRMT1 in its oligomerization, subcellular localization, substrate specificity, and regulation.

Authors:  J Tang; J D Gary; S Clarke; H R Herschman
Journal:  J Biol Chem       Date:  1998-07-03       Impact factor: 5.157
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  16 in total

1.  Activity-based protein profiling of protein arginine methyltransferase 1.

Authors:  Obiamaka Obianyo; Corey P Causey; Justin E Jones; Paul R Thompson
Journal:  ACS Chem Biol       Date:  2011-08-23       Impact factor: 5.100

Review 2.  Small Molecule Inhibitors of Protein Arginine Methyltransferases.

Authors:  Hao Hu; Kun Qian; Meng-Chiao Ho; Y George Zheng
Journal:  Expert Opin Investig Drugs       Date:  2016-02-16       Impact factor: 6.206

Review 3.  Chemical biology of protein arginine modifications in epigenetic regulation.

Authors:  Jakob Fuhrmann; Kathleen W Clancy; Paul R Thompson
Journal:  Chem Rev       Date:  2015-05-13       Impact factor: 60.622

Review 4.  Inhibitors of Protein Methyltransferases and Demethylases.

Authors:  H Ümit Kaniskan; Michael L Martini; Jian Jin
Journal:  Chem Rev       Date:  2017-03-24       Impact factor: 60.622

5.  Kinetic mechanism of protein arginine methyltransferase 6 (PRMT6).

Authors:  Obiamaka Obianyo; Paul R Thompson
Journal:  J Biol Chem       Date:  2012-01-03       Impact factor: 5.157

6.  Mechanistic studies on transcriptional coactivator protein arginine methyltransferase 1.

Authors:  Heather L Rust; Cecilia I Zurita-Lopez; Steven Clarke; Paul R Thompson
Journal:  Biochemistry       Date:  2011-04-01       Impact factor: 3.162

Review 7.  Recent advances in targeting protein arginine methyltransferase enzymes in cancer therapy.

Authors:  Emily Smith; Wei Zhou; Polina Shindiapina; Said Sif; Chenglong Li; Robert A Baiocchi
Journal:  Expert Opin Ther Targets       Date:  2018-05-21       Impact factor: 6.902

Review 8.  Current chemical biology approaches to interrogate protein methyltransferases.

Authors:  Minkui Luo
Journal:  ACS Chem Biol       Date:  2012-02-01       Impact factor: 5.100

9.  Identification of small-molecule enhancers of arginine methylation catalyzed by coactivator-associated arginine methyltransferase 1.

Authors:  Sabrina Castellano; Astrid Spannhoff; Ciro Milite; Fabrizio Dal Piaz; Donghang Cheng; Alessandra Tosco; Monica Viviano; Abdellah Yamani; Agostino Cianciulli; Marina Sala; Vincent Cura; Jean Cavarelli; Ettore Novellino; Antonello Mai; Mark T Bedford; Gianluca Sbardella
Journal:  J Med Chem       Date:  2012-11-02       Impact factor: 7.446

10.  A selective inhibitor of PRMT5 with in vivo and in vitro potency in MCL models.

Authors:  Elayne Chan-Penebre; Kristy G Kuplast; Christina R Majer; P Ann Boriack-Sjodin; Tim J Wigle; L Danielle Johnston; Nathalie Rioux; Michael J Munchhof; Lei Jin; Suzanne L Jacques; Kip A West; Trupti Lingaraj; Kimberly Stickland; Scott A Ribich; Alejandra Raimondi; Margaret Porter Scott; Nigel J Waters; Roy M Pollock; Jesse J Smith; Olena Barbash; Melissa Pappalardi; Thau F Ho; Kelvin Nurse; Khyati P Oza; Kathleen T Gallagher; Ryan Kruger; Mikel P Moyer; Robert A Copeland; Richard Chesworth; Kenneth W Duncan
Journal:  Nat Chem Biol       Date:  2015-04-27       Impact factor: 15.040
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