Literature DB >> 20154660

Rethinking screening.

Thomas Kodadek1.   

Abstract

Year:  2010        PMID： 20154660     DOI： 10.1038/nchembio.303

Source DB:  PubMed          Journal:  Nat Chem Biol        ISSN： 1552-4450            Impact factor:   15.040


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  21 in total

1.  A novel peptide-based encoding system for "one-bead one-compound" peptidomimetic and small molecule combinatorial libraries.

Authors:  Ruiwu Liu; Jan Marik; Kit S Lam
Journal:  J Am Chem Soc       Date:  2002-07-03       Impact factor: 15.419

Review 2.  Recent advances in heterocycle generation using the efficient Ugi multiple-component condensation reaction.

Authors:  Paul A Tempest
Journal:  Curr Opin Drug Discov Devel       Date:  2005-11

3.  Cleavable hydrophilic linker for one-bead-one-compound sequencing of oligomer libraries by tandem mass spectrometry.

Authors:  Margot G Paulick; Kathryn M Hart; Kristin M Brinner; Meiliana Tjandra; Deborah H Charych; Ronald N Zuckermann
Journal:  J Comb Chem       Date:  2006 May-Jun

4.  Synthetic ligands discovered by in vitro selection.

Authors:  S Jarrett Wrenn; Rebecca M Weisinger; David R Halpin; Pehr B Harbury
Journal:  J Am Chem Soc       Date:  2007-10-06       Impact factor: 15.419

5.  A new type of synthetic peptide library for identifying ligand-binding activity.

Authors:  K S Lam; S E Salmon; E M Hersh; V J Hruby; W M Kazmierski; R J Knapp
Journal:  Nature       Date:  1991-11-07       Impact factor: 49.962

Review 6.  Activity-based protein profiling: from enzyme chemistry to proteomic chemistry.

Authors:  Benjamin F Cravatt; Aaron T Wright; John W Kozarich
Journal:  Annu Rev Biochem       Date:  2008       Impact factor: 23.643

7.  Perspectives on the development of imatinib and the future of cancer research.

Authors:  Brian J Druker
Journal:  Nat Med       Date:  2009-10       Impact factor: 53.440

8.  Complex synthetic chemical libraries indexed with molecular tags.

Authors:  M H Ohlmeyer; R N Swanson; L W Dillard; J C Reader; G Asouline; R Kobayashi; M Wigler; W C Still
Journal:  Proc Natl Acad Sci U S A       Date:  1993-12-01       Impact factor: 11.205

9.  Combinatorial chemistry identifies high-affinity peptidomimetics against alpha4beta1 integrin for in vivo tumor imaging.

Authors:  Li Peng; Ruiwu Liu; Jan Marik; Xiaobing Wang; Yoshikazu Takada; Kit S Lam
Journal:  Nat Chem Biol       Date:  2006-06-11       Impact factor: 15.040

10.  Rapid synthesis of diketopiperazine macroarrays via Ugi four-component reactions on planar solid supports.

Authors:  Qi Lin; Helen E Blackwell
Journal:  Chem Commun (Camb)       Date:  2006-07-21       Impact factor: 6.222
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  22 in total

1.  Identifying mechanism-of-action targets for drugs and probes.

Authors:  Elisabet Gregori-Puigjané; Vincent Setola; Jérôme Hert; Brenda A Crews; John J Irwin; Eugen Lounkine; Lawrence Marnett; Bryan L Roth; Brian K Shoichet
Journal:  Proc Natl Acad Sci U S A       Date:  2012-06-18       Impact factor: 11.205

2.  The chemistry and pharmacology of privileged pyrroloquinazolines.

Authors:  Bo Chao; Bingbing X Li; Xiangshu Xiao
Journal:  Medchemcomm       Date:  2015-04-01       Impact factor: 3.597

3.  Potential pharmacological chaperones targeting cancer-associated MCL-1 and Parkinson disease-associated α-synuclein.

Authors:  Misook Oh; Ji Hoon Lee; Wei Wang; Hui Sun Lee; Woo Sirl Lee; Christopher Burlak; Wonpil Im; Quyen Q Hoang; Hyun-Suk Lim
Journal:  Proc Natl Acad Sci U S A       Date:  2014-07-14       Impact factor: 11.205

4.  Fragment-based domain shuffling approach for the synthesis of pyran-based macrocycles.

Authors:  Eamon Comer; Haibo Liu; Adrien Joliton; Alexandre Clabaut; Christopher Johnson; Lakshmi B Akella; Lisa A Marcaurelle
Journal:  Proc Natl Acad Sci U S A       Date:  2011-03-07       Impact factor: 11.205

Review 5.  Synthetic receptors with antibody-like binding affinities.

Authors:  Thomas Kodadek
Journal:  Curr Opin Chem Biol       Date:  2010-07-30       Impact factor: 8.822

6.  High-throughput kinase profiling: a more efficient approach toward the discovery of new kinase inhibitors.

Authors:  Chandrasekhar V Miduturu; Xianming Deng; Nicholas Kwiatkowski; Wannian Yang; Laurent Brault; Panagis Filippakopoulos; Eunah Chung; Qingkai Yang; Juerg Schwaller; Stefan Knapp; Randall W King; Jiing-Dwan Lee; Sanna Herrgard; Patrick Zarrinkar; Nathanael S Gray
Journal:  Chem Biol       Date:  2011-07-29

7.  Generating DNA synbodies from previously discovered peptides.

Authors:  Rui Liu; Bing Jiang; Hanyang Yu; John C Chaput
Journal:  Chembiochem       Date:  2011-06-20       Impact factor: 3.164

Review 8.  Probing the probes: fitness factors for small molecule tools.

Authors:  Paul Workman; Ian Collins
Journal:  Chem Biol       Date:  2010-06-25

9.  Akt2 and acid ceramidase cooperate to induce cell invasion and resistance to apoptosis.

Authors:  Norbert Berndt; Ronil Patel; Hua Yang; Maria E Balasis; Saïd M Sebti
Journal:  Cell Cycle       Date:  2013-06-06       Impact factor: 4.534

Review 10.  The identification of high-affinity G protein-coupled receptor ligands from large combinatorial libraries using multicolor quantum dot-labeled cell-based screening.

Authors:  Junjie Fu; Timothy Lee; Xin Qi
Journal:  Future Med Chem       Date:  2014-05       Impact factor: 3.808
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