Literature DB >> 20107652

Efficient synthesis of aminopyridine derivatives by copper catalyzed amination reactions.

Mohammed K Elmkaddem1, Cédric Fischmeister, Christophe M Thomas, Jean-Luc Renaud.   

Abstract

A copper(i) catalyzed amination reaction utilizing aqueous ammonia and operating under mild conditions is presented. This method was employed for the efficient synthesis of various aminopyridine derivatives bearing electron withdrawing and electron donating groups.

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Year:  2009        PMID： 20107652     DOI： 10.1039/b916569j

Source DB:  PubMed          Journal:  Chem Commun (Camb)        ISSN： 1359-7345            Impact factor:   6.222


  5 in total

1.  Installation of protected ammonia equivalents onto aromatic & heteroaromatic rings in water enabled by micellar catalysis.

Authors:  Nicholas A Isley; Sebastian Dobarco; Bruce H Lipshutz
Journal:  Green Chem       Date:  2014-01-02       Impact factor: 10.182

2.  Pyridyl CO2 Fixation Enabled by a Secondary Hydrogen Bonding Coordination Sphere.

Authors:  Jacqueline N Gayton; Qing Li; Lakeeta Sanders; Roberta R Rodrigues; Glake Hill; Jared H Delcamp
Journal:  ACS Omega       Date:  2020-05-11

3.  Metal-free cascade synthesis of unsymmetrical 2-aminopyrimidines from imidazolate enaminones.

Authors:  Xue Cui; Jianting Ma; Tingting Zeng; Junyu Xu; Youbin Li; Xuesong Wang
Journal:  RSC Adv       Date:  2021-07-14       Impact factor: 4.036

4.  Discovery of a neuroprotective chemical, (S)-N-(3-(3,6-dibromo-9H-carbazol-9-yl)-2-fluoropropyl)-6-methoxypyridin-2-amine [(-)-P7C3-S243], with improved druglike properties.

Authors:  Jacinth Naidoo; Hector De Jesus-Cortes; Paula Huntington; Sandi Estill; Lorraine K Morlock; Ruth Starwalt; Thomas J Mangano; Noelle S Williams; Andrew A Pieper; Joseph M Ready
Journal:  J Med Chem       Date:  2014-04-16       Impact factor: 7.446

5.  Facile Hydrogenative Deprotection of N-Benzyl Groups Using a Mixed Catalyst of Palladium and Niobic Acid-on-Carbon.

Authors:  Yuta Yamamoto; Eisho Shimizu; Kazuho Ban; Yoshiyuki Wada; Tomoteru Mizusaki; Masatoshi Yoshimura; Yukio Takagi; Yoshinari Sawama; Hironao Sajiki
Journal:  ACS Omega       Date:  2020-02-05
  5 in total

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