Literature DB >> 20058293

Chelator fragment libraries for targeting metalloproteinases.

Arpita Agrawal1, Sherida L Johnson, Jennifer A Jacobsen, Melissa T Miller, Li-Hsing Chen, Maurizio Pellecchia, Seth M Cohen.   

Abstract

Entities:  

Mesh:

Substances:

Year:  2010        PMID: 20058293      PMCID: PMC2825879          DOI: 10.1002/cmdc.200900516

Source DB:  PubMed          Journal:  ChemMedChem        ISSN: 1860-7179            Impact factor:   3.466


× No keyword cloud information.
  23 in total

Review 1.  Structure- and fragment-based approaches to protease inhibition.

Authors:  Sherida L Johnson; Maurizio Pellecchia
Journal:  Curr Top Med Chem       Date:  2006       Impact factor: 3.295

2.  Evaluation and binding-mode prediction of thiopyrone-based inhibitors of anthrax lethal factor.

Authors:  Jana A Lewis; John Mongan; J Andrew McCammon; Seth M Cohen
Journal:  ChemMedChem       Date:  2006-07       Impact factor: 3.466

Review 3.  The design of inhibitors for medicinally relevant metalloproteins.

Authors:  Faith E Jacobsen; Jana A Lewis; Seth M Cohen
Journal:  ChemMedChem       Date:  2007-02       Impact factor: 3.466

4.  Fragment-based drug design: how big is too big?

Authors:  Philip J Hajduk
Journal:  J Med Chem       Date:  2006-11-30       Impact factor: 7.446

5.  A library of novel hydroxamic acids targeting the metallo-protease family: design, parallel synthesis and screening.

Authors:  Marion Flipo; Terence Beghyn; Julie Charton; Virginie A Leroux; Benoit P Deprez; Rebecca F Deprez-Poulain
Journal:  Bioorg Med Chem       Date:  2006-10-12       Impact factor: 3.641

Review 6.  Recent developments in fragment-based drug discovery.

Authors:  Miles Congreve; Gianni Chessari; Dominic Tisi; Andrew J Woodhead
Journal:  J Med Chem       Date:  2008-05-06       Impact factor: 7.446

7.  Novel small-molecule inhibitors of anthrax lethal factor identified by high-throughput screening.

Authors:  Igor A Schepetkin; Andrei I Khlebnikov; Liliya N Kirpotina; Mark T Quinn
Journal:  J Med Chem       Date:  2006-08-24       Impact factor: 7.446

8.  A high-throughput screening approach to anthrax lethal factor inhibition.

Authors:  Sherida L Johnson; Li-Hsing Chen; Maurizio Pellecchia
Journal:  Bioorg Chem       Date:  2007-02-22       Impact factor: 5.275

9.  Zinc-binding groups modulate selective inhibition of MMPs.

Authors:  Arpita Agrawal; Diego Romero-Perez; Jennifer A Jacobsen; Francisco J Villarreal; Seth M Cohen
Journal:  ChemMedChem       Date:  2008-05       Impact factor: 3.466

10.  Identification and characterization of small molecule inhibitors of a class I histone deacetylase from Plasmodium falciparum.

Authors:  Vishal Patel; Ralph Mazitschek; Bradley Coleman; Cokey Nguyen; Sameer Urgaonkar; Joseph Cortese; Robert H Barker; Edward Greenberg; Weiping Tang; James E Bradner; Stuart L Schreiber; Manoj T Duraisingh; Dyann F Wirth; Jon Clardy
Journal:  J Med Chem       Date:  2009-04-23       Impact factor: 7.446

View more
  28 in total

1.  Identifying chelators for metalloprotein inhibitors using a fragment-based approach.

Authors:  Jennifer A Jacobsen; Jessica L Fullagar; Melissa T Miller; Seth M Cohen
Journal:  J Med Chem       Date:  2010-12-28       Impact factor: 7.446

2.  A Bioinorganic Approach to Fragment-Based Drug Discovery Targeting Metalloenzymes.

Authors:  Seth M Cohen
Journal:  Acc Chem Res       Date:  2017-07-17       Impact factor: 22.384

3.  Identification of the 2-Benzoxazol-2-yl-phenol Scaffold as New Hit for JMJD3 Inhibition.

Authors:  Assunta Giordano; Giovanni Forte; Stefania Terracciano; Alessandra Russo; Marina Sala; Maria C Scala; Catrine Johansson; Udo Oppermann; Raffaele Riccio; Ines Bruno; Simone Di Micco
Journal:  ACS Med Chem Lett       Date:  2019-02-25       Impact factor: 4.345

4.  Dipicolinic Acid Derivatives as Inhibitors of New Delhi Metallo-β-lactamase-1.

Authors:  Allie Y Chen; Pei W Thomas; Alesha C Stewart; Alexander Bergstrom; Zishuo Cheng; Callie Miller; Christopher R Bethel; Steven H Marshall; Cy V Credille; Christopher L Riley; Richard C Page; Robert A Bonomo; Michael W Crowder; David L Tierney; Walter Fast; Seth M Cohen
Journal:  J Med Chem       Date:  2017-08-30       Impact factor: 7.446

Review 5.  Targeting Metalloenzymes for Therapeutic Intervention.

Authors:  Allie Y Chen; Rebecca N Adamek; Benjamin L Dick; Cy V Credille; Christine N Morrison; Seth M Cohen
Journal:  Chem Rev       Date:  2018-09-07       Impact factor: 60.622

6.  A noncompetitive inhibitor for Mycobacterium tuberculosis's class IIa fructose 1,6-bisphosphate aldolase.

Authors:  Glenn C Capodagli; Wafik G Sedhom; Mary Jackson; Kateri A Ahrendt; Scott D Pegan
Journal:  Biochemistry       Date:  2013-12-24       Impact factor: 3.162

7.  Identification of 3-hydroxy-1,2-dimethylpyridine-4(1H)-thione as a metal-binding motif for the inhibition of botulinum neurotoxin A.

Authors:  Lucy Lin; Lewis D Turner; Peter Šilhár; Sabine Pellett; Eric A Johnson; Kim D Janda
Journal:  RSC Med Chem       Date:  2020-11-12

8.  Computational exploration of zinc binding groups for HDAC inhibition.

Authors:  Kai Chen; Liping Xu; Olaf Wiest
Journal:  J Org Chem       Date:  2013-04-29       Impact factor: 4.354

9.  Structure-Activity Relationships in Metal-Binding Pharmacophores for Influenza Endonuclease.

Authors:  Cy V Credille; Benjamin L Dick; Christine N Morrison; Ryjul W Stokes; Rebecca N Adamek; Nicholas C Wu; Ian A Wilson; Seth M Cohen
Journal:  J Med Chem       Date:  2018-10-31       Impact factor: 7.446

10.  Ligand-induced expansion of the S1' site in the anthrax toxin lethal factor.

Authors:  Kimberly M Maize; Elbek K Kurbanov; Rodney L Johnson; Elizabeth Ambrose Amin; Barry C Finzel
Journal:  FEBS Lett       Date:  2015-11-11       Impact factor: 4.124

View more

北京卡尤迪生物科技股份有限公司 © 2022-2023.