Literature DB >> 20046955

A Survey of Solvents for the Conrad-Limpach Synthesis of 4-Hydroxyquinolones.

Jean-Cristophe Brouet1, Shen Gu, Norton P Peet, John D Williams.   

Abstract

A study on the synthesis of a 4-hydroxyquinoline derivative using the Conrad-Limpach reaction led to the identification of inexpensive and user-friendly solvents for this thermal condensation.

Entities:  

Year:  2009        PMID： 20046955      PMCID： PMC2744084          DOI： 10.1080/00397910802542044

Source DB:  PubMed          Journal:  Synth Commun        ISSN： 0039-7911            Impact factor:   2.007


  10 in total

1.  The quest for quinine: those who won the battles and those who won the war.

Authors:  Teodoro S Kaufman; Edmundo A Rúveda
Journal:  Angew Chem Int Ed Engl       Date:  2005-01-28       Impact factor: 15.336

2.  PDE-10A inhibitors as insulin secretagogues.

Authors:  Louis-David Cantin; Steven Magnuson; David Gunn; Nicole Barucci; Marina Breuhaus; William H Bullock; Jennifer Burke; Thomas H Claus; Michelle Daly; Lynn Decarr; Ann Gore-Willse; Helana Hoover-Litty; Ellalahewage S Kumarasinghe; Yaxin Li; Sidney X Liang; James N Livingston; Timothy Lowinger; Margit Macdougall; Herbert O Ogutu; Alan Olague; Ronda Ott-Morgan; Robert W Schoenleber; Adrian Tersteegen; Philip Wickens; Zhonghua Zhang; Jian Zhu; Lei Zhu; Laurel J Sweet
Journal:  Bioorg Med Chem Lett       Date:  2007-02-25       Impact factor: 2.823

3.  The chemistry of 4-hydroxyquinolines.

Authors:  R H REITSEMA
Journal:  Chem Rev       Date:  1948-08       Impact factor: 60.622

4.  Substituted quinolines.

Authors:  C E KASLOW; R D STAYNER
Journal:  J Am Chem Soc       Date:  1948-10       Impact factor: 15.419

5.  Studies on disease-modifying antirheumatic drugs: synthesis of novel quinoline and quinazoline derivatives and their anti-inflammatory effect.

Authors:  A Baba; N Kawamura; H Makino; Y Ohta; S Taketomi; T Sohda
Journal:  J Med Chem       Date:  1996-12-20       Impact factor: 7.446

Review 6.  Chemotherapy of the drug-resistant malarias.

Authors:  L H Schmidt
Journal:  Annu Rev Microbiol       Date:  1969       Impact factor: 15.500

7.  Introduction of a carboxyl group through an acetal as a new route to carboxylic acid derivatives of sugars.

Authors:  S Carbonnel; C Fayet; J Gelas
Journal:  Carbohydr Res       Date:  1999-06-30       Impact factor: 2.104

8.  Synthesis of novel quinolone and quinoline-2-carboxylic acid (4-morpholin-4-yl-phenyl)amides: a late-stage diversification approach to potent 5HT1B antagonists.

Authors:  Carey L Horchler; John P McCauley; James E Hall; Dean H Snyder; W Craig Moore; Thomas J Hudzik; Marc J Chapdelaine
Journal:  Bioorg Med Chem       Date:  2006-10-20       Impact factor: 3.641

9.  Synthesis and antilipolytic activities of quinolyl carbanilates and related analogues.

Authors:  J H Musser; U Chakraborty; K Bailey; S Sciortino; C Whyzmuzis; D Amin; C A Sutherland
Journal:  J Med Chem       Date:  1987-01       Impact factor: 7.446

10.  Synthesis and SAR of 8-arylquinolines as potent corticotropin-releasing factor1 (CRF1) receptor antagonists.

Authors:  Charles Q Huang; Keith Wilcoxen; James R McCarthy; Mustapha Haddach; Thomas R Webb; Jian Gu; Yun-Feng Xie; Dimitri E Grigoriadis; Chen Chen
Journal:  Bioorg Med Chem Lett       Date:  2003-10-06       Impact factor: 2.823
  10 in total
  5 in total

1.  Discovery of heterocyclic replacements for the coumarin core of anti-tubercular FadD32 inhibitors.

Authors:  Chao Fang; Katie K Lee; Raymond Nietupski; Robert H Bates; Raquel Fernandez-Menendez; Eva Maria Lopez-Roman; Laura Guijarro-Lopez; Yunxing Yin; Zuozhong Peng; James E Gomez; Stewart Fisher; David Barros-Aguirre; Brian K Hubbard; Michael H Serrano-Wu; Deborah T Hung
Journal:  Bioorg Med Chem Lett       Date:  2018-09-29       Impact factor: 2.823

Review 2.  Recent advances in chemistry and therapeutic potential of functionalized quinoline motifs - a review.

Authors:  Olayinka O Ajani; King T Iyaye; Olabisi T Ademosun
Journal:  RSC Adv       Date:  2022-06-24       Impact factor: 4.036

3.  Small molecule inhibitors of anthrax lethal factor toxin.

Authors:  John D Williams; Atiyya R Khan; Steven C Cardinale; Michelle M Butler; Terry L Bowlin; Norton P Peet
Journal:  Bioorg Med Chem       Date:  2013-11-13       Impact factor: 3.641

4.  A New Scalable Synthesis of ELQ-300, ELQ-316, and other Antiparasitic Quinolones.

Authors:  Sovitj Pou; Rozalia A Dodean; Lisa Frueh; Katherine M Liebman; Rory T Gallagher; Haihong Jin; Robert T Jacobs; Aaron Nilsen; David R Stuart; J Stone Doggett; Michael K Riscoe; Rolf W Winter
Journal:  Org Process Res Dev       Date:  2021-08-04       Impact factor: 3.858

5.  Light-driven selective aerobic oxidation of (iso)quinoliniums and related heterocycles.

Authors:  Meimei Zhou; Keyang Yu; Jianxin Liu; Weimei Shi; Yingming Pan; Haitao Tang; Xiangjun Peng; Qian Liu; Hengshan Wang
Journal:  RSC Adv       Date:  2021-05-04       Impact factor: 3.361
  5 in total

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