Literature DB >> 20012167

Hydrodynamic and species transfer simulations in the USP 4 dissolution apparatus: considerations for dissolution in a low velocity pulsing flow.

Deirdre M D'Arcy1, Bo Liu, Geoff Bradley, Anne Marie Healy, Owen I Corrigan.   

Abstract

PURPOSE: To simulate the hydrodynamics in the flow-through (USP 4) dissolution apparatus and investigate the effects of hydrodynamics on mass transfer in a low velocity pulsing flow.
METHODS: Computational fluid dynamics (CFD) was used to simulate the hydrodynamics and mass transfer in pulsing flow. Experimental flow visualisation was used to qualitatively confirm simulated hydrodynamic and mass transfer features. The experimental dissolution rate at 8 ml min(-1) (22.6 mm flow-through cell) was compared to the experimental dissolution rate in a free convection system.
RESULTS: Simulations revealed periods of low velocity at all flow rates, evidence of boundary layer separation, and, at higher flow rates, residual fluid motion during zero inlet velocity periods. The simulated diffusion boundary layer thickness varied in certain regions over the course of the pulse. The experimental dissolution rate in the free convection system was faster than that at 8 ml min(-1) in the flow-through apparatus.
CONCLUSIONS: A low velocity pulsing flow running counter to gravity inhibited the experimental dissolution rate compared to that in a free convection system. From the CFD simulations generated, simulation of both hydrodynamics and species transfer is recommended to characterise the influence of hydrodynamics on dissolution in a low velocity pulsing flow.

Entities:  

Mesh:

Substances:

Year:  2009        PMID: 20012167     DOI: 10.1007/s11095-009-0010-4

Source DB:  PubMed          Journal:  Pharm Res        ISSN: 0724-8741            Impact factor:   4.200


  27 in total

1.  Robustness testing, using experimental design, of a flow-through dissolution method for a product where the actives have markedly differing solubility properties.

Authors:  M S Bloomfield; W C Butler
Journal:  Int J Pharm       Date:  2000-09-25       Impact factor: 5.875

2.  Comparison of dissolution profiles for albendazole tablets using USP apparatus 2 and 4.

Authors:  Marcela Hurtado y de la Peña; Yolanda Vargas Alvarado; Adriana Miriam Domínguez-Ramírez; Alma Rosa Cortés Arroyo
Journal:  Drug Dev Ind Pharm       Date:  2003-08       Impact factor: 3.225

Review 3.  Engineering tools for understanding the hydrodynamics of dissolution tests.

Authors:  Joseph Kukura; Paulo E Arratia; Edit S Szalai; Fernando J Muzzio
Journal:  Drug Dev Ind Pharm       Date:  2003-02       Impact factor: 3.225

4.  Gastric flow and mixing studied using computer simulation.

Authors:  Anupam Pal; Keshavamurthy Indireshkumar; Werner Schwizer; Bertil Abrahamsson; Michael Fried; James G Brasseur
Journal:  Proc Biol Sci       Date:  2004-12-22       Impact factor: 5.349

5.  Computational fluid dynamics modeling of the paddle dissolution apparatus: agitation rate, mixing patterns, and fluid velocities.

Authors:  Leonard G McCarthy; Geoff Bradley; James C Sexton; Owen I Corrigan; Anne Marie Healy
Journal:  AAPS PharmSciTech       Date:  2004-04-08       Impact factor: 3.246

6.  Hydrodynamic simulation (computational fluid dynamics) of asymmetrically positioned tablets in the paddle dissolution apparatus: impact on dissolution rate and variability.

Authors:  D M D'Arcy; O I Corrigan; A M Healy
Journal:  J Pharm Pharmacol       Date:  2005-10       Impact factor: 3.765

7.  Towards determining appropriate hydrodynamic conditions for in vitro in vivo correlations using computational fluid dynamics.

Authors:  Deirdre M D'Arcy; Anne Marie Healy; Owen I Corrigan
Journal:  Eur J Pharm Sci       Date:  2009-03-06       Impact factor: 4.384

8.  Mathematical modeling of the fluid dynamics in the flow-through cell.

Authors:  Maziar Kakhi
Journal:  Int J Pharm       Date:  2009-04-16       Impact factor: 5.875

9.  Hydrodynamic, mass transfer, and dissolution effects induced by tablet location during dissolution testing.

Authors:  Ge Bai; Piero M Armenante
Journal:  J Pharm Sci       Date:  2009-04       Impact factor: 3.534

10.  Improved method for diffusion coefficient determinations employing the silver membrane filter.

Authors:  A H Goldberg; W I Higuchi
Journal:  J Pharm Sci       Date:  1968-09       Impact factor: 3.534

View more
  8 in total

1.  Real-time UV imaging of nicotine release from transdermal patch.

Authors:  Jesper Østergaard; Emil Meng-Lund; Susan Weng Larsen; Claus Larsen; Karsten Petersson; James Lenke; Henrik Jensen
Journal:  Pharm Res       Date:  2010-09-02       Impact factor: 4.200

2.  Effects of Pump Pulsation on Hydrodynamic Properties and Dissolution Profiles in Flow-Through Dissolution Systems (USP 4).

Authors:  Hiroyuki Yoshida; Akemi Kuwana; Hiroko Shibata; Ken-Ichi Izutsu; Yukihiro Goda
Journal:  Pharm Res       Date:  2016-02-11       Impact factor: 4.200

3.  Computational fluid dynamics simulation of hydrodynamics in USP apparatus 3-the influence of dip rate.

Authors:  Satish Perivilli; Maziar Kakhi; Erika Stippler
Journal:  Pharm Res       Date:  2014-11-19       Impact factor: 4.200

4.  Particle Image Velocimetry Evaluation of Fluid Flow Profiles in USP 4 Flow-Through Dissolution Cells.

Authors:  Hiroyuki Yoshida; Akemi Kuwana; Hiroko Shibata; Ken-Ichi Izutsu; Yukihiro Goda
Journal:  Pharm Res       Date:  2015-03-20       Impact factor: 4.200

5.  Using USP I and USP IV for discriminating dissolution rates of nano- and microparticle-loaded pharmaceutical strip-films.

Authors:  Lucas Sievens-Figueroa; Natasha Pandya; Anagha Bhakay; Golshid Keyvan; Bozena Michniak-Kohn; Ecevit Bilgili; Rajesh N Davé
Journal:  AAPS PharmSciTech       Date:  2012-10-23       Impact factor: 3.246

Review 6.  In vitro dissolution considerations associated with nano drug delivery systems.

Authors:  Ritu Gupta; Yuan Chen; Huan Xie
Journal:  Wiley Interdiscip Rev Nanomed Nanobiotechnol       Date:  2021-06-15

7.  The relative importance of internal and external physical resistances to mass transfer for caffeine release from apple pectin tablets.

Authors:  Shu Cheng; Chao Zhong; Timothy A G Langrish; Yongmei Sun; Zelin Zhou; Zexin Lei
Journal:  Curr Res Food Sci       Date:  2022-03-26

8.  Determination of Intrinsic Drug Dissolution and Solute Effective Transport Rate during Laminar Fluid Flow at Different Velocities.

Authors:  Sara B E Andersson; Göran Frenning; Göran Alderborn
Journal:  Pharmaceutics       Date:  2021-06-04       Impact factor: 6.321

  8 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.