Literature DB >> 19943178

The effects of bilastine compared with cetirizine, fexofenadine, and placebo on allergen-induced nasal and ocular symptoms in patients exposed to aeroallergen in the Vienna Challenge Chamber.

Friedrich Horak1, Petra Zieglmayer, René Zieglmayer, Patrick Lemell.   

Abstract

OBJECTIVE AND
DESIGN: This double-blind cross-over study compared the potential of bilastine, cetirizine, and fexofenadine to relieve the symptoms of allergic rhinitis. SUBJECTS AND METHODS: Seventy-five allergic volunteers were challenged with grass pollen in the Vienna Challenge Chamber (VCC) on two consecutive days of allergen provocation; 6 h on day 1 and 4 h day 2. Bilastine 20 mg, cetirizine 10 mg, fexofenadine 120 mg, or placebo were taken orally 2 h after the start of provocation on day 1 only. Total nasal symptom scores, the global symptom scores, nasal secretions, and eye symptoms were assessed on both day 1 and day 2. RESULTS AND
CONCLUSIONS: Bilastine had a rapid onset of action, within 1 h, and a long duration of action, greater than 26 h. Cetirizine was similar. Fexofenadine was similar on day 1 but less effective on day 2, indicating a shorter duration of action. Bilastine, like cetirizine and fexofenadine, was safe and well tolerated in this study.

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Year:  2009        PMID: 19943178     DOI: 10.1007/s00011-009-0117-4

Source DB:  PubMed          Journal:  Inflamm Res        ISSN: 1023-3830            Impact factor:   4.575


  24 in total

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Authors:  R Leurs; M K Church; M Taglialatela
Journal:  Clin Exp Allergy       Date:  2002-04       Impact factor: 5.018

2.  Levocetirizine has a longer duration of action on improving total nasal symptoms score than fexofenadine after single administration.

Authors:  Friedrich Horak; Petra U Zieglmayer; R Zieglmayer; A Kavina; P Lemell
Journal:  Br J Clin Pharmacol       Date:  2005-07       Impact factor: 4.335

3.  Levocetirizine improves health-related quality of life and health status in persistent allergic rhinitis.

Authors:  G Walter Canonica; Jean Bousquet; Geneviève Van Hammée; Claus Bachert; Stephen R Durham; Ludger Klimek; Joaquim Mullol; Paul B Van Cauwenberge
Journal:  Respir Med       Date:  2006-05-24       Impact factor: 3.415

4.  Preclinical pharmacology of bilastine, a new selective histamine H1 receptor antagonist: receptor selectivity and in vitro antihistaminic activity.

Authors:  Reyes Corcóstegui; Luis Labeaga; Ana Innerárity; Agustin Berisa; Aurelio Orjales
Journal:  Drugs R D       Date:  2005

5.  P-glycoprotein plays a major role in the efflux of fexofenadine in the small intestine and blood-brain barrier, but only a limited role in its biliary excretion.

Authors:  Harunobu Tahara; Hiroyuki Kusuhara; Eiichi Fuse; Yuichi Sugiyama
Journal:  Drug Metab Dispos       Date:  2005-04-08       Impact factor: 3.922

6.  Controlled comparison of the efficacy and safety of cetirizine 10 mg o.d. and fexofenadine 120 mg o.d. in reducing symptoms of seasonal allergic rhinitis.

Authors:  F Horak; P Stübner; R Zieglmayer; A Kavina; C De Vos; B Burtin; F Donnelly
Journal:  Int Arch Allergy Immunol       Date:  2001-05       Impact factor: 2.749

Review 7.  Fexofenadine.

Authors:  A Markham; A J Wagstaff
Journal:  Drugs       Date:  1998-02       Impact factor: 9.546

8.  Levocetirizine improves nasal obstruction and modulates cytokine pattern in patients with seasonal allergic rhinitis: a pilot study.

Authors:  G Ciprandi; I Cirillo; A Vizzaccaro; M A Tosca
Journal:  Clin Exp Allergy       Date:  2004-06       Impact factor: 5.018

9.  Comparison of the effects of desloratadine 5-mg daily and placebo on nasal airflow and seasonal allergic rhinitis symptoms induced by grass pollen exposure.

Authors:  F Horak; P Stübner; R Zieglmeyer; A G Harris
Journal:  Allergy       Date:  2003-06       Impact factor: 13.146

10.  Multidrug resistance-associated protein 2 is primarily responsible for the biliary excretion of fexofenadine in mice.

Authors:  Xianbin Tian; Maciej J Zamek-Gliszczynski; Jun Li; Arlene S Bridges; Ken-ichi Nezasa; Nita J Patel; Thomas J Raub; Kim L R Brouwer
Journal:  Drug Metab Dispos       Date:  2007-10-03       Impact factor: 3.922

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  21 in total

Review 1.  New therapies for allergic rhinitis.

Authors:  Fulvio Braido; Francesca Sclifò; Matteo Ferrando; Giorgio Walter Canonica
Journal:  Curr Allergy Asthma Rep       Date:  2014-04       Impact factor: 4.806

2.  Effects of bilastine on T-wave morphology and the QTc interval: a randomized, double-blind, placebo-controlled, thorough QTc study.

Authors:  Claus Graff; Johannes J Struijk; Jørgen K Kanters; Mads P Andersen; Egon Toft; Benoît Tyl
Journal:  Clin Drug Investig       Date:  2012-05-01       Impact factor: 2.859

Review 3.  Bilastine: in allergic rhinitis and urticaria.

Authors:  Natalie J Carter
Journal:  Drugs       Date:  2012-06-18       Impact factor: 9.546

Review 4.  Controlled Allergen Challenge Facilities and Their Unique Contributions to Allergic Rhinitis Research.

Authors:  Michelle L North; Mena Soliman; Terry Walker; Lisa M Steacy; Anne K Ellis
Journal:  Curr Allergy Asthma Rep       Date:  2015-04       Impact factor: 4.806

5.  Comparative inhibition by bilastine and cetirizine of histamine-induced wheal and flare responses in humans.

Authors:  Martin K Church
Journal:  Inflamm Res       Date:  2011-08-28       Impact factor: 4.575

Review 6.  Ocular redness - II: Progress in development of therapeutics for the management of conjunctival hyperemia.

Authors:  Rohan Bir Singh; Lingjia Liu; Ann Yung; Sonia Anchouche; Sharad K Mittal; Tomas Blanco; Thomas H Dohlman; Jia Yin; Reza Dana
Journal:  Ocul Surf       Date:  2021-05-15       Impact factor: 6.268

7.  Bilastine: new insight into antihistamine treatment.

Authors:  Erminia Ridolo; Marcello Montagni; Laura Bonzano; Cristoforo Incorvaia; Giorgio Walter Canonica
Journal:  Clin Mol Allergy       Date:  2015-04-15

8.  Bilastine: a new nonsedating oral H1 antihistamine for treatment of allergic rhinoconjunctivitis and urticaria.

Authors:  Ole D Wolthers
Journal:  Biomed Res Int       Date:  2013-07-14       Impact factor: 3.411

9.  Critical appraisal of bilastine for the treatment of allergic rhinoconjunctivitis and urticaria.

Authors:  Belen Sadaba; Jose Ramon Azanza; Almundena Gomez-Guiu; Raquel Rodil
Journal:  Ther Clin Risk Manag       Date:  2013-05-03       Impact factor: 2.423

Review 10.  Treatment of allergic rhinitis and urticaria: a review of the newest antihistamine drug bilastine.

Authors:  Xue Yan Wang; Margaret Lim-Jurado; Narayanan Prepageran; Pongsakorn Tantilipikorn; De Yun Wang
Journal:  Ther Clin Risk Manag       Date:  2016-04-13       Impact factor: 2.423

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