Literature DB >> 19839593

Tea catechins inhibit hepatocyte growth factor receptor (MET kinase) activity in human colon cancer cells: kinetic and molecular docking studies.

Christine A Larsen1, William H Bisson, Roderick H Dashwood.   

Abstract

Most cancer deaths result from spread of the primary tumor to distant sites (metastasis). MET is an important protein for metastasis in multiple tumor types. Here we report on the ability of tea catechins to suppress MET activation in human colon cancer cells and propose a mechanism by which they might compete for the kinase domain of the MET protein.

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Year:  2009        PMID： 19839593      PMCID： PMC2784189          DOI： 10.1021/jm901330e

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


  14 in total

1.  The determination of enzyme inhibitor constants.

Authors:  M DIXON
Journal:  Biochem J       Date:  1953-08       Impact factor: 3.857

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Authors:  Chung S Yang; Shengmin Sang; Joshua D Lambert; Mao-Jung Lee
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Authors:  M Totrov; R Abagyan
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Authors:  T Cardozo; M Totrov; R Abagyan
Journal:  Proteins       Date:  1995-11

5.  A simple graphical method for determining the inhibition constants of mixed, uncompetitive and non-competitive inhibitors.

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Journal:  Biochem J       Date:  1974-01       Impact factor: 3.857

Review 6.  Tea catechins and polyphenols: health effects, metabolism, and antioxidant functions.

Authors:  Jane V Higdon; Balz Frei
Journal:  Crit Rev Food Sci Nutr       Date:  2003       Impact factor: 11.176

7.  The green tea catechins, (-)-Epigallocatechin-3-gallate (EGCG) and (-)-Epicatechin-3-gallate (ECG), inhibit HGF/Met signaling in immortalized and tumorigenic breast epithelial cells.

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Journal:  Oncogene       Date:  2006-03-23       Impact factor: 9.867

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Journal:  Med Res Rev       Date:  2008-09       Impact factor: 12.944

10.  Directed discovery of agents targeting the Met tyrosine kinase domain by virtual screening.

Authors:  Megan L Peach; Nelly Tan; Sarah J Choyke; Alessio Giubellino; Gagani Athauda; Terrence R Burke; Marc C Nicklaus; Donald P Bottaro
Journal:  J Med Chem       Date:  2009-02-26       Impact factor: 7.446
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  13 in total

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Authors:  Julio Caballero; Miguel Quiliano; Jans H Alzate-Morales; Mirko Zimic; Eric Deharo
Journal:  J Comput Aided Mol Des       Date:  2011-04-13       Impact factor: 3.686

2.  Effects of Tea Catechins on Cancer Signaling Pathways.

Authors:  Chung S Yang; Hong Wang; Jayson X Chen; Jinsong Zhang
Journal:  Enzymes       Date:  2014

3.  (-)-Epigallocatechin-3-gallate inhibits Met signaling, proliferation, and invasiveness in human colon cancer cells.

Authors:  Christine A Larsen; Roderick H Dashwood
Journal:  Arch Biochem Biophys       Date:  2010-03-31       Impact factor: 4.013

Review 4.  The chemopreventive and chemotherapeutic potentials of tea polyphenols.

Authors:  Vijay S Thakur; Karishma Gupta; Sanjay Gupta
Journal:  Curr Pharm Biotechnol       Date:  2012-01       Impact factor: 2.837

Review 5.  Tea catechins as inhibitors of receptor tyrosine kinases: mechanistic insights and human relevance.

Authors:  Christine A Larsen; Roderick H Dashwood; William H Bisson
Journal:  Pharmacol Res       Date:  2010-08-04       Impact factor: 7.658

6.  Inhibition of Eph receptor-ephrin ligand interaction by tea polyphenols.

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Journal:  Pharmacol Res       Date:  2012-06-28       Impact factor: 7.658

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8.  Ellagitannin-rich cloudberry inhibits hepatocyte growth factor induced cell migration and phosphatidylinositol 3-kinase/AKT activation in colon carcinoma cells and tumors in Min mice.

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9.  Healthy dietary patterns decrease the risk of colorectal cancer in the Mecca Region, Saudi Arabia: a case-control study.

Authors:  Firas S Azzeh; Eyad M Alshammari; Awfa Y Alazzeh; Abdelelah S Jazar; Ibrahim R Dabbour; Hani A El-Taani; Ahmed A Obeidat; Fayrooz A Kattan; Sufyan H Tashtoush
Journal:  BMC Public Health       Date:  2017-06-29       Impact factor: 3.295

10.  Epigallocatechin Gallate (EGCG) is the most effective cancer chemopreventive polyphenol in green tea.

Authors:  Guang-Jian Du; Zhiyu Zhang; Xiao-Dong Wen; Chunhao Yu; Tyler Calway; Chun-Su Yuan; Chong-Zhi Wang
Journal:  Nutrients       Date:  2012-11-08       Impact factor: 5.717
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