Literature DB >> 19449803

Synthesis of 2-aminobenzothiazole via copper(I)-catalyzed tandem reaction of 2-iodobenzenamine with isothiocyanate.

Qiuping Ding1, Xiaodan He, Jie Wu.   

Abstract

Copper(I)-catalyzed tandem reaction of 2-iodobenzenamine with isothiocyanate under mild conditions is described, which provides an efficient and practical route for the synthesis of 2-aminobenzothiazole.

Entities:  

Mesh：

Substances：

Year:  2009        PMID： 19449803     DOI： 10.1021/cc900027c

Source DB:  PubMed          Journal:  J Comb Chem        ISSN： 1520-4766


  5 in total

Review 1.  Comprehensive survey of chemical libraries for drug discovery and chemical biology: 2009.

Authors:  Roland E Dolle; Bertrand Le Bourdonnec; Karin Worm; Guillermo A Morales; Craig J Thomas; Wei Zhang
Journal:  J Comb Chem       Date:  2010-10-05

2.  Hydrothiolation of benzyl mercaptan to arylacetylene: application to the synthesis of (E) and (Z)-isomers of ON 01910·Na (Rigosertib®), a phase III clinical stage anti-cancer agent.

Authors:  Venkat R Pallela; Muralidhar R Mallireddigari; Stephen C Cosenza; Balaiah Akula; D R C Venkata Subbaiah; E Premkumar Reddy; M V Ramana Reddy
Journal:  Org Biomol Chem       Date:  2013-02-06       Impact factor: 3.876

3.  DMSO-mediated palladium-catalyzed cyclization of two isothiocyanates via C-H sulfurization: a new route to 2-aminobenzothiazoles.

Authors:  Guangkai Yao; Bing-Feng Wang; Shuai Yang; Zhi-Xiang Zhang; Han-Hong Xu; Ri-Yuan Tang
Journal:  RSC Adv       Date:  2019-01-25       Impact factor: 3.361

4.  N-[(E)-Thio-phen-2-yl-methyl-idene]-1,3-benzothia-zol-2-amine.

Authors:  Irvin N Booysen; Muhammed B Ismail; Matthew P Akerman
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2012-07-18

5.  Facile route for N 1-aryl benzotriazoles from diazoamino arynes via CuI-mediated intramolecular N-arylation.

Authors:  Raju R Kale; Virendra Prasad; H A Hussain; Vinod K Tiwari
Journal:  Tetrahedron Lett       Date:  2010-09-01       Impact factor: 2.415
  5 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.