Ju-Yeon Lee1, Yong-Chul Kim. Show Affiliations » 1. Research Center for Biomolecular Nanotechnology, Department of Life Science, Gwangju Institute of Science and Technology (GIST), 1 Oryong-dong, Buk-gu, Gwangju 500-712, Republic of Korea.
Abstract
Entities: Chemical
Mesh: See more » Amyloid Precursor Protein Secretases/antagonists & inhibitorsAmyloid Precursor Protein Secretases/metabolismAspartic Acid Endopeptidases/antagonists & inhibitorsAspartic Acid Endopeptidases/metabolismAzepines/chemical synthesisAzepines/chemistryAzepines/pharmacologyCell LineCombinatorial Chemistry TechniquesCrystallography, X-RayHumansPurinergic P2 Receptor AntagonistsReceptor, Melanocortin, Type 4/antagonists & inhibitorsReceptor, Melanocortin, Type 4/metabolismReceptors, Purinergic P2/metabolismReceptors, Purinergic P2X7Structure-Activity Relationship
Substances: See more » AzepinesP2RX7 protein, humanPurinergic P2 Receptor AntagonistsReceptor, Melanocortin, Type 4Receptors, Purinergic P2Receptors, Purinergic P2X7Amyloid Precursor Protein SecretasesAspartic Acid EndopeptidasesBACE1 protein, human
Year: 2009 PMID: 19326385 DOI: 10.1002/cmdc.200800453
Source DB: PubMed Journal: ChemMedChem ISSN: 1860-7179 Impact factor: 3.466