Literature DB >> 19058274

Pentafluorosulfanyl as a novel building block for enzyme inhibitors: trypanothione reductase inhibition and antiprotozoal activities of diarylamines.

Bernhard Stump1, Christian Eberle, W Bernd Schweizer, Marcel Kaiser, Reto Brun, R Luise Krauth-Siegel, Dieter Lentz, François Diederich.   

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Year:  2009        PMID： 19058274     DOI： 10.1002/cbic.200800565

Source DB:  PubMed          Journal:  Chembiochem        ISSN： 1439-4227            Impact factor:   3.164


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  11 in total

1.  Influence of fluorocarbon and hydrocarbon acyl groups at the surface of bovine carbonic anhydrase II on the kinetics of denaturation by sodium dodecyl sulfate.

Authors:  Andrew Lee; Katherine A Mirica; George M Whitesides
Journal:  J Phys Chem B       Date:  2010-12-23       Impact factor: 2.991

Review 2.  State of the art in African trypanosome drug discovery.

Authors:  Robert T Jacobs; Bakela Nare; Margaret A Phillips
Journal:  Curr Top Med Chem       Date:  2011       Impact factor: 3.295

3.  Discovery of practical production processes for arylsulfur pentafluorides and their higher homologues, bis- and tris(sulfur pentafluorides): Beginning of a new era of "super-trifluoromethyl" arene chemistry and its industry.

Authors:  Teruo Umemoto; Lloyd M Garrick; Norimichi Saito
Journal:  Beilstein J Org Chem       Date:  2012-03-29       Impact factor: 2.883

4.  Pyridine-promoted dediazoniation of aryldiazonium tetrafluoroborates: Application to the synthesis of SF5-substituted phenylboronic esters and iodobenzenes.

Authors:  George Iakobson; Junyi Du; Alexandra M Z Slawin; Petr Beier
Journal:  Beilstein J Org Chem       Date:  2015-08-26       Impact factor: 2.883

5.  Synthesis of Phthalocyanines with a Pentafluorosulfanyl Substituent at Peripheral Positions.

Authors:  Norihito Iida; Kenta Tanaka; Etsuko Tokunaga; Satoru Mori; Norimichi Saito; Norio Shibata
Journal:  ChemistryOpen       Date:  2015-07-24       Impact factor: 2.911

6.  Spiro-containing derivatives show antiparasitic activity against Trypanosoma brucei through inhibition of the trypanothione reductase enzyme.

Authors:  Lorenzo Turcano; Theo Battista; Esther Torrente De Haro; Antonino Missineo; Cristina Alli; Giacomo Paonessa; Gianni Colotti; Steven Harper; Annarita Fiorillo; Andrea Ilari; Alberto Bresciani
Journal:  PLoS Negl Trop Dis       Date:  2020-05-21

7.  Pentafluorosulfanyl (SF5) as a Superior 19F Magnetic Resonance Reporter Group: Signal Detection and Biological Activity of Teriflunomide Derivatives.

Authors:  Christian Prinz; Ludger Starke; Tizian-Frank Ramspoth; Janis Kerkering; Vera Martos Riaño; Jérôme Paul; Martin Neuenschwander; Andreas Oder; Silke Radetzki; Siegfried Adelhoefer; Paula Ramos Delgado; Mariya Aravina; Jason M Millward; Ariane Fillmer; Friedemann Paul; Volker Siffrin; Jens-Peter von Kries; Thoralf Niendorf; Marc Nazaré; Sonia Waiczies
Journal:  ACS Sens       Date:  2021-10-19       Impact factor: 7.711

Review 8.  Synthetic Medicinal Chemistry in Chagas' Disease: Compounds at The Final Stage of "Hit-To-Lead" Phase.

Authors:  Hugo Cerecetto; Mercedes González
Journal:  Pharmaceuticals (Basel)       Date:  2010-03-25

9.  Synthesis of kinase inhibitors containing a pentafluorosulfanyl moiety.

Authors:  Supojjanee Sansook; Cory A Ocasio; Iain J Day; Graham J Tizzard; Simon J Coles; Oleg Fedorov; James M Bennett; Jonathan M Elkins; John Spencer
Journal:  Org Biomol Chem       Date:  2017-10-18       Impact factor: 3.876

10.  Synthesis of pentafluorosulfanyl (SF5) containing aromatic amino acids.

Authors:  Lucas Grigolato; William D G Brittain; Alex S Hudson; Maria M Czyzewska; Steven L Cobb
Journal:  J Fluor Chem       Date:  2018-08       Impact factor: 2.050
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