Literature DB >> 19040385

Amorphous pharmaceutical solids: characterization, stabilization, and development of marketable formulations of poorly soluble drugs with improved oral absorption.

Ping Gao.   

Abstract

Mesh:

Year:  2008        PMID: 19040385     DOI: 10.1021/mp800203k

Source DB:  PubMed          Journal:  Mol Pharm        ISSN: 1543-8384            Impact factor:   4.939


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  11 in total

1.  Application of dissolution/permeation system for evaluation of formulation effect on oral absorption of poorly water-soluble drugs in drug development.

Authors:  Makoto Kataoka; Kiyohiko Sugano; Claudia da Costa Mathews; Jing Wen Wong; Kelly Lane Jones; Yoshie Masaoka; Shinji Sakuma; Shinji Yamashita
Journal:  Pharm Res       Date:  2011-12-02       Impact factor: 4.200

2.  Development of a Control Strategy for Benzene Impurity in HPMCAS-Stabilized Spray-Dried Dispersion Drug Products Using a Science-Based and Risk-Based Approach.

Authors:  Hongfei Yue; Sarah J Nicholson; Joel D Young; Daniel Hsieh; Rodney J Ketner; Robert G Hall; Jeremy Sackett; Elizabeth C Banks; John A Castoro; Michael E Randazzo
Journal:  Pharm Res       Date:  2015-02-28       Impact factor: 4.200

3.  Preparation, characterization and in vitro/vivo evaluation of tectorigenin solid dispersion with improved dissolution and bioavailability.

Authors:  Shuping Shuai; Shanlan Yue; Qingting Huang; Wei Wang; Junyi Yang; Ke Lan; Liming Ye
Journal:  Eur J Drug Metab Pharmacokinet       Date:  2015-02-11       Impact factor: 2.441

4.  In vitro and in vivo evaluation of amorphous solid dispersions generated by different bench-scale processes, using griseofulvin as a model compound.

Authors:  Po-Chang Chiang; Yong Cui; Yingqing Ran; Joe Lubach; Kang-Jye Chou; Linda Bao; Wei Jia; Hank La; Jonathan Hau; Amy Sambrone; Ann Qin; Yuzhong Deng; Harvey Wong
Journal:  AAPS J       Date:  2013-03-02       Impact factor: 4.009

5.  A Model-Based Methodology for Spray-Drying Process Development.

Authors:  Dan E Dobry; Dana M Settell; John M Baumann; Rod J Ray; Lisa J Graham; Ron A Beyerinck
Journal:  J Pharm Innov       Date:  2009-07-25       Impact factor: 2.750

6.  In vitro characterization of a novel polymeric system for preparation of amorphous solid drug dispersions.

Authors:  Zahra N Mahmoudi; Sampada B Upadhye; David Ferrizzi; Ali R Rajabi-Siahboomi
Journal:  AAPS J       Date:  2014-05-02       Impact factor: 4.009

7.  Acid-responsive nanospheres from an asparagine-derived amphiphile.

Authors:  Adelphe M Mfuh; Mathew P D Mahindaratne; Audrey E Yñigez-Gutierrez; Juan R Ramos Dominguez; Jefferson T Bedell; Carlos D Garcia; George R Negrete
Journal:  RSC Adv       Date:  2015       Impact factor: 3.361

8.  Evaluation of drug load and polymer by using a 96-well plate vacuum dry system for amorphous solid dispersion drug delivery.

Authors:  Po-Chang Chiang; Yingqing Ran; Kang-Jye Chou; Yong Cui; Amy Sambrone; Connie Chan; Ryan Hart
Journal:  AAPS PharmSciTech       Date:  2012-05-05       Impact factor: 3.246

9.  Density Functional Theory in the Prediction of Mutagenicity: A Perspective.

Authors:  Piers A Townsend; Matthew N Grayson
Journal:  Chem Res Toxicol       Date:  2020-08-07       Impact factor: 3.739

Review 10.  Using X-ray Diffraction Techniques for Biomimetic Drug Development, Formulation, and Polymorphic Characterization.

Authors:  Israel Rodríguez; Ritika Gautam; Arthur D Tinoco
Journal:  Biomimetics (Basel)       Date:  2020-12-30
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