Literature DB >> 18842404

One-pot synthesis and antibacterial activities of pyrazolo[4',3':5,6]pyrido[2,3-d]pyrimidine-dione derivatives.

Ayoob Bazgir1, Maryam Mohammadi Khanaposhtani, Ali Abolhasani Soorki.   

Abstract

A one-pot and efficient method for the synthesis of pyrazolo[4',3':5,6]pyrido[2,3-d]pyrimidine-dione derivatives by condensation reaction of barbituric acids, 1H-pyrazol-5-amines and aldehydes under solvent-free conditions is reported. These products were evaluated in vitro for their antibacterial activities.

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Year:  2008        PMID： 18842404     DOI： 10.1016/j.bmcl.2008.09.057

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN： 0960-894X            Impact factor:   2.823


  6 in total

1.  Design and synthesis of new imidazo[1,2-b]pyrazole derivatives, in vitro α-glucosidase inhibition, kinetic and docking studies.

Authors:  Fariba Peytam; Mehdi Adib; Reihaneh Shourgeshty; Maryam Mohammadi-Khanaposhtani; Mehdi Jahani; Somaye Imanparast; Mohammad Ali Faramarzi; Mohammad Mahdavi; Ali Akbar Moghadamnia; Hossein Rastegar; Bagher Larijani
Journal:  Mol Divers       Date:  2019-03-02       Impact factor: 2.943

2.  Grindstone Chemistry: Design, One-Pot Synthesis, and Promising Anticancer Activity of Spiro[acridine-9,2'-indoline]-1,3,8-trione Derivatives against the MCF-7 Cancer Cell Line.

Authors:  Perumal Gobinath; Ponnusamy Packialakshmi; Ali Daoud; Saud Alarifi; Akbar Idhayadhulla; Surendrakumar Radhakrishnan
Journal:  Molecules       Date:  2020-12-11       Impact factor: 4.411

3.  Synthesis, characterization, molecular docking, and anticancer activities of new 1,3,4-oxadiazole-5-fluorocytosine hybrid derivatives.

Authors:  Az-Eddine El Mansouri; Saida Lachhab; Ali Oubella; Mehdi Ahmad; Johan Neyts; Dirk Jochmans; Winston Chiu; Laura Vangeel; Steven De Jonghe; Hamid Morjani; Mustapha Ait Ali; Mohamed Zahouily; Yogesh S Sanghvi; Hassan B Lazrek
Journal:  J Mol Struct       Date:  2022-09-09       Impact factor: 3.841

4.  Crystal structure of (E)-N-{[3-methyl-1-phenyl-5-(1H-pyrrol-1-yl)-1H-pyrazol-4-yl]methyl-idene}hydroxyl-amine.

Authors:  Joel T Mague; Shaaban K Mohamed; Mehmet Akkurt; Talaat I El-Emary; Mustafa R Albayati
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2014-10-31

5.  Microwave assisted synthesis of some new thiazolopyrimidine and pyrimidothiazolopyrimidopyrimidine derivatives with potential antimicrobial activity.

Authors:  Ayman M S Youssef; Ahmed M Fouda; Rasha M Faty
Journal:  Chem Cent J       Date:  2018-05-05       Impact factor: 4.215

6.  Multi-component one-pot synthesis and antimicrobial activities of 3-methyl-1,4-diphenyl-7-thioxo-4,6,8,9-tetrahydro-pyrazolo[5,4-b]pyrimidino[5,4-e]pyridine-5-one and related derivatives.

Authors:  Talaat I El-Emary; Shawkat A Abd El-Mohsen
Journal:  Molecules       Date:  2012-12-06       Impact factor: 4.411
  6 in total

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