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10 in total

1. Derivatives of (phenylsulfonamido-methyl)nicotine and (phenylsulfonamido-methyl)thiazole as novel 11beta-hydroxysteroid dehydrogenase type 1 inhibitors: synthesis and biological activities in vitro.

Authors: Xu Zhang; Yang Zhou; Yu Shen; Li-li Du; Jun-hua Chen; Ying Leng; Jian-hua Shen
Journal: Acta Pharmacol Sin Date: 2009-08-24 Impact factor: 6.150

2. Optimization of 1,2,4-Triazolopyridines as Inhibitors of Human 11β-Hydroxysteroid Dehydrogenase Type 1 (11β-HSD-1).

Authors: Jun Li; Lawrence J Kennedy; Haixia Wang; James J Li; Steven J Walker; Zhenqiu Hong; Stephen P O'Connor; Akbar Nayeem; Daniel M Camac; Paul E Morin; Steven Sheriff; Mengmeng Wang; Timothy Harper; Rajasree Golla; Ramakrishna Seethala; Thomas Harrity; Randolph P Ponticiello; Nathan N Morgan; Joseph R Taylor; Rachel Zebo; David A Gordon; Jeffrey A Robl
Journal: ACS Med Chem Lett Date: 2014-05-22 Impact factor: 4.345

3. Ethyl 2-{(2Z)-2-[(1-naphthyl-sulfon-yl)imino]-2,3-dihydro-1,3-thia-zol-4-yl}acetate monohydrate.

Authors: Gabriel Navarrete-Vázquez; Guadalupe Morales-Vilchis; Samuel Estrada-Soto; Verónica Rodríguez-López; Hugo Tlahuext
Journal: Acta Crystallogr Sect E Struct Rep Online Date: 2010-10-09

Review 4. Current and future drug targets in weight management.

Authors: Renger F Witkamp
Journal: Pharm Res Date: 2010-12-23 Impact factor: 4.200

5. Discovery of adamantyl heterocyclic ketones as potent 11β-hydroxysteroid dehydrogenase type 1 inhibitors.

Authors: Xiangdong Su; Nigel Vicker; Mark P Thomas; Fabienne Pradaux-Caggiano; Heather Halem; Michael D Culler; Barry V L Potter
Journal: ChemMedChem Date: 2011-05-23 Impact factor: 3.466

6. Adamantyl ethanone pyridyl derivatives: potent and selective inhibitors of human 11β-hydroxysteroid dehydrogenase type 1.

Authors: Xiangdong Su; Fabienne Pradaux-Caggiano; Nigel Vicker; Mark P Thomas; Heather Halem; Michael D Culler; Barry V L Potter
Journal: ChemMedChem Date: 2011-06-28 Impact factor: 3.466

7. The regioselective synthesis of spirooxindolo pyrrolidines and pyrrolizidines via three-component reactions of acrylamides and aroylacrylic acids with isatins and α-amino acids.

Authors: Tatyana L Pavlovskaya; Fedor G Yaremenko; Victoria V Lipson; Svetlana V Shishkina; Oleg V Shishkin; Vladimir I Musatov; Alexander S Karpenko
Journal: Beilstein J Org Chem Date: 2014-01-09 Impact factor: 2.883

8. An inhibitor of 11-β hydroxysteroid dehydrogenase type 1 (PF915275) alleviates nonylphenol-induced hyperadrenalism and adiposity in rat and human cells.

Authors: Ling-Ling Chang; Wan-Song Alfred Wun; Paulus S Wang
Journal: BMC Pharmacol Toxicol Date: 2018-07-18 Impact factor: 2.483

9. Synthesis of Novel 2-(Isopropylamino)thiazol-4(5H)-one Derivatives and Their Inhibitory Activity of 11β-HSD1 and 11β-HSD2 in Aspect of Carcinogenesis Prevention.

Authors: Daria Kupczyk; Renata Studzińska; Rafał Bilski; Szymon Baumgart; Renata Kołodziejska; Alina Woźniak
Journal: Molecules Date: 2020-09-15 Impact factor: 4.411

10. Adamantyl carboxamides and acetamides as potent human 11β-hydroxysteroid dehydrogenase type 1 inhibitors.

Authors: Xiangdong Su; Heather A Halem; Mark P Thomas; Cecile Moutrille; Michael D Culler; Nigel Vicker; Barry V L Potter
Journal: Bioorg Med Chem Date: 2012-09-12 Impact factor: 3.641

10 in total