Literature DB >> 18393489

Synthesis of indoleamine 2,3-dioxygenase inhibitory analogues of the sponge alkaloid exiguamine A.

Gavin Carr1, Marco K W Chung, A Grant Mauk, Raymond J Andersen.   

Abstract

Synthetic analogues of the sponge natural product exiguamine A (3) have been prepared and evaluated for their ability to inhibit indoleamine 2,3-dioxygenase in vitro.

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Year:  2008        PMID: 18393489     DOI: 10.1021/jm800143h

Source DB:  PubMed          Journal:  J Med Chem        ISSN: 0022-2623            Impact factor:   7.446


  13 in total

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