Literature DB >> 18079987

Synthesis of oxazolidinedione derived bicalutamide analogs.

Vipin A Nair1, Suni M Mustafa, Michael L Mohler, James T Dalton, Duane D Miller.   

Abstract

The synthesis of chiral oxazolidinedione derived bicalutamide analogs has been discussed.

Entities:  

Year:  2006        PMID： 18079987      PMCID： PMC2134919          DOI： 10.1016/j.tetlet.2006.03.146

Source DB:  PubMed          Journal:  Tetrahedron Lett        ISSN： 0040-4039            Impact factor:   2.415


  12 in total

1.  Homology modeling using multiple molecular dynamics simulations and docking studies of the human androgen receptor ligand binding domain bound to testosterone and nonsteroidal ligands.

Authors:  C A Marhefka; B M Moore; T C Bishop; L Kirkovsky; A Mukherjee; J T Dalton; D D Miller
Journal:  J Med Chem       Date:  2001-05-24       Impact factor: 7.446

2.  Synthesis of irreversibly binding bicalutamide analogs for imaging studies.

Authors:  Vipin A Nair; Suni M Mustafa; Michael L Mohler; Jun Yang; Leonid I Kirkovsky; James T Dalton; Duane D Miller
Journal:  Tetrahedron Lett       Date:  2005-07-11       Impact factor: 2.415

3.  Discovery of nonsteroidal androgens.

Authors:  J T Dalton; A Mukherjee; Z Zhu; L Kirkovsky; D D Miller
Journal:  Biochem Biophys Res Commun       Date:  1998-03-06       Impact factor: 3.575

4.  Structural basis for antagonism and resistance of bicalutamide in prostate cancer.

Authors:  Casey E Bohl; Wenqing Gao; Duane D Miller; Charles E Bell; James T Dalton
Journal:  Proc Natl Acad Sci U S A       Date:  2005-04-15       Impact factor: 11.205

5.  Affinity labeling of the androgen receptor with nonsteroidal chemoaffinity ligands.

Authors:  A Mukherjee; L I Kirkovsky; Y Kimura; M M Marvel; D D Miller; J T Dalton
Journal:  Biochem Pharmacol       Date:  1999-10-15       Impact factor: 5.858

6.  Chiral nonsteroidal affinity ligands for the androgen receptor. 1. Bicalutamide analogues bearing electrophilic groups in the B aromatic ring.

Authors:  L Kirkovsky; A Mukherjee; D Yin; J T Dalton; D D Miller
Journal:  J Med Chem       Date:  2000-02-24       Impact factor: 7.446

7.  Pharmacodynamics of selective androgen receptor modulators.

Authors:  Donghua Yin; Wenqing Gao; Jeffrey D Kearbey; Huiping Xu; Kiwon Chung; Yali He; Craig A Marhefka; Karen A Veverka; Duane D Miller; James T Dalton
Journal:  J Pharmacol Exp Ther       Date:  2003-03       Impact factor: 4.030

8.  A selective androgen receptor modulator for hormonal male contraception.

Authors:  Jiyun Chen; Dong Jin Hwang; Casey E Bohl; Duane D Miller; James T Dalton
Journal:  J Pharmacol Exp Ther       Date:  2004-09-03       Impact factor: 4.030

9.  A ligand-based approach to identify quantitative structure-activity relationships for the androgen receptor.

Authors:  Casey E Bohl; Cheng Chang; Michael L Mohler; Jiyun Chen; Duane D Miller; Peter W Swaan; James T Dalton
Journal:  J Med Chem       Date:  2004-07-15       Impact factor: 7.446

10.  Comparison of the pharmacological effects of a novel selective androgen receptor modulator, the 5alpha-reductase inhibitor finasteride, and the antiandrogen hydroxyflutamide in intact rats: new approach for benign prostate hyperplasia.

Authors:  Wenqing Gao; Jeffrey D Kearbey; Vipin A Nair; Kiwon Chung; A F Parlow; Duane D Miller; James T Dalton
Journal:  Endocrinology       Date:  2004-08-12       Impact factor: 4.736
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