Literature DB >> 17997304

Thiophene containing triarylmethanes as antitubercular agents.

Maloy Kumar Parai1, Gautam Panda, Vinita Chaturvedi, Y K Manju, Sudhir Sinha.   

Abstract

A new series of thiophene containing triarylmethane derivatives were synthesized from the Friedel-Crafts alkylation of diarylcarbinols followed by incorporation of amino alkyl chains. These were evaluated against Mycobacterium tuberculosis H37R(v) and showed the activity in the range of 3.12-12.5 microg/mL in vitro.

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Year:  2007        PMID： 17997304     DOI： 10.1016/j.bmcl.2007.10.083

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN： 0960-894X            Impact factor:   2.823


  22 in total

1.  SbCl(3)-catalyzed one-pot synthesis of 4,4'-diaminotriarylmethanes under solvent-free conditions: Synthesis, characterization, and DFT studies.

Authors:  Ghasem Rezanejade Bardajee
Journal:  Beilstein J Org Chem       Date:  2011-01-31       Impact factor: 2.883

2.  Retention or inversion in stereospecific nickel-catalyzed cross-coupling of benzylic carbamates with arylboronic esters: control of absolute stereochemistry with an achiral catalyst.

Authors:  Michael R Harris; Luke E Hanna; Margaret A Greene; Curtis E Moore; Elizabeth R Jarvo
Journal:  J Am Chem Soc       Date:  2013-02-22       Impact factor: 15.419

3.  Asymmetric transition metal-catalyzed cross-coupling reactions for the construction of tertiary stereocenters.

Authors:  Elizabeth C Swift; Elizabeth R Jarvo
Journal:  Tetrahedron       Date:  2013-07-22       Impact factor: 2.457

4.  Selective synthesis of either enantiomer of an anti-breast cancer agent via a common enantioenriched intermediate.

Authors:  Aaron George Johnson; Marissa M Tranquilli; Michael R Harris; Elizabeth R Jarvo
Journal:  Tetrahedron Lett       Date:  2015-06-03       Impact factor: 2.415

5.  Synthesis of Triarylmethanes via Palladium-Catalyzed Suzuki-Miyaura Reactions of Diarylmethyl Esters.

Authors:  Amira H Dardir; Irene Casademont-Reig; David Balcells; Jonathan D Ellefsen; Matthew R Espinosa; Nilay Hazari; Nicholas E Smith
Journal:  Organometallics       Date:  2021-05-27       Impact factor: 3.837

6.  Synthesis and antimicrobial studies of some novel bis-[1,3,4]thiadiazole and bis-thiazole pendant to thieno[2,3-b]thiophene moiety.

Authors:  Nabila Abdelshafy Kheder; Yahia Nasser Mabkhot
Journal:  Int J Mol Sci       Date:  2012-03-19       Impact factor: 6.208

7.  Crystal structures and conformations of two Diels-Alder adduct derivatives: 1,8-bis-(thio-phen-2-yl)-14-oxa-tetra-cyclo-[6.5.1.0(2,7).0(9,13)]tetra-deca-2(7),3,5-trien-10-one and 1,8-diphenyl-14-oxa-tetra-cyclo[6.5.1.0(2,7).0(9,13)] tetra-deca-2,4,6-trien-10-one.

Authors:  S Gopinath; P Narayanan; K Sethusankar; Meganathan Nandakumar; Arasambattu K Mohanakrishnan
Journal:  Acta Crystallogr E Crystallogr Commun       Date:  2015-01-24

8.  Transition-Metal-Free Synthesis of Polyfunctional Triarylmethanes and 1,1-Diarylalkanes by Sequential Cross-Coupling of Benzal Diacetates with Organozinc Reagents.

Authors:  Baosheng Wei; Qianyi Ren; Thomas Bein; Paul Knochel
Journal:  Angew Chem Int Ed Engl       Date:  2021-03-17       Impact factor: 15.336

9.  NiXantphos: a deprotonatable ligand for room-temperature palladium-catalyzed cross-couplings of aryl chlorides.

Authors:  Jiadi Zhang; Ana Bellomo; Nisalak Trongsiriwat; Tiezheng Jia; Patrick J Carroll; Spencer D Dreher; Matthew T Tudge; Haolin Yin; Jerome R Robinson; Eric J Schelter; Patrick J Walsh
Journal:  J Am Chem Soc       Date:  2014-04-21       Impact factor: 15.419

10.  Facile synthesis and antimicrobial evaluation of some new heterocyclic compounds incorporating a biologically active sulfamoyl moiety.

Authors:  Elham S Darwish
Journal:  ScientificWorldJournal       Date:  2014-08-17
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