Literature DB >> 17532702

Safety and tolerability of acarbose in the treatment of type 1 and type 2 diabetes mellitus.

Dieter Neuser1, Alice Benson, Andreas Brückner, Ronald B Goldberg, Byron J Hoogwerf, Dieter Petzinna.   

Abstract

OBJECTIVE: To assess the safety profile of acarbose treatment over a 1-year period at a dose range of 50-300mg three times daily in patients with type 1 or type 2 diabetes mellitus. STUDY DESIGN AND PATIENTS: In this 56-week, double-blind, parallel-group, multicentre comparison, patients were randomised to acarbose or placebo in a 2 : 1 ratio. An 8-week forced titration phase (from 50-300mg three times daily) was followed by a 48-week maintenance phase during which patients received the highest dose tolerated during titration. Patients were assessed at 13 visits with respect to adverse events/intercurrent illnesses, abnormal laboratory values (serum chemistry, urinalysis, complete blood and reticulocyte count, serum iron and total iron binding capacity, and serum vitamin B(6), B(12), D and folate levels), discontinuation rates, ECG findings, vital signs and evaluation of the patients' diaries with regard to gastrointestinal events. A total of 359 patients (acarbose 240, placebo 119) were valid for analysis; 21% had type 1 diabetes. Most patients received concomitant insulin or sulfonylurea treatment.
RESULTS: Study withdrawal was reported for 35% of acarbose and 24% of placebo recipients (p = 0.053); adverse events were the main reason for withdrawal in acarbose recipients (20%; placebo group 5%; p < 0.01). The most common adverse events for acarbose recipients were gastrointestinal (abdominal pain, flatulence and diarrhoea), which were more frequent than in placebo patients (p < 0.01). These events occurred more often early in the study and attenuated over time.
CONCLUSION: Acarbose was safe and well tolerated by the majority of diabetic patients over a 1-year treatment period.

Entities:  

Year:  2005        PMID: 17532702     DOI: 10.2165/00044011-200525090-00003

Source DB:  PubMed          Journal:  Clin Drug Investig        ISSN: 1173-2563            Impact factor:   2.859


  19 in total

1.  Efficacy and safety of acarbose in the treatment of Type 1 diabetes mellitus: a placebo-controlled, double-blind, multicentre study.

Authors:  G Riccardi; R Giacco; M Parillo; S Turco; A A Rivellese; M R Ventura; S Contadini; G Marra; M Monteduro; F Santeusanio; P Brunetti; M C Librenti; A E Pontiroli; P Vedani; G Pozza; L Bergamini; C Bianchi
Journal:  Diabet Med       Date:  1999-03       Impact factor: 4.359

2.  Acarbose in the treatment of type I diabetes.

Authors:  P Hollander; X Pi-Sunyer; R F Coniff
Journal:  Diabetes Care       Date:  1997-03       Impact factor: 19.112

Review 3.  Acarbose: a review of US clinical experience.

Authors:  R Coniff; A Krol
Journal:  Clin Ther       Date:  1997 Jan-Feb       Impact factor: 3.393

4.  Reduction of glycosylated hemoglobin and postprandial hyperglycemia by acarbose in patients with NIDDM. A placebo-controlled dose-comparison study.

Authors:  R F Coniff; J A Shapiro; D Robbins; R Kleinfield; T B Seaton; P Beisswenger; J B McGill
Journal:  Diabetes Care       Date:  1995-06       Impact factor: 19.112

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6.  Effects of acarbose (Glucobay) in persons with type 1 diabetes: a multicentre study.

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7.  Acarbose for prevention of type 2 diabetes mellitus: the STOP-NIDDM randomised trial.

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Review 8.  Safety profile of acarbose, an alpha-glucosidase inhibitor.

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9.  The efficacy of acarbose in the treatment of patients with non-insulin-dependent diabetes mellitus. A multicenter controlled clinical trial.

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Authors: 
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