Mark J Field1, Zheng Li, Jacob B Schwarz. Show Affiliations » 1. Pfizer Global Research and Development, Sandwich Laboratories, Sandwich, Kent CT13 9NJ, UK.
Abstract
Entities: Disease
Mesh: See more » Amines/chemistryAmines/pharmacologyAmines/therapeutic useAnalgesics/chemistryAnalgesics/pharmacologyAnalgesics/therapeutic useAnimalsAnticonvulsants/chemistryAnticonvulsants/pharmacologyAnticonvulsants/therapeutic useCalcium Channels/geneticsCalcium Channels/metabolismCalcium Channels/physiologyCarboxylic Acids/chemistryCarboxylic Acids/pharmacologyCarboxylic Acids/therapeutic useCyclohexanecarboxylic Acids/chemistryCyclohexanecarboxylic Acids/pharmacologyCyclohexanecarboxylic Acids/therapeutic useGabapentinHumansLigandsMiceMice, Mutant StrainsPain/drug therapyPain/metabolismPeripheral Nervous System Diseases/drug therapyPeripheral Nervous System Diseases/metabolismPeripheral Nervous System Diseases/physiopathologyPregabalinProdrugs/chemistryProdrugs/pharmacologyProdrugs/therapeutic usegamma-Aminobutyric Acid/analogs & derivativesgamma-Aminobutyric Acid/chemistrygamma-Aminobutyric Acid/pharmacologygamma-Aminobutyric Acid/therapeutic use
Substances: See more » AminesAnalgesicsAnticonvulsantsCalcium ChannelsCarboxylic AcidsCyclohexanecarboxylic AcidsLigandsProdrugsvoltage gated calcium channel subunit Ca alpha2delta-1, humanPregabalingamma-Aminobutyric AcidGabapentin
Year: 2007 PMID: 17489571 DOI: 10.1021/jm060650z
Source DB: PubMed Journal: J Med Chem ISSN: 0022-2623 Impact factor: 7.446