Literature DB >> 16983056

A double-blind, placebo-controlled, crossover study of sildenafil in obstructive sleep apnea.

Suely Roizenblatt1, Christian Guilleminault, Dalva Poyares, Fátima Cintra, Adriana Kauati, Sergio Tufik.   

Abstract

BACKGROUND: Sildenafil prolongs the action of cyclic guanosine monophosphate and nitric oxide by inhibiting cyclic guanosine monophosphate-specific phosphodiesterase 5. It is largely used for erectile dysfunction, a highly prevalent condition in obstructive sleep apnea. Because nitric oxide promotes upper airway congestion, muscle relaxation, and pulmonary vasodilation, the aim of this study was to establish the impact of a single 50-mg dose of sildenafil on the sleep of patients with severe obstructive sleep apnea.
METHODS: Thirteen [corrected] middle-aged men with severe obstructive sleep apnea were consecutively selected for this double-blind, placebo-controlled, crossover study. Exclusion criteria were obesity, cardiovascular and/or respiratory disease, and conditions that interfere with sleep. All-night polysomnography was preceded by a single 50-mg dose of sildenafil or matching placebo randomly administered at bedtime, after a washout period of 1 week.
RESULTS: In comparison to placebo, a single 50-mg dose of sildenafil significantly increased the percentage of total sleep time with an arterial oxygen saturation of less than 90% (mean +/- SD, 15.6% +/- 9.6% vs 7.9% +/- 3.3%, [corrected] P < .01), without a difference in the nadir of oxygen desaturation. The mean arterial oxygen saturation also decreased (92.1% +/- 1.9% vs 93.8% +/- 1.3%, P = .03), [corrected] and the desaturation index increased (30.3 +/- 14.5 [corrected] events per hour vs 18.5 +/- 9.1 [corrected] events per hour, P < .001). There was an increase in apnea-hypopnea index (48.1 +/- 20.8 [corrected] events per hour vs 32.3 +/- 11.3 [corrected] events per hour, P = .001), [corrected] involving mostly obstructive events.
CONCLUSION: In patients with severe obstructive sleep apnea, a single 50-mg dose of sildenafil at bedtime worsens respiratory and desaturation events.

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Year:  2006        PMID: 16983056     DOI: 10.1001/archinte.166.16.1763

Source DB:  PubMed          Journal:  Arch Intern Med        ISSN: 0003-9926


  10 in total

1.  The Effects of Sildenafil on the Respiratory System of Patients With Obstructive Sleep Apnea and Erectile Dysfunction.

Authors:  Monica L Andersen; Sergio Tufik
Journal:  J Clin Sleep Med       Date:  2018-05-15       Impact factor: 4.062

2.  Systemic and metabolic effects of PDE5-inhibitor drugs.

Authors:  Antonio Aversa
Journal:  World J Diabetes       Date:  2010-03-15

3.  Testosterone and phosphodiesterase type-5 inhibitors: new strategy for preventing endothelial damage in internal and sexual medicine?

Authors:  Antonio Aversa; Roberto Bruzziches; Davide Francomano; Marco Natali; Andrea Lenzi
Journal:  Ther Adv Urol       Date:  2009-10

4.  Effects of sildenafil on autonomic nervous function during sleep in obstructive sleep apnea.

Authors:  Christiane Neves; Sérgio Tufik; Felipe Chediek; Dalva Poyares; Fátima Cintra; Marina Roizenblatt; Fabiano Abrantes; Marina Ariza Monteiro; Suely Roizenblatt
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5.  Sleep dysfunction in heart failure.

Authors:  Shahrokh Javaheri
Journal:  Curr Treat Options Neurol       Date:  2008-09       Impact factor: 3.598

Review 6.  Obstructive sleep apnea and erectile dysfunction: still a neglected risk factor?

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Journal:  Sleep Breath       Date:  2008-09-03       Impact factor: 2.816

7.  cGMP-phosphodiesterase inhibition enhances photic responses and synchronization of the biological circadian clock in rodents.

Authors:  Santiago A Plano; Patricia V Agostino; Horacio O de la Iglesia; Diego A Golombek
Journal:  PLoS One       Date:  2012-05-10       Impact factor: 3.240

8.  Erectile Dysfunction in Patients with Sleep Apnea--A Nationwide Population-Based Study.

Authors:  Chia-Min Chen; Ming-Ju Tsai; Po-Ju Wei; Yu-Chung Su; Chih-Jen Yang; Meng-Ni Wu; Chung-Yao Hsu; Shang-Jyh Hwang; Inn-Wen Chong; Ming-Shyan Huang
Journal:  PLoS One       Date:  2015-07-15       Impact factor: 3.240

Review 9.  Effects of obstructive sleep apnea and its treatment over the erectile function: a systematic review.

Authors:  Felix Campos-Juanatey; Marcos Fernandez-Barriales; Monica Gonzalez; Jose A Portillo-Martin
Journal:  Asian J Androl       Date:  2017 May-Jun       Impact factor: 3.285

10.  Efficacy and safety of oral sildenafil in children with Down syndrome and pulmonary hypertension.

Authors:  Maurice Beghetti; Andrzej Rudzinski; Min Zhang
Journal:  BMC Cardiovasc Disord       Date:  2017-07-04       Impact factor: 2.298

  10 in total

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