Literature DB >> 16895328

Mechanism-based profiling of enzyme families.

Michael J Evans1, Benjamin F Cravatt.   

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Year:  2006        PMID: 16895328     DOI: 10.1021/cr050288g

Source DB:  PubMed          Journal:  Chem Rev        ISSN: 0009-2665            Impact factor:   60.622


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  138 in total

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2.  Activity-based protein profiling identifies a host enzyme, carboxylesterase 1, which is differentially active during hepatitis C virus replication.

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Review 4.  Choosing an effective protein bioconjugation strategy.

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Journal:  Nat Chem Biol       Date:  2011-11-15       Impact factor: 15.040

5.  Activity-based protein profiling of protein arginine methyltransferase 1.

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6.  Strategies for discovering and derisking covalent, irreversible enzyme inhibitors.

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Journal:  Future Med Chem       Date:  2010-06       Impact factor: 3.808

7.  The Natural Product Elegaphenone Potentiates Antibiotic Effects against Pseudomonas aeruginosa.

Authors:  Weining Zhao; Ashley R Cross; Caillan Crowe-McAuliffe; Angela Weigert-Munoz; Erika E Csatary; Amy E Solinski; Joanna Krysiak; Joanna B Goldberg; Daniel N Wilson; Eva Medina; William M Wuest; Stephan A Sieber
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8.  Inhibition of serine proteases by a new class of cyclosulfamide-based carbamylating agents.

Authors:  Qingliang Yang; Yi Li; Dengfeng Dou; Xiangdong Gan; Swathi Mohan; Christopher S Groutas; Laura E Stevenson; Zhong Lai; Kevin R Alliston; Jiaying Zhong; Todd D Williams; William C Groutas
Journal:  Arch Biochem Biophys       Date:  2008-04-22       Impact factor: 4.013

9.  Rational design of fatty acid amide hydrolase inhibitors that act by covalently bonding to two active site residues.

Authors:  Katerina Otrubova; Monica Brown; Michael S McCormick; Gye W Han; Scott T O'Neal; Benjamin F Cravatt; Raymond C Stevens; Aron H Lichtman; Dale L Boger
Journal:  J Am Chem Soc       Date:  2013-04-12       Impact factor: 15.419

10.  Chemical probes identify a role for histone deacetylase 3 in Friedreich's ataxia gene silencing.

Authors:  Chunping Xu; Elisabetta Soragni; C James Chou; David Herman; Heather L Plasterer; James R Rusche; Joel M Gottesfeld
Journal:  Chem Biol       Date:  2009-09-25
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