Literature DB >> 16880176

In vitro activity of a new antibacterial rhodanine derivative against Staphylococcus epidermidis biofilms.

Maxime Gualtieri1, Lionel Bastide, Philippe Villain-Guillot, Sylvie Michaux-Charachon, Jaqueline Latouche, Jean-Paul Leonetti.   

Abstract

OBJECTIVES: Staphylococcus epidermidis biofilms form at the surface of implants and prostheses and are responsible for the failure of many antibiotic therapies. Only a few antibiotics are relatively active against biofilms, and rifampicin, a transcription inhibitor, is among the most effective molecules for treating biofilm-related infections. Having recently selected a new potential transcription inhibitor, we attempted to evaluate its efficacy against S. epidermidis biofilms.
METHODS: Biofilm-forming S. epidermidis strains were grown planktonically or as biofilms and their susceptibility to this transcription inhibitor was compared with reference antibiotics with different mechanisms of action.
CONCLUSIONS: Our results demonstrate that this new molecule is active; its effects are fast and kinetically related to those of rifampicin, but unlike rifampicin it does not select for resistant bacteria.

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Year:  2006        PMID: 16880176     DOI: 10.1093/jac/dkl314

Source DB:  PubMed          Journal:  J Antimicrob Chemother        ISSN: 0305-7453            Impact factor:   5.790


  6 in total

1.  Selective killing of nonreplicating mycobacteria.

Authors:  Ruslana Bryk; Benjamin Gold; Aditya Venugopal; Jasbir Singh; Raghu Samy; Krzysztof Pupek; Hua Cao; Carmen Popescu; Mark Gurney; Srinivas Hotha; Joseph Cherian; Kyu Rhee; Lan Ly; Paul J Converse; Sabine Ehrt; Omar Vandal; Xiuju Jiang; Jean Schneider; Gang Lin; Carl Nathan
Journal:  Cell Host Microbe       Date:  2008-03-13       Impact factor: 21.023

2.  In vitro activities of different inhibitors of bacterial transcription against Staphylococcus epidermidis biofilm.

Authors:  Philippe Villain-Guillot; Maxime Gualtieri; Lionel Bastide; Jean-Paul Leonetti
Journal:  Antimicrob Agents Chemother       Date:  2007-07-02       Impact factor: 5.191

3.  Evaluation of antimicrobial activity of certain combinations of antibiotics against in vitro Staphylococcus epidermidis biofilms.

Authors:  Fernanda Gomes; Pilar Teixeira; Howard Ceri; Rosário Oliveira
Journal:  Indian J Med Res       Date:  2012-04       Impact factor: 2.375

4.  Antibiotic susceptibility of coagulase-negative staphylococci isolated from very low birth weight babies: comprehensive comparisons of bacteria at different stages of biofilm formation.

Authors:  Yue Qu; Andrew J Daley; Taghrid S Istivan; Suzanne M Garland; Margaret A Deighton
Journal:  Ann Clin Microbiol Antimicrob       Date:  2010-05-27       Impact factor: 3.944

5.  Synthesis and Antibacterial Evaluation of (S,Z)-4-methyl-2-(4-oxo-5-((5-substituted phenylfuran-2-yl) methylene)-2-thioxothiazolidin-3-yl)Pentanoic Acids.

Authors:  Ming-Xia Song; Xian-Qing Deng; Zhi-Yu Wei; Chang-Ji Zheng; Yan Wu; Chang-Shan An; Hu-Ri Piao
Journal:  Iran J Pharm Res       Date:  2015       Impact factor: 1.696

6.  Synthesis and Biological Evaluation of Novel Fusidic Acid Derivatives as Two-in-One Agent with Potent Antibacterial and Anti-Inflammatory Activity.

Authors:  Borong Tu; Nana Cao; Bingjie Zhang; Wende Zheng; Jiahao Li; Xiaowen Tang; Kaize Su; Jinxuan Li; Zhen Zhang; Zhenping Yan; Dongli Li; Xi Zheng; Kun Zhang; Weiqian David Hong; Panpan Wu
Journal:  Antibiotics (Basel)       Date:  2022-07-30
  6 in total

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