Literature DB >> 16708409

Rapid identification of potent nonpeptidic serine protease inhibitors.

Cleo M Salisbury1, Jonathan A Ellman.   

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Year:  2006        PMID： 16708409     DOI： 10.1002/cbic.200600081

Source DB:  PubMed          Journal:  Chembiochem        ISSN： 1439-4227            Impact factor:   3.164


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  7 in total

Review 1.  The pharmacological landscape and therapeutic potential of serine hydrolases.

Authors:  Daniel A Bachovchin; Benjamin F Cravatt
Journal:  Nat Rev Drug Discov       Date:  2012-01-03       Impact factor: 84.694

Review 2.  Using specificity to strategically target proteases.

Authors:  Mark D Lim; Charles S Craik
Journal:  Bioorg Med Chem       Date:  2008-03-30       Impact factor: 3.641

3.  Fragment-based discovery of selective inhibitors of the Mycobacterium tuberculosis protein tyrosine phosphatase PtpA.

Authors:  Katherine A Rawls; P Therese Lang; Jun Takeuchi; Shinichi Imamura; Tyler D Baguley; Christoph Grundner; Tom Alber; Jonathan A Ellman
Journal:  Bioorg Med Chem Lett       Date:  2009-10-25       Impact factor: 2.823

4.  Utilization of nitrophenylphosphates and oxime-based ligation for the development of nanomolar affinity inhibitors of the Yersinia pestis outer protein H (YopH) phosphatase.

Authors:  Medhanit Bahta; George T Lountos; Beverly Dyas; Sung-Eun Kim; Robert G Ulrich; David S Waugh; Terrence R Burke
Journal:  J Med Chem       Date:  2011-03-28       Impact factor: 7.446

5.  Identification of multiple structurally distinct, nonpeptidic small molecule inhibitors of protein arginine deiminase 3 using a substrate-based fragment method.

Authors:  Haya Jamali; Hasan A Khan; Joseph R Stringer; Somenath Chowdhury; Jonathan A Ellman
Journal:  J Am Chem Soc       Date:  2015-03-05       Impact factor: 15.419

6.  Identification of a new class of nonpeptidic inhibitors of cruzain.

Authors:  Katrien Brak; Patricia S Doyle; James H McKerrow; Jonathan A Ellman
Journal:  J Am Chem Soc       Date:  2008-04-25       Impact factor: 15.419

7.  Quantitative and label-free technique for measuring protease activity and inhibition using a microfluidic cantilever array.

Authors:  Digvijay A Raorane; Mark D Lim; Fanqing Frank Chen; Charles S Craik; Arun Majumdar
Journal:  Nano Lett       Date:  2008-08-23       Impact factor: 11.189
  7 in total

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