Literature DB >> 16606858

Picrotoxin-like channel blockers of GABAA receptors.

Richard W Olsen1.   

Abstract

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Year:  2006        PMID： 16606858      PMCID： PMC1458832          DOI： 10.1073/pnas.0601121103

Source DB:  PubMed          Journal:  Proc Natl Acad Sci U S A        ISSN： 0027-8424            Impact factor:   11.205


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  22 in total

1.  Fishing for allosteric sites on GABA(A) receptors.

Authors:  Richard W Olsen; Chang-Sheng S Chang; Guodong Li; H Jacob Hanchar; Martin Wallner
Journal:  Biochem Pharmacol       Date:  2004-10-15       Impact factor: 5.858

2.  Bicyclic phosphorus esters that are potent convulsants and GABA antagonists.

Authors:  N G Bowery; J F Collins; R G Hill
Journal:  Nature       Date:  1976-06-17       Impact factor: 49.962

Review 3.  2,6,7-Trioxabicyclo[2.2.2]octanes: chemistry, toxicology and action at the GABA-gated chloride channel.

Authors:  J E Casida; C J Palmer
Journal:  Adv Biochem Psychopharmacol       Date:  1988

4.  Cage convulsants inhibit picrotoxinin binding.

Authors:  M K Ticku; R W Olsen
Journal:  Neuropharmacology       Date:  1979-03       Impact factor: 5.250

Review 5.  Picrotoxinin and related substances.

Authors:  L A Porter
Journal:  Chem Rev       Date:  1967-08       Impact factor: 60.622

6.  [35S]t-butylbicyclophosphorothionate binds with high affinity to brain-specific sites coupled to gamma-aminobutyric acid-A and ion recognition sites.

Authors:  R F Squires; J E Casida; M Richardson; E Saederup
Journal:  Mol Pharmacol       Date:  1983-03       Impact factor: 4.436

7.  A single-amino acid substitution in a gamma-aminobutyric acid subtype A receptor locus is associated with cyclodiene insecticide resistance in Drosophila populations.

Authors:  R H ffrench-Constant; J C Steichen; T A Rocheleau; K Aronstein; R T Roush
Journal:  Proc Natl Acad Sci U S A       Date:  1993-03-01       Impact factor: 11.205

8.  Interaction of picrotoxin with GABAA receptor channel-lining residues probed in cysteine mutants.

Authors:  M Xu; D F Covey; M H Akabas
Journal:  Biophys J       Date:  1995-11       Impact factor: 4.033

Review 9.  Analysis of GABAA receptor function and dissection of the pharmacology of benzodiazepines and general anesthetics through mouse genetics.

Authors:  Uwe Rudolph; Hanns Möhler
Journal:  Annu Rev Pharmacol Toxicol       Date:  2004       Impact factor: 13.820

10.  A study of the action of picrotoxin on the inhibitory neuromuscular junction of the crayfish.

Authors:  A Takeuchi; N Takeuchi
Journal:  J Physiol       Date:  1969-11       Impact factor: 5.182
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  25 in total

Review 1.  A novel GABA(A) receptor pharmacology: drugs interacting with the α(+) β(-) interface.

Authors:  Werner Sieghart; Joachim Ramerstorfer; Isabella Sarto-Jackson; Zdravko Varagic; Margot Ernst
Journal:  Br J Pharmacol       Date:  2012-05       Impact factor: 8.739

2.  Conserved toxic responses across divergent phylogenetic lineages: a meta-analysis of the neurotoxic effects of RDX among multiple species using toxicogenomics.

Authors:  Natàlia Garcia-Reyero; Tanwir Habib; Mehdi Pirooznia; Kurt A Gust; Ping Gong; Chris Warner; Mitchell Wilbanks; Edward Perkins
Journal:  Ecotoxicology       Date:  2011-03-29       Impact factor: 2.823

3.  Neurotoxins from snake venoms and α-conotoxin ImI inhibit functionally active ionotropic γ-aminobutyric acid (GABA) receptors.

Authors:  Denis S Kudryavtsev; Irina V Shelukhina; Lina V Son; Lucy O Ojomoko; Elena V Kryukova; Ekaterina N Lyukmanova; Maxim N Zhmak; Dmitry A Dolgikh; Igor A Ivanov; Igor E Kasheverov; Vladislav G Starkov; Joachim Ramerstorfer; Werner Sieghart; Victor I Tsetlin; Yuri N Utkin
Journal:  J Biol Chem       Date:  2015-07-28       Impact factor: 5.157

Review 4.  GABAA receptor: Positive and negative allosteric modulators.

Authors:  Richard W Olsen
Journal:  Neuropharmacology       Date:  2018-01-31       Impact factor: 5.250

5.  Rapid Throughput Analysis of GABAA Receptor Subtype Modulators and Blockers Using DiSBAC1(3) Membrane Potential Red Dye.

Authors:  Atefeh Mousavi Nik; Brandon Pressly; Vikrant Singh; Shane Antrobus; Susan Hulsizer; Michael A Rogawski; Heike Wulff; Isaac N Pessah
Journal:  Mol Pharmacol       Date:  2017-04-20       Impact factor: 4.436

6.  Antisense reduction of tau in adult mice protects against seizures.

Authors:  Sarah L DeVos; Dustin K Goncharoff; Guo Chen; Carey S Kebodeaux; Kaoru Yamada; Floy R Stewart; Dorothy R Schuler; Susan E Maloney; David F Wozniak; Frank Rigo; C Frank Bennett; John R Cirrito; David M Holtzman; Timothy M Miller
Journal:  J Neurosci       Date:  2013-07-31       Impact factor: 6.167

7.  Mapping convulsants' binding to the GABA-A receptor chloride ionophore: a proposed model for channel binding sites.

Authors:  A V Kalueff
Journal:  Neurochem Int       Date:  2006-09-07       Impact factor: 3.921

8.  Arginine derivatives of dicarboxylic acids from the parotid gland secretions of common toad Bufo bufo-New agonists of ionotropic γ-aminobutyric acid receptors.

Authors:  D S Lebedev; I A Ivanov; E V Kryukova; V G Starkov; V I Tsetlin; Yu N Utkin
Journal:  Dokl Biochem Biophys       Date:  2017-07-20       Impact factor: 0.788

9.  Postembryonic development of centrally generated flight motor patterns in the hawkmoth, Manduca sexta.

Authors:  Ricardo Vierk; Carsten Duch; Hans-Joachim Pflüger
Journal:  J Comp Physiol A Neuroethol Sens Neural Behav Physiol       Date:  2009-11-19       Impact factor: 1.836

10.  Agonist- and antagonist-induced conformational changes of loop F and their contributions to the rho1 GABA receptor function.

Authors:  Jianliang Zhang; Fenqin Xue; Yongchang Chang
Journal:  J Physiol       Date:  2008-11-17       Impact factor: 5.182
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