Literature DB >> 16502446

Starving the malaria parasite: inhibitors active against the aspartic proteases plasmepsins I, II, and IV.

Fraser Hof1, Andri Schütz, Christoph Fäh, Solange Meyer, Daniel Bur, Jun Liu, Daniel E Goldberg, François Diederich.   

Abstract

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Year:  2006        PMID： 16502446     DOI： 10.1002/anie.200504119

Source DB:  PubMed          Journal:  Angew Chem Int Ed Engl        ISSN： 1433-7851            Impact factor:   15.336


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  9 in total

1.  Conformational analyses of thiirane-based gelatinase inhibitors.

Authors:  Mijoon Lee; Dusan Hesek; Qicun Shi; Bruce C Noll; Jed F Fisher; Mayland Chang; Shahriar Mobashery
Journal:  Bioorg Med Chem Lett       Date:  2007-12-05       Impact factor: 2.823

2.  Crystal structures of the histo-aspartic protease (HAP) from Plasmodium falciparum.

Authors:  Prasenjit Bhaumik; Huogen Xiao; Charity L Parr; Yoshiaki Kiso; Alla Gustchina; Rickey Y Yada; Alexander Wlodawer
Journal:  J Mol Biol       Date:  2009-03-11       Impact factor: 5.469

3.  Matrix metalloproteinase 2 inhibition: combined quantum mechanics and molecular mechanics studies of the inhibition mechanism of (4-phenoxyphenylsulfonyl)methylthiirane and its oxirane analogue.

Authors:  Peng Tao; Jed F Fisher; Qicun Shi; Thom Vreven; Shahriar Mobashery; H Bernhard Schlegel
Journal:  Biochemistry       Date:  2009-10-20       Impact factor: 3.162

4.  Antimalarial activity of azadipeptide nitriles.

Authors:  Reik Löser; Jiri Gut; Philip J Rosenthal; Maxim Frizler; Michael Gütschow; Katherine T Andrews
Journal:  Bioorg Med Chem Lett       Date:  2009-10-30       Impact factor: 2.823

5.  Current developments in the therapy of protozoan infections.

Authors:  Mario Zucca; Dianella Savoia
Journal:  Open Med Chem J       Date:  2011-03-09

6.  EU-OPENSCREEN: A Novel Collaborative Approach to Facilitate Chemical Biology.

Authors:  Philip Brennecke; Dace Rasina; Oscar Aubi; Katja Herzog; Johannes Landskron; Bastien Cautain; Francisca Vicente; Jordi Quintana; Jordi Mestres; Bahne Stechmann; Bernhard Ellinger; Jose Brea; Jacek L Kolanowski; Radosław Pilarski; Mar Orzaez; Antonio Pineda-Lucena; Luca Laraia; Faranak Nami; Piotr Zielenkiewicz; Kamil Paruch; Espen Hansen; Jens P von Kries; Martin Neuenschwander; Edgar Specker; Petr Bartunek; Sarka Simova; Zbigniew Leśnikowski; Stefan Krauss; Lari Lehtiö; Ursula Bilitewski; Mark Brönstrup; Kjetil Taskén; Aigars Jirgensons; Heiko Lickert; Mads H Clausen; Jeanette H Andersen; Maria J Vicent; Olga Genilloud; Aurora Martinez; Marc Nazaré; Wolfgang Fecke; Philip Gribbon
Journal:  SLAS Discov       Date:  2019-01-07       Impact factor: 3.341

7.  Electrochemical sulfonylation of alkenes with sulfonyl hydrazides: a metal- and oxidant-free protocol for the synthesis of (E)-vinyl sulfones in water.

Authors:  Yin-Long Lai; Yunyan Mo; Shaoxi Yan; Shengling Zhang; Lejie Zhu; Jianmin Luo; Huishi Guo; Jianpeng Cai; Jianhua Liao
Journal:  RSC Adv       Date:  2020-09-08       Impact factor: 4.036

8.  Malaria-Infected Mice Are Cured by a Single Low Dose of a New Silylamide Trioxane Plus Mefloquine.

Authors:  Lauren E Woodard; Bryan T Mott; Vandana Singhal; Nirbhay Kumar; Theresa A Shapiro; Gary H Posner
Journal:  Pharmaceuticals (Basel)       Date:  2009-12-21

9.  A mild light-induced cleavage of the S-O bond of aryl sulfonate esters enables efficient sulfonylation of vinylarenes.

Authors:  Maxim Ratushnyy; Monika Kamenova; Vladimir Gevorgyan
Journal:  Chem Sci       Date:  2018-07-25       Impact factor: 9.825
  9 in total

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