Literature DB >> 16311994

Total synthesis, NMR solution structure, and binding model of the potent histone deacetylase inhibitor FR235222.

Manuela Rodriquez1, Stefania Terracciano, Elena Cini, Giulia Settembrini, Ines Bruno, Giuseppe Bifulco, Maurizio Taddei, Luigi Gomez-Paloma.   

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Year:  2006        PMID： 16311994     DOI： 10.1002/anie.200501995

Source DB:  PubMed          Journal:  Angew Chem Int Ed Engl        ISSN： 1433-7851            Impact factor:   15.336


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  5 in total

Review 1.  Discovery and mechanism of natural products as modulators of histone acetylation.

Authors:  Lilibeth A Salvador; Hendrik Luesch
Journal:  Curr Drug Targets       Date:  2012-07       Impact factor: 3.465

Review 2.  An overview of naturally occurring histone deacetylase inhibitors.

Authors:  Bumki Kim; Jiyong Hong
Journal:  Curr Top Med Chem       Date:  2015       Impact factor: 3.295

3.  Total Synthesis of Malacidin A by β-Hydroxyaspartic Acid Ligation-Mediated Cyclization and Absolute Structure Establishment.

Authors:  Zhenquan Sun; Zhuo Shang; Nicholas Forelli; Kathy Hiu Laam Po; Sheng Chen; Sean F Brady; Xuechen Li
Journal:  Angew Chem Int Ed Engl       Date:  2020-08-31       Impact factor: 15.336

4.  Concise syntheses of enantiomerically pure protected 4-hydroxypyroglutamic acid and 4-hydroxyproline from a nitroso-cyclopentadiene cycloadduct.

Authors:  Weiqiang Huang; Marvin J Miller
Journal:  Tetrahedron Asymmetry       Date:  2008-12-12

5.  Synthesis and biological evaluation of histone deacetylase inhibitors that are based on FR235222: a cyclic tetrapeptide scaffold.

Authors:  Erinprit K Singh; Suchitra Ravula; Chung-Mao Pan; Po-Shen Pan; Robert C Vasko; Stephanie A Lapera; Sujith V W Weerasinghe; Mary Kay H Pflum; Shelli R McAlpine
Journal:  Bioorg Med Chem Lett       Date:  2008-03-20       Impact factor: 2.823
  5 in total

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