Literature DB >> 16196020

Discovery of Mycobacterium tuberculosis protein tyrosine phosphatase A (MptpA) inhibitors based on natural products and a fragment-based approach.

Michael Manger1, Michael Scheck, Heino Prinz, Jens Peter von Kries, Thomas Langer, Krishna Saxena, Harald Schwalbe, Alois Fürstner, Jörg Rademann, Herbert Waldmann.   

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Year:  2005        PMID： 16196020     DOI： 10.1002/cbic.200500171

Source DB:  PubMed          Journal:  Chembiochem        ISSN： 1439-4227            Impact factor:   3.164


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  10 in total

1.  Formal synthesis of (+/-)-roseophilin.

Authors:  Abdallah Y Bitar; Alison J Frontier
Journal:  Org Lett       Date:  2009-01-01       Impact factor: 6.005

2.  Transient binding patches: a plausible concept for drug binding.

Authors:  Heino Prinz; André Schönichen
Journal:  J Chem Biol       Date:  2008-09-02

3.  Fragment-based discovery of selective inhibitors of the Mycobacterium tuberculosis protein tyrosine phosphatase PtpA.

Authors:  Katherine A Rawls; P Therese Lang; Jun Takeuchi; Shinichi Imamura; Tyler D Baguley; Christoph Grundner; Tom Alber; Jonathan A Ellman
Journal:  Bioorg Med Chem Lett       Date:  2009-10-25       Impact factor: 2.823

4.  Mycobacterial Protein Tyrosine Phosphatases A and B Inhibitors Augment the Bactericidal Activity of the Standard Anti-tuberculosis Regimen.

Authors:  Noton K Dutta; Rongjun He; Michael L Pinn; Yantao He; Francis Burrows; Zhong-Yin Zhang; Petros C Karakousis
Journal:  ACS Infect Dis       Date:  2015-12-24       Impact factor: 5.084

Review 5.  Mycobacterium tuberculosis Serine/Threonine Protein Kinases.

Authors:  Sladjana Prisic; Robert N Husson
Journal:  Microbiol Spectr       Date:  2014-10

6.  Crystal structures and inhibitor identification for PTPN5, PTPRR and PTPN7: a family of human MAPK-specific protein tyrosine phosphatases.

Authors:  Jeyanthy Eswaran; Jens Peter von Kries; Brian Marsden; Emma Longman; Judit E Debreczeni; Emilie Ugochukwu; Andrew Turnbull; Wen Hwa Lee; Stefan Knapp; Alastair J Barr
Journal:  Biochem J       Date:  2006-05-01       Impact factor: 3.857

7.  Organocatalytic multicomponent reaction for the acquisition of a selective inhibitor of mPTPB, a virulence factor of tuberculosis.

Authors:  Rongjun He; Li-Fan Zeng; Yantao He; Li Wu; Andrea Michelle Gunawan; Zhong-Yin Zhang
Journal:  Chem Commun (Camb)       Date:  2013-03-11       Impact factor: 6.222

8.  Protein tyrosine phosphatase PtpA is not required for Mycobacterium tuberculosis growth in mice.

Authors:  Christoph Grundner; Jeffery S Cox; Tom Alber
Journal:  FEMS Microbiol Lett       Date:  2008-08-22       Impact factor: 2.742

9.  Design, Synthesis, Biological Evaluation and Molecular Modeling Study of Novel Indolizine-1-Carbonitrile Derivatives as Potential Anti-Microbial Agents.

Authors:  Ehsan Faghih-Mirzaei; Mohammad Seifi; Mehdi Abaszadeh; Kamiar Zomorodian; Helia Helali
Journal:  Iran J Pharm Res       Date:  2018       Impact factor: 1.696

10.  Label-Free Fluorescent Kinase and Phosphatase Enzyme Assays with Supramolecular Host-Dye Pairs.

Authors:  Yan-Cen Liu; Shu Peng; Lora Angelova; Werner M Nau; Andreas Hennig
Journal:  ChemistryOpen       Date:  2019-11-12       Impact factor: 2.911
  10 in total

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