Literature DB >> 15982879

3-Thio-1,2,4-triazoles, novel somatostatin sst2/sst5 agonists.

Marie-Odile Contour-Galcéra1, Alban Sidhu, Pascale Plas, Pierre Roubert.   

Abstract

Novel 3-thio-1,2,4-triazoles have been obtained via a solution-phase parallel synthesis strategy, affording potent non-peptidic human somatostatin receptor subtypes 2 and 5 agonists.

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Year:  2005        PMID： 15982879     DOI： 10.1016/j.bmcl.2005.05.061

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN： 0960-894X            Impact factor:   2.823


  7 in total

1.  Theoretical analysis of somatostatin receptor 5 with antagonists and agonists for the treatment of neuroendocrine tumors.

Authors:  Santhosh Kumar Nagarajan; Sathya Babu; Thirumurthy Madhavan
Journal:  Mol Divers       Date:  2017-02-02       Impact factor: 2.943

2.  Synthesis and characterization of iron(II) quinaldate complexes.

Authors:  Dylan T Houghton; Nicholas W Gydesen; Navamoney Arulsamy; Mark P Mehn
Journal:  Inorg Chem       Date:  2010-02-01       Impact factor: 5.165

3.  Three-dimensional pharmacophore design and biochemical screening identifies substituted 1,2,4-triazoles as inhibitors of the annexin A2-S100A10 protein interaction.

Authors:  Tummala R K Reddy; Chan Li; Peter M Fischer; Lodewijk V Dekker
Journal:  ChemMedChem       Date:  2012-05-29       Impact factor: 3.466

4.  Understanding the influence of lipid bilayers and ligand molecules in determining the conformational dynamics of somatostatin receptor 2.

Authors:  Santhosh Kumar Nagarajan; Sathya Babu; Seema A Kulkarni; Aanand Vadivelu; Panneer Devaraju; Honglae Sohn; Thirumurthy Madhavan
Journal:  Sci Rep       Date:  2021-04-07       Impact factor: 4.379

5.  Retracted Article: The synthesis and biological activity of marine alkaloid derivatives and analogues.

Authors:  Shiyang Zhou; Gangliang Huang
Journal:  RSC Adv       Date:  2020-08-28       Impact factor: 4.036

6.  Design, synthesis and SAR exploration of tri-substituted 1,2,4-triazoles as inhibitors of the annexin A2-S100A10 protein interaction.

Authors:  Tummala R K Reddy; Chan Li; Xiaoxia Guo; Peter M Fischer; Lodewijk V Dekker
Journal:  Bioorg Med Chem       Date:  2014-08-07       Impact factor: 3.641

7.  A New One-Pot Synthesis of Quinoline-2-carboxylates under Heterogeneous Conditions.

Authors:  Serena Gabrielli; Alessandra Giardinieri; Susanna Sampaolesi; Roberto Ballini; Alessandro Palmieri
Journal:  Molecules       Date:  2016-06-15       Impact factor: 4.411
  7 in total

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