Literature DB >> 15949940

Module-assisted synthesis of the bifunctional labelling agent N-succinimidyl 4-[(18)F]fluorobenzoate ([(18)F]SFB).

P Mäding1, F Füchtner, F Wüst.   

Abstract

The three-step radiosynthesis of N-succinimidyl 4-[(18)F]fluorobenzoate ([(18)F]SFB) was adapted to a remotely controlled synthesis module. After optimization of the reaction conditions, the final [(18)F]SFB was obtained in decay-corrected radiochemical yields of 34-38% (related to [(18)F]fluoride; n=12) within a synthesis time of 68 min. The radiochemical purity was in the range of 93-96%.

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Year:  2005        PMID： 15949940     DOI： 10.1016/j.apradiso.2005.03.005

Source DB:  PubMed          Journal:  Appl Radiat Isot        ISSN： 0969-8043            Impact factor:   1.513


  20 in total

1.  A thiol-reactive 18F-labeling agent, N-[2-(4-18F-fluorobenzamido)ethyl]maleimide, and synthesis of RGD peptide-based tracer for PET imaging of alpha v beta 3 integrin expression.

Authors:  Weibo Cai; Xianzhong Zhang; Yun Wu; Xiaoyuan Chen
Journal:  J Nucl Med       Date:  2006-07       Impact factor: 10.057

2.  Fully automated preparation and conjugation of N-succinimidyl 4-[18F]fluorobenzoate ([18F]SFB) with RGD peptide using a GE FASTlab™ synthesizer.

Authors:  David Thonon; David Goblet; Eve Goukens; Geoffroy Kaisin; Jérôme Paris; Joël Aerts; Steve Lignon; Xavier Franci; Roland Hustinx; André Luxen
Journal:  Mol Imaging Biol       Date:  2011-12       Impact factor: 3.488

Review 3.  18 F-Labeling of Sensitive Biomolecules for Positron Emission Tomography.

Authors:  Hema S Krishnan; Longle Ma; Neil Vasdev; Steven H Liang
Journal:  Chemistry       Date:  2017-09-01       Impact factor: 5.236

4.  Microwave-assisted one-pot synthesis of N-succinimidyl-4[ ¹⁸F]fluorobenzoate ([¹⁸F]SFB).

Authors:  Shuang Hou; Duy Linh Phung; Wei-Yu Lin; Ming-wei Wang; Kan Liu; Clifton Kwang-Fu Shen
Journal:  J Vis Exp       Date:  2011-06-28       Impact factor: 1.355

5.  Highlighting the Versatility of the Tracerlab Synthesis Modules. Part 1: Fully Automated Production of [F]Labelled Radiopharmaceuticals using a Tracerlab FX(FN).

Authors:  Xia Shao; Raphaël Hoareau; Brian G Hockley; Louis J M Tluczek; Bradford D Henderson; Henry C Padgett; Peter J H Scott
Journal:  J Labelled Comp Radiopharm       Date:  2011-05-30       Impact factor: 1.921

6.  Improved 18F labeling of peptides with a fluoride-aluminum-chelate complex.

Authors:  William J McBride; Christopher A D'Souza; Robert M Sharkey; Habibe Karacay; Edmund A Rossi; Chien-Hsing Chang; David M Goldenberg
Journal:  Bioconjug Chem       Date:  2010-07-21       Impact factor: 4.774

Review 7.  Radiosyntheses using fluorine-18: the art and science of late stage fluorination.

Authors:  Erin L Cole; Megan N Stewart; Ryan Littich; Raphael Hoareau; Peter J H Scott
Journal:  Curr Top Med Chem       Date:  2014       Impact factor: 3.295

8.  Characterization of the Biodistribution and Systemic Absorption of TT-173, a New Hemostatic Agent of Recombinant Human Tissue Factor, Using Radiolabeling with 18F.

Authors:  Santiago Rojas; José Raúl Herance; Juan Domingo Gispert; Belén Arias; Ignasi Miquel; Ramón López; Pilar Sánchez; Esther Rincón; Jesús Murat
Journal:  Eur J Drug Metab Pharmacokinet       Date:  2017-08       Impact factor: 2.441

9.  Synthesis and pre-clinical evaluation of an (18)F-labeled single-chain antibody fragment for PET imaging of epithelial ovarian cancer.

Authors:  Sai Kiran Sharma; Melinda Wuest; Jenilee D Way; Vincent R Bouvet; Monica Wang; Frank R Wuest
Journal:  Am J Nucl Med Mol Imaging       Date:  2016-07-06

10.  Fully automated production of diverse 18F-labeled PET tracers on the ELIXYS multireactor radiosynthesizer without hardware modification.

Authors:  Mark Lazari; Jeffrey Collins; Bin Shen; Mohammed Farhoud; Daniel Yeh; Brandon Maraglia; Frederick T Chin; David A Nathanson; Melissa Moore; R Michael van Dam
Journal:  J Nucl Med Technol       Date:  2014-07-17
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