Literature DB >> 15911278

New inhibitors of rabbit muscle triose-phosphate isomerase.

M Fonvielle1, S Mariano, M Therisod.   

Abstract

We describe the synthesis and evaluation of three new competitive inhibitors of triose-phosphate isomerase. One of them (phosphoglycoloamidoxime: K(i) = 4.5 microM) is among the best reversible inhibitors so far reported for this enzyme.

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Year:  2005        PMID： 15911278     DOI： 10.1016/j.bmcl.2005.03.061

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN： 0960-894X            Impact factor:   2.823


  4 in total

Review 1.  Triosephosphate isomerase: a highly evolved biocatalyst.

Authors:  R K Wierenga; E G Kapetaniou; R Venkatesan
Journal:  Cell Mol Life Sci       Date:  2010-08-07       Impact factor: 9.261

2.  An enolase inhibitor for the targeted treatment of ENO1-deleted cancers.

Authors:  Yu-Hsi Lin; Nikunj Satani; Naima Hammoudi; Victoria C Yan; Yasaman Barekatain; Sunada Khadka; Jeffrey J Ackroyd; Dimitra K Georgiou; Cong-Dat Pham; Kenisha Arthur; David Maxwell; Zhenghong Peng; Paul G Leonard; Barbara Czako; Federica Pisaneschi; Pijus Mandal; Yuting Sun; Rafal Zielinski; Susana Castro Pando; Xiaobo Wang; Theresa Tran; Quanyu Xu; Qi Wu; Yongying Jiang; Zhijun Kang; John M Asara; Waldemar Priebe; William Bornmann; Joseph R Marszalek; Ronald A DePinho; Florian L Muller
Journal:  Nat Metab       Date:  2020-11-23

3.  Promiscuous Lipase-Catalyzed Knoevenagel-Phospha-Michael Reaction for the Synthesis of Antimicrobial β-Phosphono Malonates.

Authors:  Jan Samsonowicz-Górski; Dominik Koszelewski; Paweł Kowalczyk; Paweł Śmigielski; Anastasiia Hrunyk; Karol Kramkowski; Aleksandra Wypych; Mateusz Szymczak; Rafał Lizut; Ryszard Ostaszewski
Journal:  Int J Mol Sci       Date:  2022-08-08       Impact factor: 6.208

4.  Novel and Selective Rhipicephalus microplus Triosephosphate Isomerase Inhibitors with Acaricidal Activity.

Authors:  Luiz Saramago; Helga Gomes; Elena Aguilera; Hugo Cerecetto; Mercedes González; Mauricio Cabrera; Maria Fernanda Alzugaray; Itabajara da Silva Vaz Junior; Rodrigo Nunes da Fonseca; Beatriz Aguirre-López; Nallely Cabrera; Ruy Pérez-Montfort; Alicia Merlino; Jorge Moraes; Guzmán Álvarez
Journal:  Vet Sci       Date:  2018-08-23
  4 in total

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