Literature DB >> 15771244

Suitability of the upper airway models obtained from MRI studies in simulating drug lung deposition from inhalers.

T Ehtezazi1, K W Southern, D Allanson, I Jenkinson, C O'Callaghan.   

Abstract

PURPOSE: In this study, the suitability of the upper airway models, obtained by applying a magnetic resonance imaging method, in simulating in vivo aerosol deposition data is determined.
METHODS: Depositions of salbutamol sulfate from two nebulizers in two models, one with constriction at the oropharynx (the constricted cast) and another model without that constriction (the wide cast), were determined.
RESULTS: For the Sidestream and Ventstream nebulizer, 76 +/- 3% (mean +/- standard deviation) and 81 +/- 2% of the emitted dose deposited in the constricted cast, whereas 51 +/- 2% and 49 +/- 3% of the emitted dose deposited in the wide cast, respectively. These values were in good agreement with in vivo data. Mostly, increasing nebulizer charge volume (by normal saline) from 2.5 ml to 5 ml increased significantly the lung dose. However, the lung doses from the Sidestream and Ventstream nebulizer with 2.5 ml charge volume via the wide cast were (1.37 +/- 0.06 and 1.38 +/- 0.05 mg) significantly larger than those for the constricted cast with 5 ml charge volume (0.87 +/- 0.15 and 0.86 +/- 0.21 mg, respectively) (p = 0.005).
CONCLUSIONS: The upper airway models closely simulated the in vivo deposition data. Optimizing the upper airway posture during inhalation via the nebulizers would be more efficient in increasing drug lung delivery than diluting their contents.

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Year:  2005        PMID: 15771244     DOI: 10.1007/s11095-004-9023-1

Source DB:  PubMed          Journal:  Pharm Res        ISSN: 0724-8741            Impact factor:   4.200


  12 in total

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2.  Medication nebulizer performance. Effects of diluent volume, nebulizer flow, and nebulizer brand.

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3.  Lactose as a carrier in dry powder formulations: the influence of surface characteristics on drug delivery.

Authors:  X M Zeng; G P Martin; C Marriott; J Pritchard
Journal:  J Pharm Sci       Date:  2001-09       Impact factor: 3.534

4.  Deposition of inhaled particles in the mouth and throat of asthmatic subjects.

Authors:  K Svartengren; P A Lindestad; M Svartengren; G Bylin; K Philipson; P Camner
Journal:  Eur Respir J       Date:  1994-08       Impact factor: 16.671

5.  In vitro monodisperse aerosol deposition in a mouth and throat with six different inhalation devices.

Authors:  W H DeHaan; W H Finlay
Journal:  J Aerosol Med       Date:  2001

6.  Dynamic change of the upper airway during inhalation via aerosol delivery devices.

Authors:  Touraj Ehtezazi; Mark A Horsfield; Peter W Barry; Christopher O'Callaghan
Journal:  J Aerosol Med       Date:  2004

7.  An in vitro analysis of the output of salbutamol from different nebulizers.

Authors:  P W Barry; C O'Callaghan
Journal:  Eur Respir J       Date:  1999-05       Impact factor: 16.671

8.  Added external resistance reduces oropharyngeal deposition and increases lung deposition of aerosol particles in asthmatics.

Authors:  K Svartengren; P Lindestad; M Svartengren; K Philipson; G Bylin; P Camner
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9.  Oropharyngeal deposition of 3.5 microns particles inhaled through an elongated mouthpiece.

Authors:  K Svartengren; M Anderson; M Svartengren; K Philipson; P Camner
Journal:  Eur Respir J       Date:  1996-07       Impact factor: 16.671

10.  Efficient drug delivery to the lungs from a continuously operated open-vent nebulizer and low pressure compressor system.

Authors:  S P Newman; G R Pitcairn; G Hooper; M Knoch
Journal:  Eur Respir J       Date:  1994-06       Impact factor: 16.671

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  4 in total

1.  Effect of oropharyngeal length in drug lung delivery via suspension pressurized metered dose inhalers.

Authors:  T Ehtezazi; D R Allanson; I D Jenkinson; C O'Callaghan
Journal:  Pharm Res       Date:  2006-05-26       Impact factor: 4.200

2.  The interaction between the oropharyngeal geometry and aerosols via pressurised metered dose inhalers.

Authors:  T Ehtezazi; I Saleem; I Shrubb; D R Allanson; I D Jenkinson; C O'Callaghan
Journal:  Pharm Res       Date:  2009-11-10       Impact factor: 4.200

3.  Comparison of in vitro deposition of pharmaceutical aerosols in an idealized child throat with in vivo deposition in the upper respiratory tract of children.

Authors:  Conor A Ruzycki; Laleh Golshahi; Reinhard Vehring; Warren H Finlay
Journal:  Pharm Res       Date:  2014-01-07       Impact factor: 4.200

4.  Nebulized liposomal gadobenate dimeglumine contrast formulation for magnetic resonance imaging of larynx and trachea.

Authors:  Xiaohui Wei; Huawei Wu; Qing Lu; Jianrong Xu; Yuhong Xu
Journal:  Int J Nanomedicine       Date:  2011-12-19
  4 in total

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