Literature DB >> 15514818

The first tandem double palladium-catalyzed aminations: synthesis of dipyrido[1,2-a:3',2'-d]imidazole and its benzo- and aza-analogues.

Kristof T J Loones1, Bert U W Maes, Roger A Dommisse, Guy L F Lemière.   

Abstract

A new strategy for the synthesis of the title compounds via a regio- and chemoselective one-pot inter- and intramolecular Buchwald-Hartwig amination of 2-chloro-3-iodopyridine with aminoazines and -diazines is reported.

Entities:  

Mesh：

Substances：

Year:  2004        PMID： 15514818     DOI： 10.1039/b409161b

Source DB:  PubMed          Journal:  Chem Commun (Camb)        ISSN： 1359-7345            Impact factor:   6.222


  3 in total

1.  A mild, catalyst-free synthesis of 2-aminopyridines.

Authors:  Bhaskar Poola; Wonken Choung; Michael H Nantz
Journal:  Tetrahedron       Date:  2008-11-24       Impact factor: 2.457

Review 2.  Applications of Palladium-Catalyzed C-N Cross-Coupling Reactions.

Authors:  Paula Ruiz-Castillo; Stephen L Buchwald
Journal:  Chem Rev       Date:  2016-09-30       Impact factor: 60.622

3.  Bioisosteric transformations and permutations in the triazolopyrimidine scaffold to identify the minimum pharmacophore required for inhibitory activity against Plasmodium falciparum dihydroorotate dehydrogenase.

Authors:  Alka Marwaha; John White; Farah El Mazouni; Sharon A Creason; Sreekanth Kokkonda; Frederick S Buckner; Susan A Charman; Margaret A Phillips; Pradipsinh K Rathod
Journal:  J Med Chem       Date:  2012-08-21       Impact factor: 7.446
  3 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.