Literature DB >> 15274229

Design, synthesis, and biological evaluation of a small-molecule inhibitor of the histone acetyltransferase Gcn5.

Markus Biel1, Androniki Kretsovali, Efthymia Karatzali, Joseph Papamatheakis, Athanassios Giannis.   

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Year:  2004        PMID： 15274229     DOI： 10.1002/anie.200453879

Source DB:  PubMed          Journal:  Angew Chem Int Ed Engl        ISSN： 1433-7851            Impact factor:   15.336


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  36 in total

1.  Targeting of histone acetyltransferase p300 by cyclopentenone prostaglandin Δ(12)-PGJ(2) through covalent binding to Cys(1438).

Authors:  Kodihalli C Ravindra; Vivek Narayan; Gerald H Lushington; Blake R Peterson; K Sandeep Prabhu
Journal:  Chem Res Toxicol       Date:  2011-12-16       Impact factor: 3.739

2.  A dual role of linker histone H1.4 Lys 34 acetylation in transcriptional activation.

Authors:  Kinga Kamieniarz; Annalisa Izzo; Miroslav Dundr; Philipp Tropberger; Luka Ozretic; Jutta Kirfel; Elisabeth Scheer; Philippe Tropel; Jacek R Wisniewski; Laszlo Tora; Stephane Viville; Reinhard Buettner; Robert Schneider
Journal:  Genes Dev       Date:  2012-03-30       Impact factor: 11.361

3.  Epigenetic regulation of Atoh1 guides hair cell development in the mammalian cochlea.

Authors:  Zlatka P Stojanova; Tao Kwan; Neil Segil
Journal:  Development       Date:  2015-10-15       Impact factor: 6.868

4.  Stalling of spliceosome assembly at distinct stages by small-molecule inhibitors of protein acetylation and deacetylation.

Authors:  Andreas N Kuhn; Maria A van Santen; Andreas Schwienhorst; Henning Urlaub; Reinhard Lührmann
Journal:  RNA       Date:  2008-11-24       Impact factor: 4.942

Review 5.  The promise and failures of epigenetic therapies for cancer treatment.

Authors:  Pasano Bojang; Kenneth S Ramos
Journal:  Cancer Treat Rev       Date:  2013-07-05       Impact factor: 12.111

6.  Diencephalic Size Is Restricted by a Novel Interplay Between GCN5 Acetyltransferase Activity and Retinoic Acid Signaling.

Authors:  Jonathan J Wilde; Julie A Siegenthaler; Sharon Y R Dent; Lee A Niswander
Journal:  J Neurosci       Date:  2017-02-02       Impact factor: 6.167

7.  Quinoline derivative MC1626, a putative GCN5 histone acetyltransferase (HAT) inhibitor, exhibits HAT-independent activity against Toxoplasma gondii.

Authors:  Aaron T Smith; Meredith R Livingston; Antonello Mai; Patrizia Filetici; Sherry F Queener; William J Sullivan
Journal:  Antimicrob Agents Chemother       Date:  2006-12-18       Impact factor: 5.191

8.  Inhibition of lysine acetyltransferase KAT3B/p300 activity by a naturally occurring hydroxynaphthoquinone, plumbagin.

Authors:  Kodihalli C Ravindra; B Ruthrotha Selvi; Mohammed Arif; B A Ashok Reddy; Gali R Thanuja; Shipra Agrawal; Suman Kalyan Pradhan; Natesh Nagashayana; Dipak Dasgupta; Tapas K Kundu
Journal:  J Biol Chem       Date:  2009-07-01       Impact factor: 5.157

9.  Histone acetyltransferase inhibitor anacardic acid causes changes in global gene expression during in vitro Plasmodium falciparum development.

Authors:  Long Cui; Jun Miao; Tetsuya Furuya; Qi Fan; Xinyi Li; Pradipsinh K Rathod; Xin-Zhuan Su; Liwang Cui
Journal:  Eukaryot Cell       Date:  2008-05-16

10.  Stereocontrolled Synthesis of (+)-Plagiogyrin A.

Authors:  Yunlong Shi; Joshua G Pierce
Journal:  Org Lett       Date:  2016-10-03       Impact factor: 6.005
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