Literature DB >> 15151525

Leflunomide in active rheumatoid arthritis: a prospective study in daily practice.

E N Van Roon1, T L Th A Jansen, L Mourad, P M Houtman, G A W Bruyn, E N Griep, B Wilffert, H Tobi, J R B J Brouwers.   

Abstract

AIMS: We prospectively studied the efficacy, incidence of adverse drug reactions and withdrawal from leflunomide in an outpatient population with rheumatoid arthritis in a setting of care-as-usual.
METHODS: In this prospective case series study, from outpatient medical records a standard dataset was collected including patient and disease characteristics, data on leflunomide use and adverse drug reactions.
RESULTS: During the study period 136 rheumatoid arthritis patients started leflunomide. Median (range) follow-up duration was 317 (11-911) days. Sixty-five percent of patients experienced at least one adverse drug reaction related to leflunomide. During follow-up 76 patients (56%) withdrew from leflunomide treatment, mainly because of adverse drug reactions (29%) or lack of efficacy (13%). The overall incidence density for withdrawal from leflunomide was 56.2 per 100 patient-years. Complete data for calculating efficacy using a validated disease activity score on 28 joints (DAS(28)) was available for 48, 36, and 35% of patients at 2, 6, and 12 months follow-up, respectively. Within a 12-month period after start of leflunomide treatment 76% of the evaluable patients were classified as moderate or good responders according to the DAS(28) response criteria.
CONCLUSIONS: In the setting of care-as-usual, rheumatoid arthritis patients starting leflunomide frequently experienced adverse drug reactions. More than half of the patients withdrew from leflunomide treatment within a year after start of leflunomide treatment, mainly because of adverse drug reactions.

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Year:  2004        PMID: 15151525      PMCID: PMC1884519          DOI: 10.1111/j.1365-2125.2004.02075.x

Source DB:  PubMed          Journal:  Br J Clin Pharmacol        ISSN: 0306-5251            Impact factor:   4.335


  26 in total

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Journal:  BMJ       Date:  1996-05-11

2.  Treatment of active rheumatoid arthritis with leflunomide compared with placebo and methotrexate. Leflunomide Rheumatoid Arthritis Investigators Group.

Authors:  V Strand; S Cohen; M Schiff; A Weaver; R Fleischmann; G Cannon; R Fox; L Moreland; N Olsen; D Furst; J Caldwell; J Kaine; J Sharp; F Hurley; I Loew-Friedrich
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3.  Pharmacokinetics, safety, and efficacy of combination treatment with methotrexate and leflunomide in patients with active rheumatoid arthritis.

Authors:  M E Weinblatt; J M Kremer; J S Coblyn; A L Maier; S M Helfgott; M Morrell; V M Byrne; M V Kaymakcian; V Strand
Journal:  Arthritis Rheum       Date:  1999-07

4.  A comparison of the efficacy and safety of leflunomide and methotrexate for the treatment of rheumatoid arthritis.

Authors:  P Emery; F C Breedveld; E M Lemmel; J P Kaltwasser; P T Dawes; B Gömör; F Van Den Bosch; D Nordström; O Bjorneboe; R Dahl; K Horslev-Petersen; A Rodriguez De La Serna; M Molloy; M Tikly; C Oed; R Rosenburg; I Loew-Friedrich
Journal:  Rheumatology (Oxford)       Date:  2000-06       Impact factor: 7.580

5.  Treatment with leflunomide slows radiographic progression of rheumatoid arthritis: results from three randomized controlled trials of leflunomide in patients with active rheumatoid arthritis. Leflunomide Rheumatoid Arthritis Investigators Group.

Authors:  J T Sharp; V Strand; H Leung; F Hurley; I Loew-Friedrich
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6.  Modulation of inflammation and metalloproteinase expression in synovial tissue by leflunomide and methotrexate in patients with active rheumatoid arthritis. Findings in a prospective, randomized, double-blind, parallel-design clinical trial in thirty-nine patients at two centers.

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Journal:  Arthritis Rheum       Date:  2000-08

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Authors:  E D Harris
Journal:  J Rheumatol Suppl       Date:  1996-03

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Authors:  Jorge Jaimes-Hernández; Manuel Robles-San Román; Rodrigo Suárez-Otero; M Eugenia Dávalos-Zugasti; Sergio Arroyo-Borrego
Journal:  J Rheumatol       Date:  2004-02       Impact factor: 4.666

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Journal:  Arthritis Rheum       Date:  1996-05
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  8 in total

1.  Leflunomide in the treatment of rheumatoid arthritis. An analysis of predictors for treatment continuation.

Authors:  E N van Roon; M Hoekstra; H Tobi; T L Th A Jansen; H J Bernelot Moens; J R B J Brouwers; M A F J van de Laar
Journal:  Br J Clin Pharmacol       Date:  2005-09       Impact factor: 4.335

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Authors:  Khadija Shahab Turabi; Ankita Deshmukh; Sayan Paul; Dayanand Swami; Shafina Siddiqui; Urwashi Kumar; Shreelekha Naikar; Shine Devarajan; Soumya Basu; Manash K Paul; Jyotirmoi Aich
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  2022-06-13       Impact factor: 3.195

3.  Therapeutic drug monitoring of A77 1726, the active metabolite of leflunomide: serum concentrations predict response to treatment in patients with rheumatoid arthritis.

Authors:  E N van Roon; T L T A Jansen; M A F J van de Laar; M Janssen; J P Yska; R Keuper; P M Houtman; J R B J Brouwers
Journal:  Ann Rheum Dis       Date:  2004-09-02       Impact factor: 19.103

Review 4.  Benefit-risk assessment of leflunomide: an appraisal of leflunomide in rheumatoid arthritis 10 years after licensing.

Authors:  Nicola Alcorn; Sarah Saunders; Rajan Madhok
Journal:  Drug Saf       Date:  2009       Impact factor: 5.606

5.  Metabolomics of Aerobic Exercise in Chronic Stroke Survivors: A Pilot Study.

Authors:  Monica C Serra; Carolyn J Accardi; Chunyu Ma; Younja Park; ViLinh Tran; Dean P Jones; Charlene E Hafer-Macko; Alice S Ryan
Journal:  J Stroke Cerebrovasc Dis       Date:  2019-10-25       Impact factor: 2.136

6.  Polymorphisms in cytochrome P450 2C19 enzyme and cessation of leflunomide in patients with rheumatoid arthritis.

Authors:  Michael D Wiese; Matthew Schnabl; Catherine O'Doherty; Llewellyn D Spargo; Michael J Sorich; Leslie G Cleland; Susanna M Proudman
Journal:  Arthritis Res Ther       Date:  2012-07-12       Impact factor: 5.156

Review 7.  Reappraisal of the clinical use of leflunomide in rheumatoid arthritis and psoriatic arthritis.

Authors:  Peter Bb Jones; Douglas Hn White
Journal:  Open Access Rheumatol       Date:  2010-11-03

8.  The Selective Oral Immunomodulator Vidofludimus in Patients with Active Rheumatoid Arthritis: Safety Results from the COMPONENT Study.

Authors:  Andreas Muehler; Hella Kohlhof; Manfred Groeppel; Daniel Vitt
Journal:  Drugs R D       Date:  2019-12
  8 in total

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