Literature DB >> 15125944

Solid-phase synthesis of kojic acid-tripeptides and their tyrosinase inhibitory activity, storage stability, and toxicity.

Hanyoung Kim1, Jaehui Choi, Jin Ku Cho, Sun Yeou Kim, Yoon-Sik Lee.   

Abstract

A small library of kojic acid-tripeptides (Ko-X1X2X3) was prepared by solid-phase parallel synthesis and assayed to evaluate their tyrosinase inhibitory activity. Most of the kojic acid-tripeptides showed better activities than kojic acid. Kojic acid-FWY was the best compound, and it exhibited 100-fold tyrosinase inhibitory activity compared with kojic acid. In addition, their storage stabilities were approximately 15 times higher and their toxicity was lower than that of kojic acid.

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Year:  2004        PMID： 15125944     DOI： 10.1016/j.bmcl.2004.03.046

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN： 0960-894X            Impact factor:   2.823


  12 in total

1.  In vitro kinetic release study, antimicrobial activity and in vivo toxicity profile of a kojic acid ester-based nanoemulsion for topical application.

Authors:  Sharifah Nurfadhlin Afifah Syed Azhar; Siti Efliza Ashari; Syahida Ahmad; Norazlinaliza Salim
Journal:  RSC Adv       Date:  2020-12-09       Impact factor: 4.036

2.  Kinetics of mushroom tyrosinase and melanogenesis inhibition by N-acetyl-pentapeptides.

Authors:  Ching-Yi Lien; Ching-Yu Chen; Shih-Ting Lai; Chin-Feng Chan
Journal:  ScientificWorldJournal       Date:  2014-07-22

Review 3.  Skin whitening agents: medicinal chemistry perspective of tyrosinase inhibitors.

Authors:  Thanigaimalai Pillaiyar; Manoj Manickam; Vigneshwaran Namasivayam
Journal:  J Enzyme Inhib Med Chem       Date:  2017-12       Impact factor: 5.051

4.  Evaluating the Performance of a Non-Bonded Cu2+ Model Including Jahn-Teller Effect into the Binding of Tyrosinase Inhibitors.

Authors:  Lucas Sousa Martins; Jerônimo Lameira; Hendrik G Kruger; Cláudio Nahum Alves; José Rogério A Silva
Journal:  Int J Mol Sci       Date:  2020-07-06       Impact factor: 5.923

5.  Development of a kojic monooleate-enriched oil-in-water nanoemulsion as a potential carrier for hyperpigmentation treatment.

Authors:  Sharifah Nurfadhlin Afifah Syed Azhar; Siti Efliza Ashari; Norazlinaliza Salim
Journal:  Int J Nanomedicine       Date:  2018-10-15

6.  Development of Ultrasound-Assisted Extraction to Produce Skin-Whitening and Anti-Wrinkle Substances from Safflower Seed.

Authors:  Suh-Hee Yeom; Da-Hye Gam; Jun-Hee Kim; Jin-Woo Kim
Journal:  Molecules       Date:  2022-02-15       Impact factor: 4.411

7.  K-Nearest Neighbor and Random Forest-Based Prediction of Putative Tyrosinase Inhibitory Peptides of Abalone Haliotis diversicolor.

Authors:  Sasikarn Kongsompong; Teerasak E-Kobon; Pramote Chumnanpuen
Journal:  Molecules       Date:  2021-06-16       Impact factor: 4.411

8.  Dipeptides Inhibit Melanin Synthesis in Mel-Ab Cells through Down-Regulation of Tyrosinase.

Authors:  Hyun-E Lee; Eun-Hyun Kim; Hye-Ryung Choi; Uy Dong Sohn; Hye-Young Yun; Kwang Jin Baek; Nyoun Soo Kwon; Kyoung-Chan Park; Dong-Seok Kim
Journal:  Korean J Physiol Pharmacol       Date:  2012-08-10       Impact factor: 2.016

9.  Optimisation and Characterisation of Lipase-Catalysed Synthesis of a Kojic Monooleate Ester in a Solvent-Free System by Response Surface Methodology.

Authors:  Khairulazhar Jumbri; Mohd Fahruddin Al-Haniff Rozy; Siti Efliza Ashari; Rosfarizan Mohamad; Mahiran Basri; Hamid Reza Fard Masoumi
Journal:  PLoS One       Date:  2015-12-14       Impact factor: 3.240

10.  An Improved Nanoemulsion Formulation Containing Kojic Monooleate: Optimization, Characterization and In Vitro Studies.

Authors:  Muhammad Azimuddin Roselan; Siti Efliza Ashari; Nur Hana Faujan; Siti Munirah Mohd Faudzi; Rosfarizan Mohamad
Journal:  Molecules       Date:  2020-06-04       Impact factor: 4.411
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