Literature DB >> 15013018

1,2-Benzothiazine 1,1-dioxide alpha-ketoamide analogues as potent calpain I inhibitors.

Ron Bihovsky1, Ming Tao, John P Mallamo, Gregory J Wells.   

Abstract

A series of potent 1,2-benzothiazine 1,1-dioxide alpha-ketoamide inhibitors of calpain I is described.

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Year:  2004        PMID： 15013018     DOI： 10.1016/j.bmcl.2003.11.037

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN： 0960-894X            Impact factor:   2.823


  12 in total

1.  N-[2-(Amino-carbon-yl)phen-yl]-4-hydr-oxy-2-methyl-2H-1,2-benzothia-zine-3-carboxamide 1,1-dioxide.

Authors:  Muhammad Nadeem Arshad; Muhammad Zia-Ur-Rehman; Islam Ullah Khan
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2009-09-30

2.  Methyl 4-eth-oxy-2-methyl-2H-1,2-benzothia-zine-3-carboxyl-ate 1,1-dioxide.

Authors:  Muhammad Zia-Ur-Rehman; Jamil Anwar Choudary; Mark R J Elsegood; Noshin Akbar; Hamid Latif Siddiqui
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2008-07-16

3.  1-(4-Hydr-oxy-2-methyl-1,1-dioxo-2H-1,2-benzothia-zin-3-yl)ethanone.

Authors:  Matloob Ahmad; Hamid Latif Siddiqui; Muhammad Zia-Ur-Rehman; Muhammad Irfan Ashiq; Graham John Tizzard
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2008-04-02

4.  N-(3,4-Dimethyl-phen-yl)-4-hydr-oxy-2-methyl-2H-1,2-benzothia-zine-3-carboxamide 1,1-dioxide.

Authors:  Waseeq Ahmad Siddiqui; Muhammad Ali; Muhammad Zia-Ur-Rehman; Saima Sharif; Graham John Tizzard
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2009-03-28

5.  Methyl 4-hydr-oxy-2-propyl-2H-1,2-benzothia-zine-3-carboxyl-ate 1,1-dioxide.

Authors:  Muhammad Nadeem Arshad; Muhammad Zia-Ur-Rehman; Islam Ullah Khan
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2009-11-07

6.  Piperidinium 4-hydr-oxy-3-methoxy-carbon-yl-1,2-benzothia-zin-2-ide 1,1-dioxide.

Authors:  Muhammad Nadeem Arshad; Muhammad Zia-Ur-Rehman; Naveed Ahmed; Islam Ullah Khan
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2009-09-12

7.  Methyl 2-methyl-4-(oxiran-2-ylmeth-oxy)-2H-1,2-benzothia-zine-3-carboxyl-ate 1,1-dioxide.

Authors:  Matloob Ahmad; Hamid Latif Siddiqui; Muhammad Zia-Ur-Rehman; Mark R J Elsegood; George W Weaver
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2010-01-09

8.  Methyl 2-acetonyl-4-hydr-oxy-2H-1,2-benzothia-zine-3-carboxyl-ate 1,1-dioxide.

Authors:  Matloob Ahmad; Hamid Latif Siddiqui; Muhammad Zia-Ur-Rehman; Graham John Tizzard; Saeed Ahmad
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2008-07-05

9.  2-[(E)-1,1-Dioxo-2-(2,4,5-tri-fluoro-benz-yl)-3,4-di-hydro-2H-1,2-benzo-thia-zin-4-yl-idene]acetic acid.

Authors:  Shaojuan Zhu; Shagufta Parveen; Changjin Zhu
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2014-06-14

10.  Evaluation of 1,2-Benzothiazine 1,1-dioxide Derivatives In Vitro Activity towards Clinical-Relevant Microorganisms and Fibroblasts.

Authors:  Ruth K Dudek-Wicher; Berenika M Szczęśniak-Sięga; Rafał J Wiglusz; Jan Janczak; Marzenna Bartoszewicz; Adam F Junka
Journal:  Molecules       Date:  2020-07-31       Impact factor: 4.411
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