Literature DB >> 14976423

The molecular mysteries underlying P-glycoprotein-mediated multidrug resistance.

Gergely Szakács1, Kevin G Chen, Michael M Gottesman.   

Abstract

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Year:  2004        PMID: 14976423     DOI: 10.4161/cbt.3.4.743

Source DB:  PubMed          Journal:  Cancer Biol Ther        ISSN: 1538-4047            Impact factor:   4.742


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  5 in total

1.  Boosted feature selectors: a case study on prediction P-gp inhibitors and substrates.

Authors:  Gonzalo Cerruela García; Nicolás García-Pedrajas
Journal:  J Comput Aided Mol Des       Date:  2018-10-26       Impact factor: 3.686

2.  Mutational studies of G553 in TM5 of ABCG2: a residue potentially involved in dimerization.

Authors:  Orsolya Polgar; Csilla Ozvegy-Laczka; Robert W Robey; Kuniaki Morisaki; Masaki Okada; Akina Tamaki; Gabriella Koblos; N Barry Elkind; Yvona Ward; Michael Dean; Balazs Sarkadi; Susan E Bates
Journal:  Biochemistry       Date:  2006-04-25       Impact factor: 3.162

3.  Structure-Activity Relationships of 8-Hydroxyquinoline-Derived Mannich Bases with Tertiary Amines Targeting Multidrug-Resistant Cancer.

Authors:  Veronika F S Pape; Roberta Palkó; Szilárd Tóth; Miklós J Szabó; Judit Sessler; György Dormán; Éva A Enyedy; Tibor Soós; István Szatmári; Gergely Szakács
Journal:  J Med Chem       Date:  2022-05-25       Impact factor: 8.039

4.  Relation of Metal-Binding Property and Selective Toxicity of 8-Hydroxyquinoline Derived Mannich Bases Targeting Multidrug Resistant Cancer Cells.

Authors:  Veronika F S Pape; Anikó Gaál; István Szatmári; Nóra Kucsma; Norbert Szoboszlai; Christina Streli; Ferenc Fülöp; Éva A Enyedy; Gergely Szakács
Journal:  Cancers (Basel)       Date:  2021-01-05       Impact factor: 6.639

5.  Cyclosporine A enables vincristine-induced apoptosis during reversal of multidrug resistance phenotype in chronic myeloid leukemia cells.

Authors:  Paloma Silva de Souza; Flavia da Cunha Vasconcelos; Luis Felipe R Silva; Raquel Ciuvalschi Maia
Journal:  Tumour Biol       Date:  2012-01-31
  5 in total

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