Literature DB >> 14673959

Leflunomide use during the first 33 months after food and drug administration approval: experience with a national cohort of 3,325 patients.

Chokkalingam Siva1, Seth A Eisen, Rebecca Shepherd, Francesca Cunningham, Meika A Fang, William Finch, Don Salisbury, Jasvinder A Singh, Richard Stern, S Alireza Zarabadi.   

Abstract

OBJECTIVE: To describe leflunomide (LEF) use in a national cohort of 3,325 veterans.
METHODS: Prescriptions for LEF and 9 disease-modifying antirheumatic drugs written between October 1998 and June 2001 at all Veterans Affairs (VA) medical centers were obtained from VA national databases.
RESULTS: LEF was initiated with a loading dose of 100 mg daily for 3 days in 61% of patients, and 42% of patients discontinued LEF. LEF was more likely to be discontinued if a 3-day 100-mg loading dose was prescribed, patients were younger than 44 years or older than 75 years, or reported an annual family income <$60,000. Review of medical records of 291 discontinuers revealed that the most common reasons for discontinuation were inefficacy (30%), gastrointestinal symptoms (29%), medication noncompliance or lost to followup (14%), and elevated liver enzymes (5%).
CONCLUSION: LEF is relatively safe in clinical practice. The VA's national databases provide an excellent, inexpensive resource for postmarketing evaluation of rheumatologic medications.

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Year:  2003        PMID: 14673959     DOI: 10.1002/art.11452

Source DB:  PubMed          Journal:  Arthritis Rheum        ISSN: 0004-3591


  14 in total

1.  Treatment adherence to disease-modifying antirheumatic drugs in patients with rheumatoid arthritis and systemic lupus erythematosus.

Authors:  Sofia de Achaval; Maria E Suarez-Almazor
Journal:  Int J Clin Rheumtol       Date:  2010-06-01

2.  Putting recommendations into practice: Australian rheumatologists' opinions on leflunomide use in rheumatoid arthritis.

Authors:  Ashley M Hopkins; Michael D Wiese; Catherine E O'Doherty; Susanna M Proudman
Journal:  Clin Rheumatol       Date:  2016-11-25       Impact factor: 2.980

3.  Population pharmacokinetics of the active metabolite of leflunomide in pediatric subjects with polyarticular course juvenile rheumatoid arthritis.

Authors:  Jun Shi; Steven J Kovacs; Yaning Wang; Thomas M Ludden; Vijay O Bhargava
Journal:  J Pharmacokinet Pharmacodyn       Date:  2005-08       Impact factor: 2.745

4.  Improving treatment adherence in patients with rheumatologic disease.

Authors:  Sofia de Achaval; Maria E Suarez-Almazor
Journal:  J Musculoskelet Med       Date:  2010-10-12

5.  Clinical effectiveness and safety of leflunomide in inflammatory arthritis: a report from the RAPPORT database with supporting patient survey.

Authors:  Morgan Schultz; Stephanie O Keeling; Steven J Katz; Walter P Maksymowych; Dean T Eurich; Jill J Hall
Journal:  Clin Rheumatol       Date:  2017-05-27       Impact factor: 2.980

6.  Leflunomide in the treatment of rheumatoid arthritis. An analysis of predictors for treatment continuation.

Authors:  E N van Roon; M Hoekstra; H Tobi; T L Th A Jansen; H J Bernelot Moens; J R B J Brouwers; M A F J van de Laar
Journal:  Br J Clin Pharmacol       Date:  2005-09       Impact factor: 4.335

7.  Leflunomide in active rheumatoid arthritis: a prospective study in daily practice.

Authors:  E N Van Roon; T L Th A Jansen; L Mourad; P M Houtman; G A W Bruyn; E N Griep; B Wilffert; H Tobi; J R B J Brouwers
Journal:  Br J Clin Pharmacol       Date:  2004-08       Impact factor: 4.335

8.  Genetic polymorphism of CYP1A2 but not total or free teriflunomide concentrations is associated with leflunomide cessation in rheumatoid arthritis.

Authors:  Ashley M Hopkins; Michael D Wiese; Susanna M Proudman; Catherine E O'Doherty; Richard N Upton; David J R Foster
Journal:  Br J Clin Pharmacol       Date:  2015-10-28       Impact factor: 4.335

9.  Leflunomide in active rheumatoid arthritis: a prospective study in daily practice.

Authors:  E N Van Roon; T L Th A Jansen; L Mourad; P M Houtman; G A W Bruyn; E N Griep; B Wilffert; H Tobi; J R B J Brouwers
Journal:  Br J Clin Pharmacol       Date:  2004-06       Impact factor: 4.335

Review 10.  Benefit-risk assessment of leflunomide: an appraisal of leflunomide in rheumatoid arthritis 10 years after licensing.

Authors:  Nicola Alcorn; Sarah Saunders; Rajan Madhok
Journal:  Drug Saf       Date:  2009       Impact factor: 5.606

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