Literature DB >> 14673950

Messenger RNA levels and enzyme activities of 5 alpha-reductase types 1 and 2 in human benign prostatic hyperplasia (BPH) tissue.

Toshiro Shirakawa1, Hiroshi Okada, Bishnu Acharya, Zhujun Zhang, Nobuyuki Hinata, Yoshitaka Wada, Tatsuya Uji, Sadao Kamidono, Akinobu Gotoh.   

Abstract

BACKGROUND: Benign prostatic hyperplasia (BPH) development requires testicular androgens and aging. The principle prostatic androgen is dihydrotestosterone (DHT). Testosterone is converted to DHT by the enzyme 5 alpha-reductase. Two distinct 5 alpha-reductase enzymes, types 1 and 2, have been identified. While some studies have suggested that type 2 isoenzyme predominates in the prostate, studies on the prostatic localization of the two isoenzymes are controversial. The purpose of this study was to determine the quantitative expressions of 5 alpha-reductase types 1 and 2 in BPH tissues.
METHODS: We examined the localizations of types 1 and 2 isoenzymes in BPH tissues using immunohistochemical staining and a real-time quantitative RT-PCR assay using the TaqMan system. We measured the enzyme activities of types 1 and 2 at pH values of 7.5 and 5.0, respectively.
RESULTS: Our immunohistochemical study showed that type 1 isoenzyme was expressed predominantly in epithelial cells, whereas type 2 isoenzyme was expressed in both stromal and epithelial cells. The real-time RT-PCR assay demonstrated that the copy numbers of type 1 isoenzyme mRNA were significantly higher than those of type 2 isoenzyme mRNA. There were significant associations between enzyme activity at pH 7.5 and type 1 isoenzyme mRNA expression, and between the activity at pH 5.0 and type 2 mRNA expressions.
CONCLUSIONS: We demonstrated that 5 alpha-reductase type 1 had a specific enzyme activity in the prostate, which supports the hypothesis that the type 1 isoenzyme may play a significant role in maintaining prostate enlargement along with the type 2 isoenzyme. Copyright 2003 Wiley-Liss, Inc.

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Year:  2004        PMID: 14673950     DOI: 10.1002/pros.10313

Source DB:  PubMed          Journal:  Prostate        ISSN: 0270-4137            Impact factor:   4.104


  9 in total

Review 1.  Estrogen and androgen signaling in the pathogenesis of BPH.

Authors:  Clement K M Ho; Fouad K Habib
Journal:  Nat Rev Urol       Date:  2011-01       Impact factor: 14.432

2.  In-silico and in-vivo evaluation of sesamol and its derivatives for benign prostatic hypertrophy.

Authors:  Abhishek Shah; Aarti Abhishek Shah; Krishnadas Nandakumar; Avinash Kumar; Aravinda Pai; Richard Lobo
Journal:  3 Biotech       Date:  2021-08-14       Impact factor: 2.406

3.  Androgen receptor and immune inflammation in benign prostatic hyperplasia and prostate cancer.

Authors:  Kouji Izumi; Lei Li; Chawnshang Chang
Journal:  Clin Investig (Lond)       Date:  2014-10-01

Review 4.  Androgen receptor roles in the development of benign prostate hyperplasia.

Authors:  Kouji Izumi; Atsushi Mizokami; Wen-Jye Lin; Kuo-Pao Lai; Chawnshang Chang
Journal:  Am J Pathol       Date:  2013-04-06       Impact factor: 4.307

5.  The 5 alpha-reductase isozyme family: a review of basic biology and their role in human diseases.

Authors:  Faris Azzouni; Alejandro Godoy; Yun Li; James Mohler
Journal:  Adv Urol       Date:  2011-12-25

Review 6.  Differential expression of 5-alpha reductase isozymes in the prostate and its clinical implications.

Authors:  Kai Wang; Dong-Dong Fan; Song Jin; Nian-Zeng Xing; Yi-Nong Niu
Journal:  Asian J Androl       Date:  2014 Mar-Apr       Impact factor: 3.285

7.  5α-reductase 1 mRNA levels are positively correlated with TRAMP mouse prostate most severe lesion scores.

Authors:  Alexander B Opoku-Acheampong; Jamie N Henningson; Amanda P Beck; Brian L Lindshield
Journal:  PLoS One       Date:  2017-05-11       Impact factor: 3.240

8.  Determination of the potency of a novel saw palmetto supercritical CO2 extract (SPSE) for 5α-reductase isoform II inhibition using a cell-free in vitro test system.

Authors:  Pilar Pais; Agustí Villar; Santiago Rull
Journal:  Res Rep Urol       Date:  2016-04-21

9.  The impact of finasteride and dutasteride treatments on proliferation, apoptosis, androgen receptor, 5α-reductase 1 and 5α-reductase 2 in TRAMP mouse prostates.

Authors:  Alexander B Opoku-Acheampong; Jamie N Henningson; Brian L Lindshield
Journal:  Heliyon       Date:  2017-07-24
  9 in total

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