Literature DB >> 14578687

A randomized phase II evaluation of bryostatin-1 (NSC #339555) in recurrent or persistent platinum-sensitive ovarian cancer: a Gynecologic Oncology Group Study.

Deborah K Armstrong1, John A Blessing, Katherine Y Look, Russell Schilder, Evelyn R Nunez.   

Abstract

OBJECTIVES: The Gynecologic Oncology Group (GOG) performed a randomized phase II study to determine the antitumor activity and toxicity of two different schedules of bryostatin-1 administration in patients with recurrent or persistent platinum-sensitive epithelial ovarian cancer or primary peritoneal carcinoma.
METHODS: Eligible patients were randomized to receive either bryostatin-1 25 microg/m2 as a 1h infusion weekly for 3 weeks followed by a 1-week rest (Regimen I) or bryostatin-1 120 microg/m2 as a 72 h continuous infusion every 2 weeks (Regimen II).
RESULTS: Fifty-five patients were enrolled on this study. There was one durable response among 27 eligible patients (response rate=3.7%) on Regimen II and no responses in the 27 eligible patients on Regimen I. Nineteen patients (eleven on Regimen I and eight on Regimen II) had stable disease. The most common adverse event was myalgia, with 12 of 27 patients (44%) on each regimen experiencing some degree of myalgia. There were no other significant toxicities on either treatment arm.
CONCLUSIONS: Both of these schedules and doses of bryostatin-1 are inactive as single agents in previously treated epithelial ovarian cancer.

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Year:  2003        PMID: 14578687     DOI: 10.1023/a:1025490818450

Source DB:  PubMed          Journal:  Invest New Drugs        ISSN: 0167-6997            Impact factor:   3.850


  12 in total

1.  Differential p53-dependent mechanism of radiosensitization in vitro and in vivo by the protein kinase C-specific inhibitor PKC412.

Authors:  K Zaugg; S Rocha; H Resch; I Hegyi; C Oehler; C Glanzmann; D Fabbro; S Bodis; M Pruschy
Journal:  Cancer Res       Date:  2001-01-15       Impact factor: 12.701

2.  Sensitization of human cervical carcinoma cells to cis-diamminedichloroplatinum(II) by bryostatin 1.

Authors:  A Basu; J S Lazo
Journal:  Cancer Res       Date:  1992-06-01       Impact factor: 12.701

3.  The addition of bryostatin 1 to cyclophosphamide, doxorubicin, vincristine, and prednisone (CHOP) chemotherapy improves response in a CHOP-resistant human diffuse large cell lymphoma xenograft model.

Authors:  R M Mohammad; N R Wall; J A Dutcher; A M Al-Katib
Journal:  Clin Cancer Res       Date:  2000-12       Impact factor: 12.531

4.  The in vivo effect of bryostatin-1 on paclitaxel-induced tumor growth, mitotic entry, and blood flow.

Authors:  J A Koutcher; M Motwani; K L Zakian; X K Li; C Matei; J P Dyke; D Ballon; H H Yoo; G K Schwartz
Journal:  Clin Cancer Res       Date:  2000-04       Impact factor: 12.531

5.  Pharmacology and clinical experience with bryostatin 1: a novel anticancer drug.

Authors: 
Journal:  Expert Opin Investig Drugs       Date:  1999-12       Impact factor: 6.206

Review 6.  Protein kinase C isozymes, novel phorbol ester receptors and cancer chemotherapy.

Authors:  O P Barry; M G Kazanietz
Journal:  Curr Pharm Des       Date:  2001-11       Impact factor: 3.116

Review 7.  Chemistry and clinical biology of the bryostatins.

Authors:  R Mutter; M Wills
Journal:  Bioorg Med Chem       Date:  2000-08       Impact factor: 3.641

8.  Bryostatin 1 enhances paclitaxel-induced mitochondrial dysfunction and apoptosis in human leukemia cells (U937) ectopically expressing Bcl-xL.

Authors:  S Wang; Z Wang; L H Boise; P Dent; S Grant
Journal:  Leukemia       Date:  1999-10       Impact factor: 11.528

9.  Cyclophosphamide and cisplatin compared with paclitaxel and cisplatin in patients with stage III and stage IV ovarian cancer.

Authors:  W P McGuire; W J Hoskins; M F Brady; P R Kucera; E E Partridge; K Y Look; D L Clarke-Pearson; M Davidson
Journal:  N Engl J Med       Date:  1996-01-04       Impact factor: 91.245

10.  A phase I study of intravenous bryostatin 1 in patients with advanced cancer.

Authors:  J Prendiville; D Crowther; N Thatcher; P J Woll; B W Fox; A McGown; N Testa; P Stern; R McDermott; M Potter
Journal:  Br J Cancer       Date:  1993-08       Impact factor: 7.640

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  2 in total

1.  A Gynecologic Oncology Group phase II trial of the protein kinase C-beta inhibitor, enzastaurin and evaluation of markers with potential predictive and prognostic value in persistent or recurrent epithelial ovarian and primary peritoneal malignancies.

Authors:  Lydia Usha; Michael W Sill; Kathleen M Darcy; Doris M Benbrook; Jean A Hurteau; David P Michelin; Robert S Mannel; Parviz Hanjani; Koen De Geest; Andrew K Godwin
Journal:  Gynecol Oncol       Date:  2011-03-17       Impact factor: 5.482

Review 2.  Marine-derived angiogenesis inhibitors for cancer therapy.

Authors:  Ying-Qing Wang; Ze-Hong Miao
Journal:  Mar Drugs       Date:  2013-03-15       Impact factor: 5.118

  2 in total

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